CS192594B2 - Method of preparing benzisothiazolones - Google Patents

Method of preparing benzisothiazolones

Info

Publication number
CS192594B2
CS192594B2 CS775981A CS598177A CS192594B2 CS 192594 B2 CS192594 B2 CS 192594B2 CS 775981 A CS775981 A CS 775981A CS 598177 A CS598177 A CS 598177A CS 192594 B2 CS192594 B2 CS 192594B2
Authority
CS
Czechoslovakia
Prior art keywords
benzisothiazolones
preparing
preparing benzisothiazolones
Prior art date
Application number
CS775981A
Other languages
English (en)
Inventor
Keith H Baggaley
Original Assignee
Robapharm Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robapharm Ag filed Critical Robapharm Ag
Publication of CS192594B2 publication Critical patent/CS192594B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
CS775981A 1975-11-18 1976-11-17 Method of preparing benzisothiazolones CS192594B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4737375 1975-11-18

Publications (1)

Publication Number Publication Date
CS192594B2 true CS192594B2 (en) 1979-08-31

Family

ID=10444739

Family Applications (4)

Application Number Title Priority Date Filing Date
CS767392A CS192570B2 (en) 1975-11-18 1976-11-17 Method of producing benzisothiazolones
CS775979A CS192592B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones
CS775980A CS192593B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones
CS775981A CS192594B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones

Family Applications Before (3)

Application Number Title Priority Date Filing Date
CS767392A CS192570B2 (en) 1975-11-18 1976-11-17 Method of producing benzisothiazolones
CS775979A CS192592B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones
CS775980A CS192593B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones

Country Status (28)

Country Link
US (5) US4113728A (cs)
JP (1) JPS5262273A (cs)
AR (3) AR217411A1 (cs)
AT (1) AT355017B (cs)
AU (2) AU504599B2 (cs)
BE (1) BE848371A (cs)
BG (4) BG24811A3 (cs)
CA (1) CA1064511A (cs)
CH (1) CH627465A5 (cs)
CS (4) CS192570B2 (cs)
DD (1) DD127645A5 (cs)
DE (1) DE2652201A1 (cs)
DK (1) DK517776A (cs)
ES (3) ES453420A1 (cs)
FI (1) FI763285A (cs)
FR (1) FR2332019A1 (cs)
HU (1) HU173958B (cs)
IL (1) IL50690A (cs)
NL (1) NL7612796A (cs)
NO (1) NO763922L (cs)
NZ (1) NZ182325A (cs)
PH (1) PH13918A (cs)
PL (1) PL193742A1 (cs)
PT (1) PT65851B (cs)
RO (4) RO75730A (cs)
SE (1) SE7612919L (cs)
SU (4) SU682129A3 (cs)
ZA (1) ZA766489B (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
DE2602643C2 (de) * 1976-01-24 1984-12-20 Bayer Ag, 5090 Leverkusen 1,2-Benzisothiazolinone-3, Verfahren zu ihrer Herstellung sowie Arzneimittel
US4190663A (en) * 1976-01-24 1980-02-26 Bayer Aktiengesellschaft Anti-thrombotic 1,2-benzisothiazolin-3-ones
DE2860750D1 (en) * 1977-06-20 1981-09-17 Beecham Group Plc Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions
EP0001503B1 (en) * 1977-10-08 1981-01-07 Beecham Group Plc Antithrombotic compositions containing benzisothiazolones
ATE7296T1 (de) * 1979-10-08 1984-05-15 Merck & Co. Inc. 2-aryl-1,2-benzisothiazolinon-1,1-dioxide und sie enthaltende pharmazeutische zusammensetzungen.
DE3226284A1 (de) * 1982-07-14 1984-01-19 A. Nattermann & Cie GmbH, 5000 Köln Neue benzisoselenazolone, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3238006A1 (de) * 1982-10-13 1984-04-19 Bayer Ag, 5090 Leverkusen Azolyl-methylamine, ihre herstellung und verwendung in mikrobiziden mitteln
DE3500577A1 (de) * 1985-01-10 1986-07-10 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 1,2-benzisothiazolonen
US4732984A (en) * 1985-10-17 1988-03-22 American Home Products Corporation Piperazinoisothiazolones with psychotropic activity
DE3617976A1 (de) * 1986-05-28 1988-01-14 Alter Sa 1,4-dihydropyridin, verfahren zu dessen herstellung und dessen verwendung in antithrombotischen medikamenten
US4831031A (en) * 1988-01-22 1989-05-16 Pfizer Inc. Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity
US5128457A (en) * 1988-07-01 1992-07-07 Miles Inc. Chromogenic thiol indicators based on an isobenzothiazolone ring system
CA1340759C (en) * 1988-07-01 1999-09-21 James P. Albarella Isobenzothiazolone chromogenic thiol indicators and their derivatives
US5236917A (en) * 1989-05-04 1993-08-17 Sterling Winthrop Inc. Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
CA2738314C (en) * 2008-09-23 2017-01-10 Georgetown University 1,2-benzisothiazolinone and isoindolinone derivatives
WO2013025897A1 (en) 2011-08-16 2013-02-21 Georgetown University Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives
US20180318818A1 (en) 2015-10-19 2018-11-08 Emory University Redox Dehydration Coupling Catalysts and Methods Related Thereto

