ECSP066468A - Antagonistas de receptores muscarínicos de acetilcolina - Google Patents

Antagonistas de receptores muscarínicos de acetilcolina

Info

Publication number
ECSP066468A
ECSP066468A EC2006006468A ECSP066468A ECSP066468A EC SP066468 A ECSP066468 A EC SP066468A EC 2006006468 A EC2006006468 A EC 2006006468A EC SP066468 A ECSP066468 A EC SP066468A EC SP066468 A ECSP066468 A EC SP066468A
Authority
EC
Ecuador
Prior art keywords
acetilcoline
muscarinic receptors
receptors antagonists
antagonists
muscarinic
Prior art date
Application number
EC2006006468A
Other languages
English (en)
Inventor
Jakob Busch-Petersen
Michael Robert Palovich
Zehong Wan
Chongjie Zhu
Hongxing Yan
Original Assignee
Glaxogroup Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxogroup Ltd filed Critical Glaxogroup Ltd
Publication of ECSP066468A publication Critical patent/ECSP066468A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Neurology (AREA)
  • Emergency Medicine (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se proporcionan antagonistas de receptores de acetilcolina muscarínicos y composiciones farmacéuticas para usarlos.
EC2006006468A 2003-10-14 2006-03-31 Antagonistas de receptores muscarínicos de acetilcolina ECSP066468A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51100903P 2003-10-14 2003-10-14
PCT/US2004/033638 WO2005037280A1 (en) 2003-10-14 2004-10-12 Muscarinic acetycholine receptor antagonists

Publications (1)

Publication Number Publication Date
ECSP066468A true ECSP066468A (es) 2006-11-16

Family

ID=34465175

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006006468A ECSP066468A (es) 2003-10-14 2006-03-31 Antagonistas de receptores muscarínicos de acetilcolina

Country Status (34)

Country Link
US (3) US7276521B2 (es)
EP (1) EP1677795B1 (es)
JP (4) JP2007508390A (es)
KR (3) KR20080067023A (es)
CN (3) CN101230061A (es)
AP (3) AP2007004239A0 (es)
AR (1) AR046103A1 (es)
AT (1) ATE494285T1 (es)
AU (1) AU2004281724B2 (es)
BR (1) BRPI0415361A (es)
CA (1) CA2542657C (es)
CY (1) CY1111364T1 (es)
DE (1) DE602004030930D1 (es)
DK (1) DK1677795T3 (es)
EA (3) EA013435B1 (es)
EC (1) ECSP066468A (es)
ES (1) ES2358673T3 (es)
HR (1) HRP20110232T1 (es)
IL (2) IL174843A0 (es)
IS (1) IS2918B (es)
MA (1) MA28110A1 (es)
MX (1) MXPA06004244A (es)
MY (1) MY143366A (es)
NO (1) NO20062042L (es)
NZ (2) NZ546312A (es)
OA (1) OA13316A (es)
PE (1) PE20050963A1 (es)
PL (1) PL1677795T3 (es)
PT (1) PT1677795E (es)
SG (1) SG147436A1 (es)
SI (1) SI1677795T1 (es)
TW (3) TW200811172A (es)
UA (2) UA89734C2 (es)
WO (1) WO2005037280A1 (es)

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Also Published As

Publication number Publication date
MY143366A (en) 2011-04-29
CA2542657A1 (en) 2005-04-28
CN101230061A (zh) 2008-07-30
MA28110A1 (fr) 2006-08-01
AP2006003566A0 (en) 2006-04-30
UA89734C2 (en) 2010-02-25
DE602004030930D1 (de) 2011-02-17
ATE494285T1 (de) 2011-01-15
IS8441A (is) 2006-05-05
JP4796552B2 (ja) 2011-10-19
JP2011162556A (ja) 2011-08-25
EA200600773A1 (ru) 2008-04-28
EA200702619A1 (ru) 2008-04-28
BRPI0415361A (pt) 2006-12-12
NZ546312A (en) 2008-09-26
HRP20110232T1 (hr) 2011-05-31
US7576096B2 (en) 2009-08-18
ES2358673T3 (es) 2011-05-12
PE20050963A1 (es) 2006-01-11
US7276521B2 (en) 2007-10-02
WO2005037280A1 (en) 2005-04-28
EA200702617A1 (ru) 2008-04-28
IL174843A0 (en) 2006-08-20
EP1677795B1 (en) 2011-01-05
DK1677795T3 (da) 2011-04-18
US20070105895A1 (en) 2007-05-10
US7579361B2 (en) 2009-08-25
SG147436A1 (en) 2008-11-28
IL188112A (en) 2012-10-31
AR046103A1 (es) 2005-11-23
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OA13316A (en) 2007-04-13
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CY1111364T1 (el) 2015-08-05
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TWI409060B (zh) 2013-09-21

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