AR217449A1 - Procedimiento para la preparacion de derivados de 1,2-benzoisotiozol 3-ona y una sal de adicion acida farmaceuticamente aceptable - Google Patents

Procedimiento para la preparacion de derivados de 1,2-benzoisotiozol 3-ona y una sal de adicion acida farmaceuticamente aceptable

Info

Publication number
AR217449A1
AR217449A1 AR269610A AR26961077A AR217449A1 AR 217449 A1 AR217449 A1 AR 217449A1 AR 269610 A AR269610 A AR 269610A AR 26961077 A AR26961077 A AR 26961077A AR 217449 A1 AR217449 A1 AR 217449A1
Authority
AR
Argentina
Prior art keywords
benzoisotiozol
procedure
preparation
pharmaceutically acceptable
addition salt
Prior art date
Application number
AR269610A
Other languages
English (en)
Original Assignee
Beecham Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Ltd filed Critical Beecham Group Ltd
Application granted granted Critical
Publication of AR217449A1 publication Critical patent/AR217449A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
AR269610A 1975-11-18 1977-10-17 Procedimiento para la preparacion de derivados de 1,2-benzoisotiozol 3-ona y una sal de adicion acida farmaceuticamente aceptable AR217449A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4737375 1975-11-18

Publications (1)

Publication Number Publication Date
AR217449A1 true AR217449A1 (es) 1980-03-31

Family

ID=10444739

Family Applications (3)

Application Number Title Priority Date Filing Date
AR265414A AR217411A1 (es) 1975-11-18 1976-11-10 Procedimiento para la preparacion de derivados de 1,2-benzoisotiazol-3-ona y una sal de adicion acida farmaceuticamente aceptable
AR269610A AR217449A1 (es) 1975-11-18 1977-10-17 Procedimiento para la preparacion de derivados de 1,2-benzoisotiozol 3-ona y una sal de adicion acida farmaceuticamente aceptable
AR269611A AR215271A1 (es) 1975-11-18 1977-10-17 Un procedimiento para la preparacion de derivados de 1,2-benzoisotiazol-3-ona y una sal de adicion acida farmaceuticamente aceptable

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR265414A AR217411A1 (es) 1975-11-18 1976-11-10 Procedimiento para la preparacion de derivados de 1,2-benzoisotiazol-3-ona y una sal de adicion acida farmaceuticamente aceptable

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR269611A AR215271A1 (es) 1975-11-18 1977-10-17 Un procedimiento para la preparacion de derivados de 1,2-benzoisotiazol-3-ona y una sal de adicion acida farmaceuticamente aceptable

Country Status (28)

Country Link
US (5) US4113728A (es)
JP (1) JPS5262273A (es)
AR (3) AR217411A1 (es)
AT (1) AT355017B (es)
AU (2) AU504599B2 (es)
BE (1) BE848371A (es)
BG (4) BG24810A3 (es)
CA (1) CA1064511A (es)
CH (1) CH627465A5 (es)
CS (4) CS192592B2 (es)
DD (1) DD127645A5 (es)
DE (1) DE2652201A1 (es)
DK (1) DK517776A (es)
ES (3) ES453420A1 (es)
FI (1) FI763285A (es)
FR (1) FR2332019A1 (es)
HU (1) HU173958B (es)
IL (1) IL50690A (es)
NL (1) NL7612796A (es)
NO (1) NO763922L (es)
NZ (1) NZ182325A (es)
PH (1) PH13918A (es)
PL (1) PL193742A1 (es)
PT (1) PT65851B (es)
RO (4) RO69608A (es)
SE (1) SE7612919L (es)
SU (4) SU682129A3 (es)
ZA (1) ZA766489B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
DE2602643C2 (de) * 1976-01-24 1984-12-20 Bayer Ag, 5090 Leverkusen 1,2-Benzisothiazolinone-3, Verfahren zu ihrer Herstellung sowie Arzneimittel
US4190663A (en) * 1976-01-24 1980-02-26 Bayer Aktiengesellschaft Anti-thrombotic 1,2-benzisothiazolin-3-ones
DE2860750D1 (en) * 1977-06-20 1981-09-17 Beecham Group Plc Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions
DE2860430D1 (en) * 1977-10-08 1981-02-26 Beecham Group Ltd Antithrombotic compositions containing benzisothiazolones
ATE7296T1 (de) * 1979-10-08 1984-05-15 Merck & Co. Inc. 2-aryl-1,2-benzisothiazolinon-1,1-dioxide und sie enthaltende pharmazeutische zusammensetzungen.
DE3226284A1 (de) * 1982-07-14 1984-01-19 A. Nattermann & Cie GmbH, 5000 Köln Neue benzisoselenazolone, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3238006A1 (de) * 1982-10-13 1984-04-19 Bayer Ag, 5090 Leverkusen Azolyl-methylamine, ihre herstellung und verwendung in mikrobiziden mitteln
DE3500577A1 (de) * 1985-01-10 1986-07-10 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 1,2-benzisothiazolonen
US4732984A (en) * 1985-10-17 1988-03-22 American Home Products Corporation Piperazinoisothiazolones with psychotropic activity
DE3617976A1 (de) * 1986-05-28 1988-01-14 Alter Sa 1,4-dihydropyridin, verfahren zu dessen herstellung und dessen verwendung in antithrombotischen medikamenten
US4831031A (en) * 1988-01-22 1989-05-16 Pfizer Inc. Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity
US5128457A (en) * 1988-07-01 1992-07-07 Miles Inc. Chromogenic thiol indicators based on an isobenzothiazolone ring system
CA1340759C (en) * 1988-07-01 1999-09-21 James P. Albarella Isobenzothiazolone chromogenic thiol indicators and their derivatives
US5236917A (en) * 1989-05-04 1993-08-17 Sterling Winthrop Inc. Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
WO2010039545A2 (en) * 2008-09-23 2010-04-08 Georgetown University 1,2-benzisothiazolinone and isoindolinone derivatives
CA2845551C (en) 2011-08-16 2020-06-09 Georgetown University Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives
US20180318818A1 (en) 2015-10-19 2018-11-08 Emory University Redox Dehydration Coupling Catalysts and Methods Related Thereto

