EG18184A - Process for preparing of substituted bridged diazabicyclo-alkyl quinoline carboxylic acid - Google Patents

Process for preparing of substituted bridged diazabicyclo-alkyl quinoline carboxylic acid

Info

Publication number
EG18184A
EG18184A EG580/86A EG58086A EG18184A EG 18184 A EG18184 A EG 18184A EG 580/86 A EG580/86 A EG 580/86A EG 58086 A EG58086 A EG 58086A EG 18184 A EG18184 A EG 18184A
Authority
EG
Egypt
Prior art keywords
diazabicyclo
preparing
carboxylic acid
quinoline carboxylic
alkyl
Prior art date
Application number
EG580/86A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of EG18184A publication Critical patent/EG18184A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Materials For Photolithography (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
EG580/86A 1985-09-18 1986-09-15 Process for preparing of substituted bridged diazabicyclo-alkyl quinoline carboxylic acid EG18184A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77747185A 1985-09-18 1985-09-18

Publications (1)

Publication Number Publication Date
EG18184A true EG18184A (en) 1992-12-30

Family

ID=25110350

Family Applications (1)

Application Number Title Priority Date Filing Date
EG580/86A EG18184A (en) 1985-09-18 1986-09-15 Process for preparing of substituted bridged diazabicyclo-alkyl quinoline carboxylic acid

Country Status (42)

Country Link
US (3) US4861779A (sv)
EP (1) EP0215650B1 (sv)
JP (1) JPH0798819B2 (sv)
KR (1) KR870000961B1 (sv)
CN (1) CN1014789B (sv)
AT (1) ATE72245T1 (sv)
AU (1) AU576302B2 (sv)
BG (2) BG49275A3 (sv)
CA (1) CA1340734C (sv)
CY (1) CY1774A (sv)
CZ (1) CZ277825B6 (sv)
DD (1) DD259190A5 (sv)
DE (2) DE19675019I2 (sv)
DK (1) DK171276B1 (sv)
EG (1) EG18184A (sv)
ES (1) ES2001428A6 (sv)
FI (1) FI87565C (sv)
GR (1) GR862363B (sv)
HK (1) HK132795A (sv)
HU (1) HU200462B (sv)
IE (1) IE58966B1 (sv)
IL (1) IL80033A (sv)
IN (1) IN166416B (sv)
LU (1) LU90356I2 (sv)
MA (1) MA20770A1 (sv)
MW (1) MW5886A1 (sv)
MX (1) MX173358B (sv)
MY (1) MY102518A (sv)
NO (1) NO170335C (sv)
NZ (1) NZ217614A (sv)
OA (1) OA08410A (sv)
PH (2) PH24048A (sv)
PL (1) PL149987B1 (sv)
PT (1) PT83388B (sv)
SG (1) SG28094G (sv)
SK (1) SK667886A3 (sv)
SU (1) SU1482531A3 (sv)
UA (1) UA6340A1 (sv)
YU (1) YU45024B (sv)
ZA (1) ZA867063B (sv)
ZM (1) ZM8586A1 (sv)
ZW (1) ZW19386A1 (sv)

