DK517776A - Fremgangsmade til femstilling af heterocycliske forbindelser - Google Patents

Fremgangsmade til femstilling af heterocycliske forbindelser

Info

Publication number
DK517776A
DK517776A DK517776A DK517776A DK517776A DK 517776 A DK517776 A DK 517776A DK 517776 A DK517776 A DK 517776A DK 517776 A DK517776 A DK 517776A DK 517776 A DK517776 A DK 517776A
Authority
DK
Denmark
Prior art keywords
procedure
heterocyclic compounds
preparing heterocyclic
preparing
compounds
Prior art date
Application number
DK517776A
Other languages
Danish (da)
English (en)
Inventor
K H Baggaley
Original Assignee
Beecham Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Ltd filed Critical Beecham Group Ltd
Publication of DK517776A publication Critical patent/DK517776A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
DK517776A 1975-11-18 1976-11-17 Fremgangsmade til femstilling af heterocycliske forbindelser DK517776A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4737375 1975-11-18

Publications (1)

Publication Number Publication Date
DK517776A true DK517776A (da) 1977-05-19

Family

ID=10444739

Family Applications (1)

Application Number Title Priority Date Filing Date
DK517776A DK517776A (da) 1975-11-18 1976-11-17 Fremgangsmade til femstilling af heterocycliske forbindelser

Country Status (28)

Country Link
US (5) US4113728A (un)
JP (1) JPS5262273A (un)
AR (3) AR217411A1 (un)
AT (1) AT355017B (un)
AU (2) AU504599B2 (un)
BE (1) BE848371A (un)
BG (4) BG24808A3 (un)
CA (1) CA1064511A (un)
CH (1) CH627465A5 (un)
CS (4) CS192593B2 (un)
DD (1) DD127645A5 (un)
DE (1) DE2652201A1 (un)
DK (1) DK517776A (un)
ES (3) ES453420A1 (un)
FI (1) FI763285A (un)
FR (1) FR2332019A1 (un)
HU (1) HU173958B (un)
IL (1) IL50690A (un)
NL (1) NL7612796A (un)
NO (1) NO763922L (un)
NZ (1) NZ182325A (un)
PH (1) PH13918A (un)
PL (1) PL193742A1 (un)
PT (1) PT65851B (un)
RO (4) RO75777A (un)
SE (1) SE7612919L (un)
SU (4) SU682129A3 (un)
ZA (1) ZA766489B (un)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
US4190663A (en) * 1976-01-24 1980-02-26 Bayer Aktiengesellschaft Anti-thrombotic 1,2-benzisothiazolin-3-ones
DE2602643C2 (de) * 1976-01-24 1984-12-20 Bayer Ag, 5090 Leverkusen 1,2-Benzisothiazolinone-3, Verfahren zu ihrer Herstellung sowie Arzneimittel
EP0000254B1 (en) * 1977-06-20 1981-06-10 Beecham Group Plc Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions
DE2860430D1 (en) * 1977-10-08 1981-02-26 Beecham Group Ltd Antithrombotic compositions containing benzisothiazolones
ATE7296T1 (de) * 1979-10-08 1984-05-15 Merck & Co. Inc. 2-aryl-1,2-benzisothiazolinon-1,1-dioxide und sie enthaltende pharmazeutische zusammensetzungen.
DE3226284A1 (de) * 1982-07-14 1984-01-19 A. Nattermann & Cie GmbH, 5000 Köln Neue benzisoselenazolone, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3238006A1 (de) * 1982-10-13 1984-04-19 Bayer Ag, 5090 Leverkusen Azolyl-methylamine, ihre herstellung und verwendung in mikrobiziden mitteln
DE3500577A1 (de) * 1985-01-10 1986-07-10 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 1,2-benzisothiazolonen
US4732984A (en) * 1985-10-17 1988-03-22 American Home Products Corporation Piperazinoisothiazolones with psychotropic activity
DE3617976A1 (de) * 1986-05-28 1988-01-14 Alter Sa 1,4-dihydropyridin, verfahren zu dessen herstellung und dessen verwendung in antithrombotischen medikamenten
US4831031A (en) * 1988-01-22 1989-05-16 Pfizer Inc. Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity
CA1340759C (en) * 1988-07-01 1999-09-21 James P. Albarella Isobenzothiazolone chromogenic thiol indicators and their derivatives
US5128457A (en) * 1988-07-01 1992-07-07 Miles Inc. Chromogenic thiol indicators based on an isobenzothiazolone ring system
US5236917A (en) * 1989-05-04 1993-08-17 Sterling Winthrop Inc. Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
WO2010039545A2 (en) * 2008-09-23 2010-04-08 Georgetown University 1,2-benzisothiazolinone and isoindolinone derivatives
US9428472B2 (en) 2011-08-16 2016-08-30 Georgetown University Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives
WO2017070157A1 (en) * 2015-10-19 2017-04-27 Emory University Redox dehydration coupling catalysts and methods related thereto