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE565380A (cs) * 1957-03-08
US3012039A (en) * 1958-03-14 1961-12-05 Ici Ltd 2-p-chlorobenzyl-1, 2-benzisothiazolone
DE1147947B (de) * 1961-07-25 1963-05-02 Knoll Ag Verfahren zur Herstellung neuer 1, 2-Benzisothiazolone
SE392103B (sv) * 1970-04-27 1977-03-14 Sherwin Williams Co Sett att framstella 1,2-bensisotiazolin-3-oner
US3661974A (en) * 1970-04-27 1972-05-09 Sherwin Williams Co 2-carbalkoxy-phenyl sulfenamides
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
GB1582214A (en) * 1977-05-31 1981-01-07 Beecham Group Ltd Antithrombotic compositions
DE2734882A1 (de) * 1977-08-03 1979-02-22 Basf Ag 3- eckige klammer auf 4-(1,3-diazacycloalken-2-yl)-phenyl eckige klammer zu -1,2-benzisothiazole, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
BG24811A3 (en) 1978-05-12
AT355017B (de) 1980-02-11
BG24809A3 (en) 1978-05-12
IL50690A (en) 1980-01-31
NO763922L (cs) 1977-05-20
DE2652201A1 (de) 1977-06-02
CS192593B2 (en) 1979-08-31
ES453420A1 (es) 1978-02-16
ES465174A1 (es) 1978-10-01
AU504599B2 (en) 1979-10-18
FR2332019A1 (fr) 1977-06-17
JPS5262273A (en) 1977-05-23
CH627465A5 (de) 1982-01-15
CS192570B2 (en) 1979-08-31
AR217449A1 (es) 1980-03-31
DK517776A (da) 1977-05-19
PL193742A1 (pl) 1979-05-21
FI763285A (cs) 1977-05-19
ES465173A1 (es) 1978-10-01
SU679141A3 (ru) 1979-08-05
SU682129A3 (ru) 1979-08-25
RO75540A (ro) 1980-11-30
CS192592B2 (en) 1979-08-31
US4113728A (en) 1978-09-12
PT65851A (en) 1976-12-01
AU520890B2 (en) 1982-03-04
AU4716379A (en) 1979-09-27
AR215271A1 (es) 1979-09-28
BG24808A3 (en) 1978-05-12
BE848371A (fr) 1977-05-16
RO75777A (ro) 1981-02-28
CA1064511A (en) 1979-10-16
SE7612919L (sv) 1977-05-19
ATA849176A (de) 1979-07-15
NZ182325A (en) 1979-03-16
FR2332019B1 (cs) 1983-05-20
ZA766489B (en) 1977-10-26
RO69608A (ro) 1982-07-06
US4212872A (en) 1980-07-15
NL7612796A (nl) 1977-05-23
BG24810A3 (en) 1978-05-12
US4350702A (en) 1982-09-21
SU701536A3 (ru) 1979-11-30
SU671728A3 (ru) 1979-06-30
US4243669A (en) 1981-01-06
AU1916376A (en) 1978-05-04
IL50690A0 (en) 1976-12-31
PT65851B (en) 1978-05-15
HU173958B (hu) 1979-09-28
AR217411A1 (es) 1980-03-31
DD127645A5 (cs) 1977-10-05
RO75730A (ro) 1981-02-28
US4212979A (en) 1980-07-15
PH13918A (en) 1980-11-04

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