CS192570B2 - Method of producing benzisothiazolones - Google Patents

Method of producing benzisothiazolones

Info

Publication number
CS192570B2
CS192570B2 CS767392A CS739276A CS192570B2 CS 192570 B2 CS192570 B2 CS 192570B2 CS 767392 A CS767392 A CS 767392A CS 739276 A CS739276 A CS 739276A CS 192570 B2 CS192570 B2 CS 192570B2
Authority
CS
Czechoslovakia
Prior art keywords
benzisothiazolones
producing
producing benzisothiazolones
Prior art date
Application number
CS767392A
Other languages
English (en)
Inventor
Keith H Baggaley
Original Assignee
Robapharm Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robapharm Ag filed Critical Robapharm Ag
Publication of CS192570B2 publication Critical patent/CS192570B2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
CS767392A 1975-11-18 1976-11-17 Method of producing benzisothiazolones CS192570B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4737375 1975-11-18

Publications (1)

Publication Number Publication Date
CS192570B2 true CS192570B2 (en) 1979-08-31

Family

ID=10444739

Family Applications (4)

Application Number Title Priority Date Filing Date
CS775981A CS192594B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones
CS775979A CS192592B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones
CS767392A CS192570B2 (en) 1975-11-18 1976-11-17 Method of producing benzisothiazolones
CS775980A CS192593B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CS775981A CS192594B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones
CS775979A CS192592B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS775980A CS192593B2 (en) 1975-11-18 1976-11-17 Method of preparing benzisothiazolones

Country Status (28)

Country Link
US (5) US4113728A (cs)
JP (1) JPS5262273A (cs)
AR (3) AR217411A1 (cs)
AT (1) AT355017B (cs)
AU (2) AU504599B2 (cs)
BE (1) BE848371A (cs)
BG (4) BG24811A3 (cs)
CA (1) CA1064511A (cs)
CH (1) CH627465A5 (cs)
CS (4) CS192594B2 (cs)
DD (1) DD127645A5 (cs)
DE (1) DE2652201A1 (cs)
DK (1) DK517776A (cs)
ES (3) ES453420A1 (cs)
FI (1) FI763285A (cs)
FR (1) FR2332019A1 (cs)
HU (1) HU173958B (cs)
IL (1) IL50690A (cs)
NL (1) NL7612796A (cs)
NO (1) NO763922L (cs)
NZ (1) NZ182325A (cs)
PH (1) PH13918A (cs)
PL (1) PL193742A1 (cs)
PT (1) PT65851B (cs)
RO (4) RO69608A (cs)
SE (1) SE7612919L (cs)
SU (4) SU682129A3 (cs)
ZA (1) ZA766489B (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
DE2602643C2 (de) * 1976-01-24 1984-12-20 Bayer Ag, 5090 Leverkusen 1,2-Benzisothiazolinone-3, Verfahren zu ihrer Herstellung sowie Arzneimittel
US4190663A (en) * 1976-01-24 1980-02-26 Bayer Aktiengesellschaft Anti-thrombotic 1,2-benzisothiazolin-3-ones
DE2860750D1 (en) * 1977-06-20 1981-09-17 Beecham Group Plc Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions
EP0001503B1 (en) * 1977-10-08 1981-01-07 Beecham Group Plc Antithrombotic compositions containing benzisothiazolones
ATE7296T1 (de) * 1979-10-08 1984-05-15 Merck & Co. Inc. 2-aryl-1,2-benzisothiazolinon-1,1-dioxide und sie enthaltende pharmazeutische zusammensetzungen.
DE3226284A1 (de) * 1982-07-14 1984-01-19 A. Nattermann & Cie GmbH, 5000 Köln Neue benzisoselenazolone, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3238006A1 (de) * 1982-10-13 1984-04-19 Bayer Ag, 5090 Leverkusen Azolyl-methylamine, ihre herstellung und verwendung in mikrobiziden mitteln
DE3500577A1 (de) * 1985-01-10 1986-07-10 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 1,2-benzisothiazolonen
US4732984A (en) * 1985-10-17 1988-03-22 American Home Products Corporation Piperazinoisothiazolones with psychotropic activity
DE3617976A1 (de) * 1986-05-28 1988-01-14 Alter Sa 1,4-dihydropyridin, verfahren zu dessen herstellung und dessen verwendung in antithrombotischen medikamenten
US4831031A (en) * 1988-01-22 1989-05-16 Pfizer Inc. Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity
CA1340759C (en) * 1988-07-01 1999-09-21 James P. Albarella Isobenzothiazolone chromogenic thiol indicators and their derivatives
US5128457A (en) * 1988-07-01 1992-07-07 Miles Inc. Chromogenic thiol indicators based on an isobenzothiazolone ring system
US5236917A (en) * 1989-05-04 1993-08-17 Sterling Winthrop Inc. Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
AU2009298888A1 (en) * 2008-09-23 2010-04-08 Georgetown University 1,2-benzisothiazolinone and isoindolinone derivatives
CA2845551C (en) 2011-08-16 2020-06-09 Georgetown University Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives
WO2017070157A1 (en) 2015-10-19 2017-04-27 Emory University Redox dehydration coupling catalysts and methods related thereto