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE565380A (es) * 1957-03-08
US3012039A (en) * 1958-03-14 1961-12-05 Ici Ltd 2-p-chlorobenzyl-1, 2-benzisothiazolone
DE1147947B (de) * 1961-07-25 1963-05-02 Knoll Ag Verfahren zur Herstellung neuer 1, 2-Benzisothiazolone
US3661974A (en) * 1970-04-27 1972-05-09 Sherwin Williams Co 2-carbalkoxy-phenyl sulfenamides
SE392103B (sv) * 1970-04-27 1977-03-14 Sherwin Williams Co Sett att framstella 1,2-bensisotiazolin-3-oner
NZ182325A (en) * 1975-11-18 1979-03-16 Beecham Group Ltd 2-substituted-1,2-benzisothiazol-3-ones
GB1582214A (en) * 1977-05-31 1981-01-07 Beecham Group Ltd Antithrombotic compositions
DE2734882A1 (de) * 1977-08-03 1979-02-22 Basf Ag 3- eckige klammer auf 4-(1,3-diazacycloalken-2-yl)-phenyl eckige klammer zu -1,2-benzisothiazole, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
DD127645A5 (es) 1977-10-05
US4350702A (en) 1982-09-21
SU671728A3 (ru) 1979-06-30
AT355017B (de) 1980-02-11
CH627465A5 (de) 1982-01-15
AU4716379A (en) 1979-09-27
SU682129A3 (ru) 1979-08-25
SU679141A3 (ru) 1979-08-05
RO75730A (ro) 1981-02-28
NO763922L (es) 1977-05-20
CS192592B2 (en) 1979-08-31
AU1916376A (en) 1978-05-04
BG24811A3 (en) 1978-05-12
AU520890B2 (en) 1982-03-04
HU173958B (hu) 1979-09-28
PT65851B (en) 1978-05-15
PH13918A (en) 1980-11-04
FI763285A (es) 1977-05-19
NL7612796A (nl) 1977-05-23
CS192570B2 (en) 1979-08-31
IL50690A (en) 1980-01-31
CA1064511A (en) 1979-10-16
FR2332019A1 (fr) 1977-06-17
US4212979A (en) 1980-07-15
IL50690A0 (en) 1976-12-31
AU504599B2 (en) 1979-10-18
BG24808A3 (en) 1978-05-12
JPS5262273A (en) 1977-05-23
AR217411A1 (es) 1980-03-31
AR215271A1 (es) 1979-09-28
RO75777A (ro) 1981-02-28
ATA849176A (de) 1979-07-15
RO69608A (ro) 1982-07-06
US4212872A (en) 1980-07-15
CS192593B2 (en) 1979-08-31
US4243669A (en) 1981-01-06
PT65851A (en) 1976-12-01
ES465173A1 (es) 1978-10-01
DK517776A (da) 1977-05-19
ES453420A1 (es) 1978-02-16
PL193742A1 (pl) 1979-05-21
BE848371A (fr) 1977-05-16
DE2652201A1 (de) 1977-06-02
BG24809A3 (en) 1978-05-12
SE7612919L (sv) 1977-05-19
US4113728A (en) 1978-09-12
BG24810A3 (en) 1978-05-12
RO75540A (ro) 1980-11-30
NZ182325A (en) 1979-03-16
SU701536A3 (ru) 1979-11-30
ZA766489B (en) 1977-10-26
CS192594B2 (en) 1979-08-31
FR2332019B1 (es) 1983-05-20
ES465174A1 (es) 1978-10-01

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