ECSP034529A - Derivado de tiazolidinodiona y su uso como antidiabetico - Google Patents

Derivado de tiazolidinodiona y su uso como antidiabetico

Info

Publication number
ECSP034529A
ECSP034529A EC2003004529A ECSP034529A ECSP034529A EC SP034529 A ECSP034529 A EC SP034529A EC 2003004529 A EC2003004529 A EC 2003004529A EC SP034529 A ECSP034529 A EC SP034529A EC SP034529 A ECSP034529 A EC SP034529A
Authority
EC
Ecuador
Prior art keywords
compound
tiazolidinodiona
antidiabetic
derived
thiazolidine
Prior art date
Application number
EC2003004529A
Other languages
English (en)
Inventor
Michael Millan
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9900427&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP034529(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of ECSP034529A publication Critical patent/ECSP034529A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se describe un compuesto, sal de potasio de 5-(4-(2-(N-metil-N-(2-piridil)amino)etoxi)bencil)tiazolidino-2,4-diona , o un solvato farmacéuticamente aceptable del mismo, una composición farmacéutica que contiene a dicho compuesto, y el uso de dicho compuesto en medicina, en particular en el tratamiento de diabetes mellitas.
EC2003004529A 2000-09-29 2003-03-28 Derivado de tiazolidinodiona y su uso como antidiabetico ECSP034529A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0023970.7A GB0023970D0 (en) 2000-09-29 2000-09-29 Novel pharmaceutical

Publications (1)

Publication Number Publication Date
ECSP034529A true ECSP034529A (es) 2003-05-26

Family

ID=9900427

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2003004529A ECSP034529A (es) 2000-09-29 2003-03-28 Derivado de tiazolidinodiona y su uso como antidiabetico

Country Status (34)

Country Link
US (1) US20040038968A1 (es)
EP (2) EP1325000B1 (es)
JP (1) JP2004509960A (es)
KR (2) KR100822135B1 (es)
CN (2) CN101961333A (es)
AP (1) AP1841A (es)
AT (1) ATE368038T1 (es)
AU (2) AU9203401A (es)
BG (1) BG107678A (es)
BR (1) BR0114364A (es)
CA (1) CA2423978A1 (es)
CY (1) CY1107767T1 (es)
CZ (1) CZ2003849A3 (es)
DE (1) DE60129576T2 (es)
DK (1) DK1325000T3 (es)
DZ (1) DZ3481A1 (es)
EA (1) EA005110B1 (es)
EC (1) ECSP034529A (es)
ES (1) ES2290169T3 (es)
GB (1) GB0023970D0 (es)
HK (1) HK1058192A1 (es)
HU (1) HUP0301199A3 (es)
IL (2) IL155140A0 (es)
MA (1) MA25913A1 (es)
MX (1) MXPA03002867A (es)
NO (2) NO324970B1 (es)
NZ (1) NZ524932A (es)
OA (1) OA12400A (es)
PL (1) PL361157A1 (es)
PT (1) PT1325000E (es)
SK (1) SK3792003A3 (es)
UA (1) UA76121C2 (es)
WO (1) WO2002026736A1 (es)
ZA (1) ZA200302438B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU225919B1 (en) * 1999-12-18 2007-12-28 Richter Gedeon Nyrt Thiazolidine-derivatives, process for their preparation pharmaceutical and intermediates
HUP0800755A2 (en) 2008-12-11 2010-09-28 Richter Gedeon Nyrt Crystalline forms of rosiglitazone

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5521201A (en) * 1987-09-04 1996-05-28 Beecham Group P.L.C. Method for treatment of atherosclerosis
ATE186724T1 (de) * 1987-09-04 1999-12-15 Beecham Group Plc Substituierte thiazolidindionderivate
GB9124513D0 (en) * 1991-11-19 1992-01-08 Smithkline Beecham Plc Novel process
GB9308487D0 (en) * 1993-04-23 1993-06-09 Smithkline Beecham Plc Novel compounds
GB9712866D0 (en) * 1997-06-18 1997-08-20 Smithkline Beecham Plc Novel method of treatment
GB9723295D0 (en) * 1997-11-04 1998-01-07 Smithkline Beecham Plc Novel process
CN1183130C (zh) * 1999-09-24 2005-01-05 中国人民解放军军事医学科学院毒物药物研究所 噻唑烷类衍生物及其医药用途
HU225919B1 (en) * 1999-12-18 2007-12-28 Richter Gedeon Nyrt Thiazolidine-derivatives, process for their preparation pharmaceutical and intermediates

Also Published As

Publication number Publication date
UA76121C2 (en) 2006-07-17
EA200300423A1 (ru) 2003-08-28
IL155140A0 (en) 2003-10-31
BG107678A (bg) 2003-11-28
EP1325000A1 (en) 2003-07-09
EP1795531A1 (en) 2007-06-13
SK3792003A3 (en) 2004-04-06
IL155140A (en) 2010-06-30
BR0114364A (pt) 2003-12-09
NO324970B1 (no) 2008-01-14
AU9203401A (en) 2002-04-08
EA005110B1 (ru) 2004-10-28
GB0023970D0 (en) 2000-11-15
DE60129576T2 (de) 2008-04-17
HUP0301199A3 (en) 2005-04-28
CZ2003849A3 (cs) 2004-03-17
HUP0301199A2 (hu) 2003-11-28
CY1107767T1 (el) 2013-04-18
CN1620453B (zh) 2010-12-08
KR20070089258A (ko) 2007-08-30
NO20031434D0 (no) 2003-03-28
CN101961333A (zh) 2011-02-02
AP1841A (en) 2008-04-30
ES2290169T3 (es) 2008-02-16
DZ3481A1 (fr) 2002-04-04
JP2004509960A (ja) 2004-04-02
EP1325000B1 (en) 2007-07-25
KR100822135B1 (ko) 2008-04-15
NZ524932A (en) 2005-06-24
HK1058192A1 (en) 2004-05-07
ZA200302438B (en) 2004-04-28
CA2423978A1 (en) 2002-04-04
ATE368038T1 (de) 2007-08-15
US20040038968A1 (en) 2004-02-26
KR20030032058A (ko) 2003-04-23
DK1325000T3 (da) 2007-11-12
AU2001292034B2 (en) 2005-04-21
PL361157A1 (en) 2004-09-20
NO20075507L (no) 2003-05-27
MA25913A1 (fr) 2003-10-01
MXPA03002867A (es) 2004-12-06
DE60129576D1 (de) 2007-09-06
OA12400A (en) 2004-09-06
CN1620453A (zh) 2005-05-25
NO20031434L (no) 2003-05-27
PT1325000E (pt) 2007-10-25
AP2003002766A0 (en) 2003-03-31
WO2002026736A1 (en) 2002-04-04

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