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE565380A (cs) * 1957-03-08
US3012039A (en) * 1958-03-14 1961-12-05 Ici Ltd 2-p-chlorobenzyl-1, 2-benzisothiazolone
DE1147947B (de) * 1961-07-25 1963-05-02 Knoll Ag Verfahren zur Herstellung neuer 1, 2-Benzisothiazolone
SE392103B (sv) * 1970-04-27 1977-03-14 Sherwin Williams Co Sett att framstella 1,2-bensisotiazolin-3-oner
US3661974A (en) * 1970-04-27 1972-05-09 Sherwin Williams Co 2-carbalkoxy-phenyl sulfenamides
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
GB1582214A (en) * 1977-05-31 1981-01-07 Beecham Group Ltd Antithrombotic compositions
DE2734882A1 (de) * 1977-08-03 1979-02-22 Basf Ag 3- eckige klammer auf 4-(1,3-diazacycloalken-2-yl)-phenyl eckige klammer zu -1,2-benzisothiazole, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
AT355017B (de) 1980-02-11
US4243669A (en) 1981-01-06
BG24810A3 (en) 1978-05-12
CS192593B2 (en) 1979-08-31
HU173958B (hu) 1979-09-28
DD127645A5 (cs) 1977-10-05
SE7612919L (sv) 1977-05-19
AU1916376A (en) 1978-05-04
SU679141A3 (ru) 1979-08-05
BG24811A3 (en) 1978-05-12
DK517776A (da) 1977-05-19
NO763922L (cs) 1977-05-20
IL50690A (en) 1980-01-31
US4212979A (en) 1980-07-15
BG24809A3 (en) 1978-05-12
RO69608A (ro) 1982-07-06
US4212872A (en) 1980-07-15
NL7612796A (nl) 1977-05-23
AR217411A1 (es) 1980-03-31
CA1064511A (en) 1979-10-16
FR2332019B1 (cs) 1983-05-20
ES453420A1 (es) 1978-02-16
AU520890B2 (en) 1982-03-04
ES465173A1 (es) 1978-10-01
AR215271A1 (es) 1979-09-28
CS192594B2 (en) 1979-08-31
PH13918A (en) 1980-11-04
FI763285A (cs) 1977-05-19
SU701536A3 (ru) 1979-11-30
FR2332019A1 (fr) 1977-06-17
RO75777A (ro) 1981-02-28
ZA766489B (en) 1977-10-26
US4113728A (en) 1978-09-12
ATA849176A (de) 1979-07-15
PT65851B (en) 1978-05-15
CH627465A5 (de) 1982-01-15
RO75540A (ro) 1980-11-30
IL50690A0 (en) 1976-12-31
RO75730A (ro) 1981-02-28
PT65851A (en) 1976-12-01
SU671728A3 (ru) 1979-06-30
SU682129A3 (ru) 1979-08-25
AU4716379A (en) 1979-09-27
BE848371A (fr) 1977-05-16
DE2652201A1 (de) 1977-06-02
US4350702A (en) 1982-09-21
AU504599B2 (en) 1979-10-18
ES465174A1 (es) 1978-10-01
PL193742A1 (pl) 1979-05-21
CS192592B2 (en) 1979-08-31
AR217449A1 (es) 1980-03-31
BG24808A3 (en) 1978-05-12
JPS5262273A (en) 1977-05-23
NZ182325A (en) 1979-03-16

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