ECSP11011081A - 3-aminociclopentancarboxamidas - Google Patents

3-aminociclopentancarboxamidas

Info

Publication number
ECSP11011081A
ECSP11011081A EC2011011081A ECSP11011081A ECSP11011081A EC SP11011081 A ECSP11011081 A EC SP11011081A EC 2011011081 A EC2011011081 A EC 2011011081A EC SP11011081 A ECSP11011081 A EC SP11011081A EC SP11011081 A ECSP11011081 A EC SP11011081A
Authority
EC
Ecuador
Prior art keywords
aminociclopentancarboxamidas
compound
formula
pharmaceutically acceptable
acceptable salt
Prior art date
Application number
EC2011011081A
Other languages
English (en)
Spanish (es)
Inventor
Rajes Devraj
Robert Hughes
Steven Ronald Turner
Wei Huang
Donald Joseph Rogier Jr
John Isidro Trujillo
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ECSP11011081A publication Critical patent/ECSP11011081A/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
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    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
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    • A61P11/06Antiasthmatics
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    • A61P13/12Drugs for disorders of the urinary system of the kidneys
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
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    • A61P3/02Nutrients, e.g. vitamins, minerals
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
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    • AHUMAN NECESSITIES
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
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    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
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    • A61P37/08Antiallergic agents
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    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
  • Nutrition Science (AREA)
  • Hospice & Palliative Care (AREA)
  • Virology (AREA)
  • Ophthalmology & Optometry (AREA)
EC2011011081A 2008-11-26 2011-05-25 3-aminociclopentancarboxamidas ECSP11011081A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26

Publications (1)

Publication Number Publication Date
ECSP11011081A true ECSP11011081A (es) 2011-12-30

Family

ID=41693100

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2011011081A ECSP11011081A (es) 2008-11-26 2011-05-25 3-aminociclopentancarboxamidas

Country Status (38)

Country Link
US (2) US8293903B2 (OSRAM)
EP (1) EP2370442B9 (OSRAM)
JP (1) JP5108153B2 (OSRAM)
KR (1) KR101374412B1 (OSRAM)
CN (1) CN102227429B (OSRAM)
AP (1) AP3113A (OSRAM)
AU (1) AU2009321221B2 (OSRAM)
BR (1) BRPI0920936A2 (OSRAM)
CA (1) CA2743030C (OSRAM)
CL (1) CL2011001223A1 (OSRAM)
CO (1) CO6361921A2 (OSRAM)
CR (1) CR20110275A (OSRAM)
CU (1) CU24022B1 (OSRAM)
CY (1) CY1114020T1 (OSRAM)
DK (1) DK2370442T5 (OSRAM)
DO (1) DOP2011000154A (OSRAM)
EA (1) EA020470B1 (OSRAM)
EC (1) ECSP11011081A (OSRAM)
ES (1) ES2415430T3 (OSRAM)
GE (1) GEP20146064B (OSRAM)
HR (1) HRP20130409T2 (OSRAM)
IL (1) IL212732A (OSRAM)
MA (1) MA32834B1 (OSRAM)
ME (1) ME01144B (OSRAM)
MX (1) MX2011005526A (OSRAM)
MY (1) MY152557A (OSRAM)
NI (1) NI201100102A (OSRAM)
NZ (1) NZ592919A (OSRAM)
PE (1) PE20110831A1 (OSRAM)
PL (1) PL2370442T3 (OSRAM)
PT (1) PT2370442E (OSRAM)
RS (2) RS52810B9 (OSRAM)
SI (1) SI2370442T1 (OSRAM)
SV (1) SV2011003923A (OSRAM)
TN (1) TN2011000254A1 (OSRAM)
UA (1) UA99978C2 (OSRAM)
WO (1) WO2010061329A1 (OSRAM)
ZA (1) ZA201104069B (OSRAM)

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GEP20146064B (en) * 2008-11-26 2014-03-25 Pfizer 3-minocyclopentanecarboxamides as chemokine receptor modulators
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1r,2r,3r)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
SG11201608303QA (en) 2014-04-04 2016-11-29 Del Mar Pharmaceuticals Use of dianhydrogalactitol and analogs or derivatives thereof to treat non-small-cell carcinoma of the lung and ovarian cancer
JP2016029038A (ja) * 2014-07-17 2016-03-03 参天製薬株式会社 加齢黄斑変性の予防または治療剤
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲(江蘇)醫藥有限公司 環戊烷化合物

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HK1161261A1 (en) 2012-08-24
NI201100102A (es) 2011-09-27
CU20110121A7 (es) 2013-05-31
SI2370442T1 (sl) 2013-06-28
DK2370442T3 (da) 2013-06-17
NZ592919A (en) 2013-05-31
KR20110075036A (ko) 2011-07-05
CL2011001223A1 (es) 2011-09-02
PL2370442T3 (pl) 2013-08-30
CN102227429B (zh) 2014-05-28
CR20110275A (es) 2011-07-01
ES2415430T9 (es) 2013-11-25
US20130197008A1 (en) 2013-08-01
BRPI0920936A2 (pt) 2020-08-11
UA99978C2 (en) 2012-10-25
CY1114020T1 (el) 2016-07-27
AU2009321221B2 (en) 2013-04-04
HRP20130409T2 (hr) 2013-11-22
AP3113A (en) 2015-01-31
EP2370442B9 (en) 2013-09-04
TN2011000254A1 (fr) 2012-12-17
MY152557A (en) 2014-10-31
JP2012509931A (ja) 2012-04-26
MX2011005526A (es) 2011-06-06
AP2011005732A0 (en) 2011-06-30
PE20110831A1 (es) 2011-11-20
JP5108153B2 (ja) 2012-12-26
DK2370442T5 (da) 2013-09-23
PT2370442E (pt) 2013-06-27
CN102227429A (zh) 2011-10-26
EP2370442A1 (en) 2011-10-05
WO2010061329A1 (en) 2010-06-03
CA2743030C (en) 2013-10-22
KR101374412B1 (ko) 2014-03-17
CU24022B1 (es) 2014-07-30
AU2009321221A1 (en) 2010-06-03
GEP20146064B (en) 2014-03-25
RS52810B9 (sr) 2019-06-28
US20110144129A1 (en) 2011-06-16
RS52810B (sr) 2013-10-31
US8946413B2 (en) 2015-02-03
IL212732A0 (en) 2011-07-31
EA201170721A1 (ru) 2011-12-30
US8293903B2 (en) 2012-10-23
MA32834B1 (fr) 2011-11-01
CO6361921A2 (es) 2012-01-20
ME01144B (me) 2013-03-20
SV2011003923A (es) 2011-07-28
ZA201104069B (en) 2012-02-29
HRP20130409T1 (en) 2013-06-30
IL212732A (en) 2016-06-30
RS52810B8 (sr) 2019-08-30
EP2370442B1 (en) 2013-04-24
ES2415430T3 (es) 2013-07-25
EA020470B1 (ru) 2014-11-28
CA2743030A1 (en) 2010-06-03
DOP2011000154A (es) 2011-07-31

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