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE565380A (un) * 1957-03-08
US3012039A (en) * 1958-03-14 1961-12-05 Ici Ltd 2-p-chlorobenzyl-1, 2-benzisothiazolone
DE1147947B (de) * 1961-07-25 1963-05-02 Knoll Ag Verfahren zur Herstellung neuer 1, 2-Benzisothiazolone
SE392103B (sv) * 1970-04-27 1977-03-14 Sherwin Williams Co Sett att framstella 1,2-bensisotiazolin-3-oner
US3661974A (en) * 1970-04-27 1972-05-09 Sherwin Williams Co 2-carbalkoxy-phenyl sulfenamides
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
GB1582214A (en) * 1977-05-31 1981-01-07 Beecham Group Ltd Antithrombotic compositions
DE2734882A1 (de) * 1977-08-03 1979-02-22 Basf Ag 3- eckige klammer auf 4-(1,3-diazacycloalken-2-yl)-phenyl eckige klammer zu -1,2-benzisothiazole, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
CS192592B2 (en) 1979-08-31
FR2332019B1 (un) 1983-05-20
US4113728A (en) 1978-09-12
AU520890B2 (en) 1982-03-04
AR215271A1 (es) 1979-09-28
RO75777A (ro) 1981-02-28
SU682129A3 (ru) 1979-08-25
NO763922L (un) 1977-05-20
ATA849176A (de) 1979-07-15
RO75540A (ro) 1980-11-30
NL7612796A (nl) 1977-05-23
IL50690A (en) 1980-01-31
SU671728A3 (ru) 1979-06-30
ES453420A1 (es) 1978-02-16
RO75730A (ro) 1981-02-28
FI763285A (un) 1977-05-19
US4243669A (en) 1981-01-06
AU1916376A (en) 1978-05-04
CS192594B2 (en) 1979-08-31
CS192593B2 (en) 1979-08-31
BG24809A3 (en) 1978-05-12
JPS5262273A (en) 1977-05-23
SU701536A3 (ru) 1979-11-30
RO69608A (ro) 1982-07-06
US4212872A (en) 1980-07-15
AR217411A1 (es) 1980-03-31
AT355017B (de) 1980-02-11
CH627465A5 (de) 1982-01-15
AU504599B2 (en) 1979-10-18
IL50690A0 (en) 1976-12-31
AR217449A1 (es) 1980-03-31
ES465173A1 (es) 1978-10-01
SU679141A3 (ru) 1979-08-05
ES465174A1 (es) 1978-10-01
SE7612919L (sv) 1977-05-19
NZ182325A (en) 1979-03-16
PT65851B (en) 1978-05-15
BG24810A3 (en) 1978-05-12
AU4716379A (en) 1979-09-27
BE848371A (fr) 1977-05-16
DE2652201A1 (de) 1977-06-02
US4350702A (en) 1982-09-21
BG24808A3 (en) 1978-05-12
DD127645A5 (un) 1977-10-05
ZA766489B (en) 1977-10-26
US4212979A (en) 1980-07-15
CA1064511A (en) 1979-10-16
FR2332019A1 (fr) 1977-06-17
PT65851A (en) 1976-12-01
HU173958B (hu) 1979-09-28
PL193742A1 (pl) 1979-05-21
BG24811A3 (en) 1978-05-12
PH13918A (en) 1980-11-04
CS192570B2 (en) 1979-08-31

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