EA016628B1 - Применение бензоконденсированных гетероциклических сульфамидных производных в качестве нейропротективных агентов - Google Patents
Применение бензоконденсированных гетероциклических сульфамидных производных в качестве нейропротективных агентов Download PDFInfo
- Publication number
- EA016628B1 EA016628B1 EA200870087A EA200870087A EA016628B1 EA 016628 B1 EA016628 B1 EA 016628B1 EA 200870087 A EA200870087 A EA 200870087A EA 200870087 A EA200870087 A EA 200870087A EA 016628 B1 EA016628 B1 EA 016628B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- dihydrobenzo
- dioxinyl
- compound
- group
- formula
- Prior art date
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
- A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A61P39/06—Free radical scavengers or antioxidants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
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- Neurosurgery (AREA)
- Epidemiology (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
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- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Biochemistry (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Toxicology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US75149405P | 2005-12-19 | 2005-12-19 | |
| US11/612,146 US20070155823A1 (en) | 2005-12-19 | 2006-12-18 | Use of benzo-fused heterocycle sulfamide derivatives as neuroprotective agents |
| PCT/US2006/048451 WO2007075698A2 (en) | 2005-12-19 | 2006-12-19 | Use of benzo-fused heterocycle sulfamide derivatives as neuroprotective agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200870087A1 EA200870087A1 (ru) | 2009-12-30 |
| EA016628B1 true EA016628B1 (ru) | 2012-06-29 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200870087A EA016628B1 (ru) | 2005-12-19 | 2006-12-19 | Применение бензоконденсированных гетероциклических сульфамидных производных в качестве нейропротективных агентов |
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| US (1) | US20070155823A1 (https=) |
| EP (1) | EP1968571B1 (https=) |
| JP (1) | JP5190373B2 (https=) |
| KR (1) | KR20080089405A (https=) |
| AT (1) | ATE536182T1 (https=) |
| AU (1) | AU2006331783A1 (https=) |
| BR (1) | BRPI0620060A2 (https=) |
| CA (1) | CA2634088A1 (https=) |
| CR (1) | CR10171A (https=) |
| CY (1) | CY1112444T1 (https=) |
| DK (1) | DK1968571T3 (https=) |
| EA (1) | EA016628B1 (https=) |
| ES (1) | ES2375845T3 (https=) |
| HR (1) | HRP20120018T1 (https=) |
| IL (1) | IL192106A0 (https=) |
| MY (1) | MY149175A (https=) |
| NO (1) | NO20083033L (https=) |
| NZ (1) | NZ569041A (https=) |
| PL (1) | PL1968571T3 (https=) |
| PT (1) | PT1968571E (https=) |
| RS (1) | RS52220B (https=) |
| SI (1) | SI1968571T1 (https=) |
| WO (1) | WO2007075698A2 (https=) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY147767A (en) | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
| KR20080012360A (ko) * | 2005-05-20 | 2008-02-11 | 얀센 파마슈티카 엔.브이. | 설파미드 유도체의 제조 방법 |
| US8497298B2 (en) | 2005-12-19 | 2013-07-30 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels |
| US8937096B2 (en) | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
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Also Published As
| Publication number | Publication date |
|---|---|
| RS52220B (sr) | 2012-10-31 |
| ATE536182T1 (de) | 2011-12-15 |
| IL192106A0 (en) | 2009-08-03 |
| WO2007075698A2 (en) | 2007-07-05 |
| NO20083033L (no) | 2008-09-16 |
| BRPI0620060A2 (pt) | 2011-11-01 |
| CA2634088A1 (en) | 2007-07-05 |
| KR20080089405A (ko) | 2008-10-06 |
| DK1968571T3 (da) | 2012-02-27 |
| AU2006331783A1 (en) | 2007-07-05 |
| HK1124544A1 (en) | 2009-07-17 |
| JP2009520031A (ja) | 2009-05-21 |
| NZ569041A (en) | 2011-04-29 |
| SI1968571T1 (sl) | 2012-03-30 |
| PT1968571E (pt) | 2012-02-01 |
| US20070155823A1 (en) | 2007-07-05 |
| PL1968571T3 (pl) | 2012-04-30 |
| EP1968571A2 (en) | 2008-09-17 |
| CR10171A (es) | 2009-01-16 |
| WO2007075698A3 (en) | 2007-08-16 |
| EP1968571B1 (en) | 2011-12-07 |
| EA200870087A1 (ru) | 2009-12-30 |
| ES2375845T3 (es) | 2012-03-06 |
| HRP20120018T1 (hr) | 2012-01-31 |
| JP5190373B2 (ja) | 2013-04-24 |
| MY149175A (en) | 2013-07-31 |
| CY1112444T1 (el) | 2015-12-09 |
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