ES2019243A6 - Procedimiento para preparar nuevos derivados de tieno-triazolo-diazepina. - Google Patents
Procedimiento para preparar nuevos derivados de tieno-triazolo-diazepina.Info
- Publication number
- ES2019243A6 ES2019243A6 ES9000912A ES9000912A ES2019243A6 ES 2019243 A6 ES2019243 A6 ES 2019243A6 ES 9000912 A ES9000912 A ES 9000912A ES 9000912 A ES9000912 A ES 9000912A ES 2019243 A6 ES2019243 A6 ES 2019243A6
- Authority
- ES
- Spain
- Prior art keywords
- thieno
- triazolo
- compositions containing
- therapeutic compositions
- diazepine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 239000000203 mixture Substances 0.000 title abstract 3
- 230000001225 therapeutic effect Effects 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 4
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- 239000005864 Sulphur Substances 0.000 abstract 2
- 230000003266 anti-allergic effect Effects 0.000 abstract 2
- 230000001088 anti-asthma Effects 0.000 abstract 2
- 239000000924 antiasthmatic agent Substances 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 230000002496 gastric effect Effects 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 238000002360 preparation method Methods 0.000 abstract 2
- 230000001012 protector Effects 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR NUEVOS DERIVADOS DE TIENO-TRIAZOLO-DIZEPINA DE FORMULA FORMULA EN DONDE <Y> REPRESENTA OXIGENO O AZUFRE Y <R> REPRESENTA DIVERSOS SUSTITUYENTES, QUE CONSISTE EN HACER REACCIONAR BAJO CIRCULACION DE NITROGENO, UN EXCESO DE UN COMPUESTO DE TIENO-TRIAZONOLO-DIAZEPINA DE FORMULA II DADA EN LA MEMORIA DESCRIPTIVA, CON EL APROPIADO DERIVADO DE R - N = C = Y EN DONDE <R> E <Y> SON COMO ANTES SE DEFINEN, EN EL SENO DE UN DISOLVENTE APROTICO Y A UNA TEMPERATURA COMPRENDIDA ENTRE LA TEMPERATURA Y APROXIMADAMENTE 70GC.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB898907256A GB8907256D0 (en) | 1989-03-31 | 1989-03-31 | New derivatives of hetrazepine as anti-asthmatic anti-allergic and gastro-intestinal protectors |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2019243A6 true ES2019243A6 (es) | 1991-06-01 |
Family
ID=10654231
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES9000912A Expired - Fee Related ES2019243A6 (es) | 1989-03-31 | 1990-03-30 | Procedimiento para preparar nuevos derivados de tieno-triazolo-diazepina. |
Country Status (30)
Country | Link |
---|---|
US (1) | US5492906A (es) |
JP (1) | JPH07103127B2 (es) |
KR (1) | KR900014396A (es) |
AT (1) | AT394561B (es) |
AU (1) | AU622007B2 (es) |
BE (1) | BE1003699A3 (es) |
CA (1) | CA2013518C (es) |
CH (1) | CH680365A5 (es) |
DE (1) | DE4010316C2 (es) |
DK (1) | DK80890A (es) |
ES (1) | ES2019243A6 (es) |
FI (1) | FI95036C (es) |
FR (2) | FR2645022B1 (es) |
GB (2) | GB8907256D0 (es) |
GR (1) | GR1000394B (es) |
HK (1) | HK95192A (es) |
IE (1) | IE64564B1 (es) |
IN (1) | IN174015B (es) |
IT (1) | IT1240350B (es) |
LU (1) | LU87710A1 (es) |
MA (1) | MA21790A1 (es) |
MY (1) | MY105538A (es) |
NL (1) | NL194827C (es) |
NO (1) | NO173784C (es) |
NZ (1) | NZ233011A (es) |
OA (1) | OA09442A (es) |
PT (1) | PT93629B (es) |
SE (1) | SE505417C2 (es) |
TN (1) | TNSN90042A1 (es) |
ZA (1) | ZA901765B (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PH30676A (en) * | 1986-07-22 | 1997-09-16 | Boehringer Ingelhein Kg | Hetrazepine compounds which have useful pharmaceutical utility |
US5382579A (en) * | 1988-10-31 | 1995-01-17 | Eisai Co., Ltd. | Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals |
US5304553A (en) * | 1988-10-31 | 1994-04-19 | Eisai Co., Ltd. | 1,4-diazepine derivative and its pharmaceutical use |
US5221671A (en) * | 1988-10-31 | 1993-06-22 | Eisai Co., Ltd. | Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals |
DE4027470A1 (de) * | 1990-08-30 | 1992-03-05 | Boehringer Ingelheim Kg | Neue hetrazepinoide amide |
ES2061406B1 (es) * | 1993-05-07 | 1995-06-01 | Uriach & Cia Sa J | Nuevos derivados de la 2-(quinolina) con actividad farmacologica. |
FI101989B (fi) * | 1996-11-22 | 1998-09-30 | Stora Enso Oyj | Menetelmät neste- ja kaasutiiviin pakkauskartongin sekä pakkauksen val mistamiseksi sekä menetelmien mukaisesti valmistetut tuotteet |
