EA036479B1 - Пептид, активирующий рецептор гпп-1 и рецептор глюкагона, фармацевтическая композиция на его основе и их применение для профилактики или лечения ожирения - Google Patents
Пептид, активирующий рецептор гпп-1 и рецептор глюкагона, фармацевтическая композиция на его основе и их применение для профилактики или лечения ожирения Download PDFInfo
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- EA036479B1 EA036479B1 EA201791498A EA201791498A EA036479B1 EA 036479 B1 EA036479 B1 EA 036479B1 EA 201791498 A EA201791498 A EA 201791498A EA 201791498 A EA201791498 A EA 201791498A EA 036479 B1 EA036479 B1 EA 036479B1
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- EA
- Eurasian Patent Office
- Prior art keywords
- peptide
- obesity
- glucagon
- pharmaceutical composition
- receptor
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Endocrinology (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Toxicology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Immunology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1020140193691A KR102418477B1 (ko) | 2014-12-30 | 2014-12-30 | 글루카곤 유도체 |
| PCT/KR2015/014481 WO2016108617A1 (en) | 2014-12-30 | 2015-12-30 | Glucagon derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA201791498A1 EA201791498A1 (ru) | 2017-10-31 |
| EA036479B1 true EA036479B1 (ru) | 2020-11-16 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA201791498A EA036479B1 (ru) | 2014-12-30 | 2015-12-30 | Пептид, активирующий рецептор гпп-1 и рецептор глюкагона, фармацевтическая композиция на его основе и их применение для профилактики или лечения ожирения |
Country Status (18)
| Country | Link |
|---|---|
| US (3) | US10513550B2 (OSRAM) |
| EP (1) | EP3240802B1 (OSRAM) |
| JP (1) | JP6758297B2 (OSRAM) |
| KR (1) | KR102418477B1 (OSRAM) |
| CN (1) | CN107250155B (OSRAM) |
| AR (1) | AR103323A1 (OSRAM) |
| AU (1) | AU2015372767B2 (OSRAM) |
| BR (1) | BR112017013845A2 (OSRAM) |
| CA (1) | CA2972001C (OSRAM) |
| EA (1) | EA036479B1 (OSRAM) |
| IL (1) | IL253001B (OSRAM) |
| MX (1) | MX389593B (OSRAM) |
| PH (1) | PH12017501205A1 (OSRAM) |
| SG (2) | SG11201705130XA (OSRAM) |
| TW (1) | TWI696631B (OSRAM) |
| UA (1) | UA122967C2 (OSRAM) |
| WO (1) | WO2016108617A1 (OSRAM) |
| ZA (1) | ZA201704328B (OSRAM) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11135271B2 (en) * | 2014-12-30 | 2021-10-05 | Hanmi Pharm. Co., Ltd. | Glucagon derivatives with improved stability |
| US10696725B2 (en) | 2015-06-30 | 2020-06-30 | Hanmi Pharm. Co., Ltd. | Glucagon derivative and a composition comprising a long acting conjugate of the same |
| TWI622596B (zh) | 2015-10-26 | 2018-05-01 | 美國禮來大藥廠 | 升糖素受體促效劑 |
| CN116063453A (zh) | 2015-12-31 | 2023-05-05 | 韩美药品株式会社 | 胰高血糖素/glp-1/gip受体三重激动剂 |
| JP2025526148A (ja) | 2022-08-18 | 2025-08-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 長時間作用型ｇｌｐ－１／グルカゴン受容体アゴニスト及びｎｐｙ２受容体アゴニストを含む組合せ治療 |
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