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US4992546A (en) * 1987-07-31 1991-02-12 Warner-Lambert Company Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives
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DE3902079A1 (de) * 1988-04-15 1989-10-26 Bayer Ag I.m. injektionsformen von gyrase-inhibitoren
WO1990002123A1 (en) * 1988-08-23 1990-03-08 Pfizer Inc. Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
US5147873A (en) * 1988-08-23 1992-09-15 Pfizer Inc. Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
US4895943A (en) * 1988-10-25 1990-01-23 Pfizer Inc. Preparation of 1,4-diazabicyclo(3.2.2)nonane
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US5235054A (en) * 1992-07-15 1993-08-10 Pfizer Inc. 3-carboxaldehyde substituted quinolines and naphthyridines
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US5929086A (en) 1996-05-10 1999-07-27 Pharmacia & Upjohn Company Topical administration of antimicrobial agents for the treatment of systemic bacterial diseases
US6056436A (en) * 1997-02-20 2000-05-02 University Of Maryland Simultaneous measurement of temperature and strain using optical sensors
CN1210277C (zh) 1999-05-04 2005-07-13 神经研究公司 杂芳基二氮杂双环烷烃及其制备方法和应用
FR2809730B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo[3.2.2] nonanebenzoxazole, -benzothiazole et -benzimidazole, leur preparation et leur application therapeutique
FR2809731B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo-[3.2.2] nonane-pheylisoxazole, leur preparation et leur application en therapeutique
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JP2006504690A (ja) * 2002-09-10 2006-02-09 ファイザー・プロダクツ・インク Cns及びその他の障害の治療に有用なジアザ二環式化合物
JP4890762B2 (ja) 2002-09-25 2012-03-07 メモリー・ファーマシューティカルズ・コーポレイション インダゾール、ベンゾチアゾール、及びベンゾイソチアゾール、並びにそれらの調製及び使用
DE10312346A1 (de) * 2003-03-20 2004-09-30 Bayer Healthcare Ag Kontrolliertes Freisetzungssystem
DE10351448A1 (de) 2003-11-04 2005-06-09 Bayer Healthcare Ag Geschmackstoffhaltige Arzneimittelformulierungen mit verbesserten pharmazeutischen Eigenschaften
DE602004010299T2 (de) 2003-12-22 2008-09-18 Memory Pharmaceuticals Corp. Indole, 1h-indazole, 1,2-benzisoxazole und 1,2-benzisothiazole und deren herstellung und anwendungen
CN103724343A (zh) * 2004-03-25 2014-04-16 记忆药物公司 吲唑、苯并噻唑、苯并异噻唑、苯并异噁唑及其制备和用途
WO2006001894A1 (en) * 2004-04-22 2006-01-05 Memory Pharmaceutical Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof
BRPI0510212A (pt) * 2004-05-07 2007-10-16 Memory Pharm Corp 1h-indazóis, benzotiazóis, 1,2 - benzoisoxazóis, 1,2-benzoisotiazóis, e cromonas e a preparação e usos dos mesmos
DE102005055385A1 (de) * 2004-12-09 2006-06-14 Bayer Healthcare Ag Arzneimittel zur hygienischen Applikation im Ohr
MX2007007328A (es) 2004-12-22 2007-07-25 Memory Pharm Corp Ligandos del receptor alfa-7 nicotinico y preparacion y sus usos.
US8106066B2 (en) * 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
CA2641685A1 (en) 2006-02-10 2007-08-16 Neurosearch A/S 3-heteroaryl-3,9-diazabicyclo[3.3.1]nonane derivatives as nicotinic acetylcholine receptor agonists
WO2007090886A1 (en) * 2006-02-10 2007-08-16 Neurosearch A/S 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
CA2641683A1 (en) 2006-02-10 2007-08-16 Neurosearch A/S 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
DE102006010643A1 (de) 2006-03-08 2007-09-13 Bayer Healthcare Aktiengesellschaft Arzneimittel enthaltend Fluorchinolone
DE102006010642A1 (de) * 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
DE102007026550A1 (de) * 2007-06-08 2008-12-11 Bayer Healthcare Ag Extrudate mit verbesserter Geschmacksmaskierung
DE102007055341A1 (de) * 2007-11-19 2009-05-20 Bayer Animal Health Gmbh Stabilisierung öliger Suspensionen enthaltend hydrophobe Kieselsäuren
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MX2011009414A (es) * 2009-03-11 2011-10-19 Kyorin Seiyaku Kk 7-cicloalquiloaminoquinolonas como inhibidores de gsk-3.
CN103200930A (zh) 2010-10-12 2013-07-10 拜耳知识产权有限责任公司 非淀粉基软咀嚼品
KR102253847B1 (ko) 2012-12-19 2021-05-21 바이엘 애니멀 헬스 게엠베하 향상된 수용성 및 우수한 저장 안정성을 가지는 정제
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DE3641312A1 (de) * 1986-12-03 1988-06-09 Bayer Ag Verfahren zur herstellung von chinolincarbonsaeuren
US4923879A (en) * 1987-07-31 1990-05-08 Warner-Lambert Company 1,8-Naphthyridines and their use as antibacterial agents
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent

Also Published As

Publication number Publication date
YU161786A (en) 1987-10-31
FI863756A0 (fi) 1986-09-17
EP0215650A2 (en) 1987-03-25
NO863718L (no) 1987-03-19
PH24048A (en) 1990-03-05
JPH0798819B2 (ja) 1995-10-25
LU90356I2 (fr) 1999-04-26
IE862479L (en) 1987-03-18
HU200462B (en) 1990-06-28
KR870003106A (ko) 1987-04-15
CZ277825B6 (en) 1993-06-16
ATE72245T1 (de) 1992-02-15
IN166416B (sv) 1990-05-05
DK445886D0 (da) 1986-09-17
DE3683711D1 (de) 1992-03-12
CZ667886A3 (en) 1993-02-17
BG61091B2 (bg) 1996-10-31
YU45024B (en) 1991-06-30
MX3751A (es) 1993-09-01
PL149987B1 (en) 1990-04-30
FI87565C (sv) 1993-01-25
ZW19386A1 (en) 1986-12-10
PL261410A1 (en) 1987-11-16
CN1014789B (zh) 1991-11-20
MX173358B (es) 1994-02-23
US4775668A (en) 1988-10-04
JPS62103083A (ja) 1987-05-13
IL80033A0 (en) 1986-12-31
OA08410A (fr) 1988-06-30
DK445886A (da) 1987-05-27
PT83388B (pt) 1989-05-12
IL80033A (en) 1992-05-25
PT83388A (en) 1986-10-01
ZA867063B (en) 1988-04-27
DD259190A5 (de) 1988-08-17
HK132795A (en) 1995-09-01
IE58966B1 (en) 1993-12-01
MY102518A (en) 1992-07-31
CA1340734C (en) 1999-09-14
FI863756A (fi) 1987-03-19
EP0215650A3 (en) 1987-12-02
MA20770A1 (fr) 1987-04-01
NO170335B (no) 1992-06-29
SK278605B6 (en) 1997-11-05
SU1482531A3 (ru) 1989-05-23
ZM8586A1 (en) 1987-03-27
CY1774A (en) 1995-10-20
SG28094G (en) 1994-10-28
NZ217614A (en) 1989-11-28
BG49275A3 (en) 1991-09-16
NO170335C (no) 1992-10-07
AU576302B2 (en) 1988-08-18
NO863718D0 (no) 1986-09-17
FI87565B (fi) 1992-10-15
UA6340A1 (uk) 1994-12-29
KR870000961B1 (ko) 1987-05-14
AU6276886A (en) 1987-03-19
PH25338A (en) 1991-04-30
DK171276B1 (da) 1996-08-19
MW5886A1 (en) 1987-12-09
EP0215650B1 (en) 1992-01-29
GR862363B (en) 1987-01-19
DE19675019I2 (de) 2004-01-29
SK667886A3 (en) 1997-11-05
US5091383A (en) 1992-02-25
US4861779A (en) 1989-08-29
CN86106385A (zh) 1987-06-03
HUT43070A (en) 1987-09-28
ES2001428A6 (es) 1988-05-16

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