EA007483B1 - Применение модулятора рецепторов глюкокортикоидов и агониста рецепторов глюкокортикоидов при получении лекарственного средства - Google Patents
Применение модулятора рецепторов глюкокортикоидов и агониста рецепторов глюкокортикоидов при получении лекарственного средства Download PDFInfo
- Publication number
- EA007483B1 EA007483B1 EA200400337A EA200400337A EA007483B1 EA 007483 B1 EA007483 B1 EA 007483B1 EA 200400337 A EA200400337 A EA 200400337A EA 200400337 A EA200400337 A EA 200400337A EA 007483 B1 EA007483 B1 EA 007483B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- octahydro
- phenylmethyl
- methyl
- hydroxy
- propynyl
- Prior art date
Links
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Classifications
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- C07D455/06—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine containing benzo [a] quinolizine ring systems
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| RU2507204C2 (ru) * | 2009-08-31 | 2014-02-20 | Мерк Шарп И Доум Корп. | Положительные аллостерические модуляторы м1-рецепторов на основе пираниларилметилбензохиназолинона |
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| US6777399B2 (en) | 2000-08-05 | 2004-08-17 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative compositions |
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| US8846702B2 (en) | 2009-08-31 | 2014-09-30 | Merck Sharp & Dohme Corp. | Pyranyl aryl methyl benzoquinazolinone M1 receptor positive allosteric modulators |
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