ECSP18094790A - Piridinas sustituidas con heteroarilo y métodos de uso referencia cruzada a solicitudes relacionadas - Google Patents

Piridinas sustituidas con heteroarilo y métodos de uso referencia cruzada a solicitudes relacionadas

Info

Publication number
ECSP18094790A
ECSP18094790A ECSENADI201894790A ECDI201894790A ECSP18094790A EC SP18094790 A ECSP18094790 A EC SP18094790A EC SENADI201894790 A ECSENADI201894790 A EC SENADI201894790A EC DI201894790 A ECDI201894790 A EC DI201894790A EC SP18094790 A ECSP18094790 A EC SP18094790A
Authority
EC
Ecuador
Prior art keywords
methods
heteroaryl
cross reference
use cross
related requests
Prior art date
Application number
ECSENADI201894790A
Other languages
English (en)
Spanish (es)
Inventor
Andrew Bogdan
Stephen N Greszler
Xueqing Wang
Ghjuvanni Petru Diunisu Coti
Robert Altenbach
Marlon Cowart
Der Plas Steven Emiel Van
Hans Kelgtermans
Philip Kym
Original Assignee
Galapagos Nv
Abbvie Sarl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Galapagos Nv, Abbvie Sarl filed Critical Galapagos Nv
Publication of ECSP18094790A publication Critical patent/ECSP18094790A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ECSENADI201894790A 2016-06-03 2018-12-26 Piridinas sustituidas con heteroarilo y métodos de uso referencia cruzada a solicitudes relacionadas ECSP18094790A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662345315P 2016-06-03 2016-06-03

Publications (1)

Publication Number Publication Date
ECSP18094790A true ECSP18094790A (es) 2019-01-31

Family

ID=59014678

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSENADI201894790A ECSP18094790A (es) 2016-06-03 2018-12-26 Piridinas sustituidas con heteroarilo y métodos de uso referencia cruzada a solicitudes relacionadas

Country Status (35)

Country Link
US (2) US10138227B2 (enExample)
EP (1) EP3464282B1 (enExample)
JP (3) JP6968094B2 (enExample)
KR (2) KR102719916B1 (enExample)
CN (2) CN114671864B (enExample)
AR (2) AR108672A1 (enExample)
AU (3) AU2017273215B2 (enExample)
CA (1) CA3022216A1 (enExample)
CL (1) CL2018003323A1 (enExample)
CO (1) CO2018012171A2 (enExample)
CR (1) CR20180547A (enExample)
CY (1) CY1124031T1 (enExample)
DK (1) DK3464282T3 (enExample)
DO (1) DOP2018000257A (enExample)
EC (1) ECSP18094790A (enExample)
ES (1) ES2806873T3 (enExample)
HR (1) HRP20201068T1 (enExample)
HU (1) HUE050248T2 (enExample)
IL (3) IL303196B2 (enExample)
LT (1) LT3464282T (enExample)
MX (2) MX385054B (enExample)
MY (1) MY199604A (enExample)
PE (1) PE20190511A1 (enExample)
PH (1) PH12018502534B1 (enExample)
PL (1) PL3464282T3 (enExample)
PT (1) PT3464282T (enExample)
RS (1) RS60574B1 (enExample)
RU (2) RU2021127810A (enExample)
SG (1) SG11201808842VA (enExample)
SI (1) SI3464282T1 (enExample)
SM (1) SMT202000394T1 (enExample)
TW (4) TW202515560A (enExample)
UY (2) UY40612A (enExample)
WO (1) WO2017208115A1 (enExample)
ZA (1) ZA201808423B (enExample)

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HUE050248T2 (hu) 2020-12-28
CN114671864B (zh) 2025-04-08
NZ788542A (en) 2025-06-27
TWI797926B (zh) 2023-04-01
CN109311864A (zh) 2019-02-05
KR102719916B1 (ko) 2024-10-23
ES2806873T3 (es) 2021-02-18
IL262415B (en) 2021-12-01
AU2017273215A1 (en) 2018-10-25
DK3464282T3 (da) 2020-07-27
IL303196A (en) 2023-07-01
JP2023172889A (ja) 2023-12-06
HRP20201068T1 (hr) 2020-11-13
IL303196B2 (en) 2025-04-01
SI3464282T1 (sl) 2020-12-31
JP7622122B2 (ja) 2025-01-27
UY40612A (es) 2024-02-15
CN114671864A (zh) 2022-06-28
JP6968094B2 (ja) 2021-11-17
MX385054B (es) 2025-03-14
MX2018014758A (es) 2019-04-29
RU2018138707A3 (enExample) 2020-08-24
EP3464282B1 (en) 2020-04-22
TW202515560A (zh) 2025-04-16
KR20220162806A (ko) 2022-12-08
TW201802085A (zh) 2018-01-16
MY199604A (en) 2023-11-08
TWI752961B (zh) 2022-01-21
IL303196B1 (en) 2024-12-01
RS60574B1 (sr) 2020-08-31
AR108672A1 (es) 2018-09-12
AU2024202468A1 (en) 2024-05-02
AU2017273215B2 (en) 2021-09-09
AR124916A2 (es) 2023-05-17
US20170349576A1 (en) 2017-12-07
TW202329959A (zh) 2023-08-01
AU2021282409B2 (en) 2024-01-18
KR102469995B1 (ko) 2022-11-24
SG11201808842VA (en) 2018-11-29
AU2021282409A1 (en) 2021-12-23
MX2021009322A (es) 2021-09-08
NZ747222A (en) 2025-06-27
RU2021127810A (ru) 2021-10-25
CO2018012171A2 (es) 2018-11-30
JP2022009448A (ja) 2022-01-14
IL288243B1 (en) 2023-07-01
LT3464282T (lt) 2020-09-10
CY1124031T1 (el) 2022-03-24
RU2018138707A (ru) 2020-07-14
PL3464282T3 (pl) 2020-12-14
PE20190511A1 (es) 2019-04-10
IL288243A (en) 2022-01-01
TW202214614A (zh) 2022-04-16
CR20180547A (es) 2019-10-30
WO2017208115A1 (en) 2017-12-07
CL2018003323A1 (es) 2019-03-22
IL262415A (en) 2018-12-31
PT3464282T (pt) 2020-07-17
IL288243B2 (en) 2023-11-01
JP2019517455A (ja) 2019-06-24
ZA201808423B (en) 2019-08-28
UY37272A (es) 2018-01-02
SMT202000394T1 (it) 2020-09-10
PH12018502534A1 (en) 2019-10-21
KR20190015215A (ko) 2019-02-13
JP7392211B2 (ja) 2023-12-06
EP3464282A1 (en) 2019-04-10
TWI849782B (zh) 2024-07-21
US10604515B2 (en) 2020-03-31
RU2756743C2 (ru) 2021-10-05
PH12018502534B1 (en) 2020-09-23
US10138227B2 (en) 2018-11-27
CN109311864B (zh) 2022-05-10
US20190055229A1 (en) 2019-02-21
CA3022216A1 (en) 2017-12-07
BR112018074815A2 (pt) 2019-03-19
DOP2018000257A (es) 2018-12-31

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