ES2291017T3 - Efectos inotropicos y diureticos de la exendina y glp-1. - Google Patents
Efectos inotropicos y diureticos de la exendina y glp-1. Download PDFInfo
- Publication number
- ES2291017T3 ES2291017T3 ES99906762T ES99906762T ES2291017T3 ES 2291017 T3 ES2291017 T3 ES 2291017T3 ES 99906762 T ES99906762 T ES 99906762T ES 99906762 T ES99906762 T ES 99906762T ES 2291017 T3 ES2291017 T3 ES 2291017T3
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- Spain
- Prior art keywords
- xaa
- solvent
- ala
- peptide
- glp
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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Classifications
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
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- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A—HUMAN NECESSITIES
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- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
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- Life Sciences & Earth Sciences (AREA)
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- Gastroenterology & Hepatology (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
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| US7512298P | 1998-02-13 | 1998-02-13 | |
| US75122P | 1998-02-13 |
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| ES2291017T3 true ES2291017T3 (es) | 2008-02-16 |
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| ES99906762T Expired - Lifetime ES2291017T3 (es) | 1998-02-13 | 1999-02-05 | Efectos inotropicos y diureticos de la exendina y glp-1. |
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|---|---|
| EP (1) | EP1054594B1 (https=) |
| JP (1) | JP4677095B2 (https=) |
| AT (1) | ATE366115T1 (https=) |
| AU (1) | AU759058C (https=) |
| CA (1) | CA2320371C (https=) |
| DE (1) | DE69936446T2 (https=) |
| ES (1) | ES2291017T3 (https=) |
| WO (1) | WO1999040788A1 (https=) |
Families Citing this family (102)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2686899B1 (fr) | 1992-01-31 | 1995-09-01 | Rhone Poulenc Rorer Sa | Nouveaux polypeptides biologiquement actifs, leur preparation et compositions pharmaceutiques les contenant. |
| US6852690B1 (en) | 1995-08-22 | 2005-02-08 | Amylin Pharmaceuticals, Inc. | Method and composition for enhanced parenteral nutrition |
| ES2278589T3 (es) | 1999-01-14 | 2007-08-16 | Amylin Pharmaceuticals, Inc. | Excendinas destinadas a la inhibicion de glucagon. |
| US7399489B2 (en) | 1999-01-14 | 2008-07-15 | Amylin Pharmaceuticals, Inc. | Exendin analog formulations |
| US6902744B1 (en) | 1999-01-14 | 2005-06-07 | Amylin Pharmaceuticals, Inc. | Exendin agonist formulations and methods of administration thereof |
| US6506724B1 (en) | 1999-06-01 | 2003-01-14 | Amylin Pharmaceuticals, Inc. | Use of exendins and agonists thereof for the treatment of gestational diabetes mellitus |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5424286A (en) * | 1993-05-24 | 1995-06-13 | Eng; John | Exendin-3 and exendin-4 polypeptides, and pharmaceutical compositions comprising same |
| US5512549A (en) * | 1994-10-18 | 1996-04-30 | Eli Lilly And Company | Glucagon-like insulinotropic peptide analogs, compositions, and methods of use |
| ATE493998T1 (de) * | 1996-08-08 | 2011-01-15 | Amylin Pharmaceuticals Inc | Pharmazeutische zusammensetzung mit einem exendin-4-peptid |
| ES2293688T5 (es) * | 1997-08-08 | 2011-05-04 | Amylin Pharmaceuticals, Inc. | Nuevos compuestos análogos de la exendina. |
-
1999
- 1999-02-05 EP EP99906762A patent/EP1054594B1/en not_active Expired - Lifetime
- 1999-02-05 WO PCT/US1999/002554 patent/WO1999040788A1/en not_active Ceased
- 1999-02-05 JP JP2000531064A patent/JP4677095B2/ja not_active Expired - Fee Related
- 1999-02-05 DE DE69936446T patent/DE69936446T2/de not_active Expired - Lifetime
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- 1999-02-05 AT AT99906762T patent/ATE366115T1/de not_active IP Right Cessation
- 1999-02-05 ES ES99906762T patent/ES2291017T3/es not_active Expired - Lifetime
- 1999-02-05 CA CA2320371A patent/CA2320371C/en not_active Expired - Fee Related
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| ATE366115T1 (de) | 2007-07-15 |
| JP4677095B2 (ja) | 2011-04-27 |
| EP1054594B1 (en) | 2007-07-04 |
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| DE69936446T2 (de) | 2008-03-06 |
| CA2320371C (en) | 2012-01-17 |
| DE69936446D1 (de) | 2007-08-16 |
| JP2002509078A (ja) | 2002-03-26 |
| WO1999040788A1 (en) | 1999-08-19 |
| EP1054594A4 (en) | 2002-04-17 |
| EP1054594A1 (en) | 2000-11-29 |
| AU759058C (en) | 2005-09-15 |
| AU2659699A (en) | 1999-08-30 |
| AU759058B2 (en) | 2003-04-03 |
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