WO1998058930A1 (fr) * | 1997-06-25 | 1998-12-30 | Nikken Chemicals Co., Ltd. | Composes de triazolo-1,4-diazepine et composition medicinale les contenant |
FR2779652B1 (fr) * | 1998-06-15 | 2001-06-08 | Sod Conseils Rech Applic | Utilisation de diazepines pour la preparation de medicaments destines a traiter les etats pathologiques ou les maladies dans lesquels un des recepteurs de la somatostatine est implique |
US6987105B2 (en) * | 2000-04-28 | 2006-01-17 | Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College | Synthesis and use of thienotriazolodiazepines |
KR20110117731A (ko) * | 2003-05-30 | 2011-10-27 | 랜박시 래보러터리스 리미티드 | 치환된 피롤 유도체와 hmg―co 억제제로서의 이의 용도 |
AU2006313430B2 (en) * | 2005-11-08 | 2012-09-06 | Ranbaxy Laboratories Limited | Process for (3R,5R)-7-[2-(4-fluorophenyl)-5-isopropyl-3-phenyl-4- [(4-hydroxy methyl phenyl amino) carbonyl]-pyrrol-1-yl]-3, 5-dihydroxy-heptanoic acid hemi calcium salt |
WO2008020314A2 (en) * | 2006-03-14 | 2008-02-21 | Ranbaxy Laboratories Limited | Statin stabilizing dosage formulations |
WO2008010087A2 (en) * | 2006-07-14 | 2008-01-24 | Ranbaxy Laboratories Limited | Polymorphic forms of an hmg-coa reductase inhibitor and uses thereof |
KR101675984B1 (ko) * | 2015-02-23 | 2016-11-14 | 한양대학교 에리카산학협력단 | 티에노디아제핀 유도체 또는 이의 약학적으로 허용가능한 염, 및 이를 유효성분으로 포함하는 약학적 조성물 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PH30676A (en) * | 1986-07-22 | 1997-09-16 | Boehringer Ingelhein Kg | Hetrazepine compounds which have useful pharmaceutical utility |
WO1988009792A1 (en) * | 1987-06-08 | 1988-12-15 | Yoshitomi Pharmaceutical Industries, Ltd. | Ester-substituted thienotriazolodiazepine compounds and their medicinal use |
FI95708C (fi) * | 1988-10-31 | 1996-03-11 | Eisai Co Ltd | Analogiamenetelmä 1,4-diatsepiinijohdannaisen ja sen farmaseuttisesti sopivan suolan valmistamiseksi |
NL9000627A (nl) * | 1990-03-29 | 1991-10-16 | Scras | Werkwijze ter bereiding van nieuwe thienotriazolo-diazepines. |
-
1989
- 1989-03-31 GB GB898907256A patent/GB8907256D0/en active Pending
-
1990
- 1990-03-07 ZA ZA901765A patent/ZA901765B/xx unknown
- 1990-03-07 NO NO901070A patent/NO173784C/no not_active IP Right Cessation
- 1990-03-07 IN IN220DE1990 patent/IN174015B/en unknown
- 1990-03-07 IE IE80690A patent/IE64564B1/en not_active IP Right Cessation
- 1990-03-08 GR GR900100165A patent/GR1000394B/el not_active IP Right Cessation
- 1990-03-09 AT AT0056790A patent/AT394561B/de not_active IP Right Cessation
- 1990-03-12 SE SE9000871A patent/SE505417C2/sv not_active IP Right Cessation
- 1990-03-19 NL NL9000626A patent/NL194827C/nl not_active IP Right Cessation
- 1990-03-21 NZ NZ233011A patent/NZ233011A/xx unknown
- 1990-03-26 JP JP2073582A patent/JPH07103127B2/ja not_active Expired - Lifetime
- 1990-03-27 BE BE9000343A patent/BE1003699A3/fr not_active IP Right Cessation
- 1990-03-29 CH CH1044/90A patent/CH680365A5/fr not_active IP Right Cessation
- 1990-03-29 GB GB9007000A patent/GB2229723B/en not_active Expired - Fee Related
- 1990-03-29 LU LU87710A patent/LU87710A1/fr unknown
- 1990-03-30 OA OA59759A patent/OA09442A/xx unknown
- 1990-03-30 AU AU52425/90A patent/AU622007B2/en not_active Ceased
- 1990-03-30 KR KR1019900004522A patent/KR900014396A/ko active IP Right Grant
- 1990-03-30 PT PT93629A patent/PT93629B/pt active IP Right Grant
- 1990-03-30 FI FI901605A patent/FI95036C/fi not_active IP Right Cessation
- 1990-03-30 TN TNTNSN90042A patent/TNSN90042A1/fr unknown
- 1990-03-30 DK DK080890A patent/DK80890A/da not_active Application Discontinuation
- 1990-03-30 IT IT19884A patent/IT1240350B/it active IP Right Grant
- 1990-03-30 MA MA22056A patent/MA21790A1/fr unknown
- 1990-03-30 DE DE4010316A patent/DE4010316C2/de not_active Expired - Fee Related
- 1990-03-30 CA CA002013518A patent/CA2013518C/en not_active Expired - Fee Related
- 1990-03-30 MY MYPI90000509A patent/MY105538A/en unknown
- 1990-03-30 ES ES9000912A patent/ES2019243A6/es not_active Expired - Fee Related
- 1990-04-02 FR FR909004155A patent/FR2645022B1/fr not_active Expired - Fee Related
- 1990-04-02 FR FR909004156A patent/FR2645153B1/fr not_active Expired - Fee Related
-
1992
- 1992-02-18 US US07/837,580 patent/US5492906A/en not_active Expired - Lifetime
- 1992-11-26 HK HK951/92A patent/HK95192A/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 20050331 |