AR199720A1 - Procedimiento para la preparacion de derivados de 3-formilrifamicina "sv" - Google Patents

Procedimiento para la preparacion de derivados de 3-formilrifamicina "sv"

Info

Publication number
AR199720A1
AR199720A1 AR252101A AR25210174A AR199720A1 AR 199720 A1 AR199720 A1 AR 199720A1 AR 252101 A AR252101 A AR 252101A AR 25210174 A AR25210174 A AR 25210174A AR 199720 A1 AR199720 A1 AR 199720A1
Authority
AR
Argentina
Prior art keywords
formylrifamycin
derivatives
procedure
preparation
Prior art date
Application number
AR252101A
Other languages
English (en)
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Application granted granted Critical
Publication of AR199720A1 publication Critical patent/AR199720A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/02Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with oxygen atoms attached in positions 3 and 6, e.g. morphine, morphinone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/09Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems
    • C07D489/10Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14
    • C07D489/12Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14 the bridge containing only two carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR252101A 1972-03-27 1974-01-29 Procedimiento para la preparacion de derivados de 3-formilrifamicina "sv" AR199720A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT2242172 1972-03-27

Publications (1)

Publication Number Publication Date
AR199720A1 true AR199720A1 (es) 1974-09-23

Family

ID=11196065

Family Applications (3)

Application Number Title Priority Date Filing Date
AR246583A AR205434A1 (es) 1972-03-27 1973-01-01 Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv
AR252101A AR199720A1 (es) 1972-03-27 1974-01-29 Procedimiento para la preparacion de derivados de 3-formilrifamicina "sv"
AR252100A AR203839A1 (es) 1972-03-27 1974-01-29 Procedimiento para la preparacion de hidrazonos de 3-formilrifamicia sv

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR246583A AR205434A1 (es) 1972-03-27 1973-01-01 Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR252100A AR203839A1 (es) 1972-03-27 1974-01-29 Procedimiento para la preparacion de hidrazonos de 3-formilrifamicia sv

Country Status (24)

Country Link
US (1) US3865812A (es)
JP (1) JPS5142120B2 (es)
AR (3) AR205434A1 (es)
AT (1) AT322106B (es)
AU (1) AU467606B2 (es)
BE (1) BE797344A (es)
CA (1) CA999858A (es)
CH (1) CH567511A5 (es)
CS (1) CS168642B2 (es)
DD (1) DD104517A5 (es)
DE (1) DE2314478C3 (es)
ES (1) ES413043A1 (es)
FR (1) FR2182906B1 (es)
GB (1) GB1388652A (es)
HU (1) HU167316B (es)
IE (1) IE37817B1 (es)
IL (1) IL41532A0 (es)
LU (1) LU67287A1 (es)
NL (1) NL171360C (es)
PL (1) PL89269B1 (es)
RO (1) RO62882A (es)
SE (1) SE381257B (es)
SU (1) SU497777A3 (es)
ZA (1) ZA73939B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1053787B (it) * 1974-10-29 1981-10-10 Pastori A Macrolidi azotati e loro preparazione
GB1478563A (en) * 1975-03-05 1977-07-06 Lepetit Spa Rifamycin derivatives
DE2728869A1 (de) * 1976-06-25 1977-12-29 Antibiotice Iasi Intreprindere Rifamycinen und verfahren zu deren herstellung
US4179439A (en) * 1977-07-01 1979-12-18 Intreprinderea De Antibiotice Iasi Rifamycins and method for their preparation
JPS5419997A (en) * 1977-07-15 1979-02-15 Intorepurinderea De Anteibiote 33formylrifamycin sv derivative
JPS6025436B2 (ja) * 1977-07-15 1985-06-18 イントレプリンデレア・デ・アンテイビオテイスイアシ 水溶性リフアマイシン
DE2918140C2 (de) * 1979-05-05 1985-02-07 Fresenius AG, 6380 Bad Homburg Dialysator
AU536524B2 (en) * 1979-06-28 1984-05-10 Gruppo Lepetit S.P.A. Water soluble hydrozones of 3-formylifamyan
US4447432A (en) * 1981-11-17 1984-05-08 Farmitalia Carlo Erba S.P.A. Azino rifamycins

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH489520A (fr) * 1964-07-31 1970-04-30 Lepetit Spa Procédé de préparation d'un dérivé de la rifamycine SV
FR208F (es) * 1964-07-31

Also Published As

Publication number Publication date
AT322106B (de) 1975-05-12
AU5342973A (en) 1974-09-19
CH567511A5 (es) 1975-10-15
FR2182906A1 (es) 1973-12-14
LU67287A1 (es) 1973-07-13
JPS5142120B2 (es) 1976-11-13
HU167316B (es) 1975-09-27
GB1388652A (en) 1975-03-26
JPS495998A (es) 1974-01-19
NL171360B (nl) 1982-10-18
AR203839A1 (es) 1975-10-31
DE2314478C3 (de) 1981-01-08
US3865812A (en) 1975-02-11
CA999858A (en) 1976-11-16
SU497777A3 (ru) 1975-12-30
BE797344A (fr) 1973-07-16
PL89269B1 (es) 1976-11-30
CS168642B2 (es) 1976-06-29
NL7304085A (es) 1973-10-01
IE37817B1 (en) 1977-10-26
DD104517A5 (es) 1974-03-12
AU467606B2 (en) 1975-12-04
ATA266074A (de) 1975-06-15
NL171360C (nl) 1983-03-16
ES413043A1 (es) 1976-01-16
DE2314478B2 (de) 1980-04-30
DE2314478A1 (de) 1973-10-04
IE37817L (en) 1973-09-27
RO62882A (fr) 1977-11-15
AR205434A1 (es) 1976-05-07
ZA73939B (en) 1973-11-28
IL41532A0 (en) 1973-04-30
FR2182906B1 (es) 1975-10-31
SE381257B (sv) 1975-12-01

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