ECSP11011327A - Derivados de aminotetralina, composiciones farmacéuticas que los contienen, y sus usos en terapia - Google Patents

Derivados de aminotetralina, composiciones farmacéuticas que los contienen, y sus usos en terapia

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Publication number
ECSP11011327A
ECSP11011327A EC2011011327A ECSP11011327A ECSP11011327A EC SP11011327 A ECSP11011327 A EC SP11011327A EC 2011011327 A EC2011011327 A EC 2011011327A EC SP11011327 A ECSP11011327 A EC SP11011327A EC SP11011327 A ECSP11011327 A EC SP11011327A
Authority
EC
Ecuador
Prior art keywords
pharmaceutical compositions
therapy
contain
derivatives
aminotetraline derivatives
Prior art date
Application number
EC2011011327A
Other languages
English (en)
Inventor
Charles W Hutchins
Udo Lange
Andreas Kling
Wilfried Hornberger
Mario Mezler
Wilhelm Amberg
Michael Ochse
Berthold Behl
Original Assignee
Abbott Gmbh & Co Kg
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co Kg, Abbott Lab filed Critical Abbott Gmbh & Co Kg
Publication of ECSP11011327A publication Critical patent/ECSP11011327A/es

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    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/05—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by nitrogen atoms, not being part of nitro or nitroso groups
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

Derivados de aminotetralina de la fórmula (I)o una sal fisiológicamente tolerable de los mismos.La invención se relaciona con composiciones farmacéuticas que comprenden dichos derivados de aminotetralina, y el uso de dichos derivados de aminotetralina con propósitos terapéuticos. Los derivados de aminotetralina son inhibidores de GlyT1.
EC2011011327A 2009-02-16 2011-09-14 Derivados de aminotetralina, composiciones farmacéuticas que los contienen, y sus usos en terapia ECSP11011327A (es)

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