ECSP088402A - Compuestos y composiciones que contienen diarilamina, y su utilización como moduladores de los receptores c-kit - Google Patents

Compuestos y composiciones que contienen diarilamina, y su utilización como moduladores de los receptores c-kit

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Publication number
ECSP088402A
ECSP088402A EC2008008402A ECSP088402A ECSP088402A EC SP088402 A ECSP088402 A EC SP088402A EC 2008008402 A EC2008008402 A EC 2008008402A EC SP088402 A ECSP088402 A EC SP088402A EC SP088402 A ECSP088402 A EC SP088402A
Authority
EC
Ecuador
Prior art keywords
compounds
kit
diarilamine
modulators
receivers
Prior art date
Application number
EC2008008402A
Other languages
English (en)
Inventor
Pascal Furet
Shifeng Pan
Donald Karanewsky
Shuli You
Yi Liu
Vito Guagnano
Valentina Molteni
Xiaolin Li
Donatella Chianelli
Jon Loren
Juliet Nabakka
Xiaodong Liu
Original Assignee
Irm Llc
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Irm Llc, Novartis Ag filed Critical Irm Llc
Publication of ECSP088402A publication Critical patent/ECSP088402A/es

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    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract

La presente solicitud describe compuestos que incluyen una característica estructural diarilamina. También se describen métodos para hacer tales compuestos, métodos para usar tales compuestos para modular la actividad de los receptores c-kit, y composiciones farmacéuticas y medicamentos que comprenden tales compuestos. También se describen aquí métodos de usar tales compuestos, composiciones farmacéuticas y medicamentos para tratar y/o evitar y/o inhibir y/o mejorar la patología y/o sintomatología de enfermedades o condiciones asociadas con la actividad de los receptores c-kits.
EC2008008402A 2005-09-27 2008-04-25 Compuestos y composiciones que contienen diarilamina, y su utilización como moduladores de los receptores c-kit ECSP088402A (es)

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US20090264649A1 (en) 2009-10-22
US20080139597A1 (en) 2008-06-12
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US20080167308A1 (en) 2008-07-10
EP1928236A4 (en) 2010-07-07
US7563894B2 (en) 2009-07-21
US7638523B2 (en) 2009-12-29
RU2008116313A (ru) 2009-11-10
EP1928236B1 (en) 2011-11-23
WO2007038669A9 (en) 2008-05-29
NZ566862A (en) 2010-12-24
JP2009510086A (ja) 2009-03-12
JP5335426B2 (ja) 2013-11-06
US20070149538A1 (en) 2007-06-28
WO2007038669A2 (en) 2007-04-05
CN101272685A (zh) 2008-09-24
EP1928236A2 (en) 2008-06-11
RU2436776C2 (ru) 2011-12-20
TNSN08140A1 (es) 2009-07-14
KR20080048041A (ko) 2008-05-30
US20090012094A1 (en) 2009-01-08
US7592349B2 (en) 2009-09-22
ATE534293T1 (de) 2011-12-15
MA29851B1 (fr) 2008-10-03
AU2006297089A1 (en) 2007-04-05
US20080139559A1 (en) 2008-06-12
WO2007038669A3 (en) 2007-11-22
NO20081975L (no) 2008-06-02
US7514447B2 (en) 2009-04-07
BRPI0616575A2 (pt) 2011-06-21
IL189927A0 (en) 2008-08-07
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CA2622494A1 (en) 2007-04-05

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