DK243676A - Fremgangsmade til fremstilling af pyrrolforbindelser - Google Patents

Fremgangsmade til fremstilling af pyrrolforbindelser

Info

Publication number
DK243676A
DK243676A DK243676A DK243676A DK243676A DK 243676 A DK243676 A DK 243676A DK 243676 A DK243676 A DK 243676A DK 243676 A DK243676 A DK 243676A DK 243676 A DK243676 A DK 243676A
Authority
DK
Denmark
Prior art keywords
preparing
procedure
pyrrol compounds
pyrrol
compounds
Prior art date
Application number
DK243676A
Other languages
English (en)
Other versions
DK154976C (da
DK154976B (da
Inventor
J Carson
Original Assignee
Mcneilab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mcneilab Inc filed Critical Mcneilab Inc
Publication of DK243676A publication Critical patent/DK243676A/da
Publication of DK154976B publication Critical patent/DK154976B/da
Application granted granted Critical
Publication of DK154976C publication Critical patent/DK154976C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/337Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
DK243676A 1975-06-02 1976-06-02 Fremgangsmaade til fremstilling af 5-aroyl-1-laverealkylpyrrol-2-eddikesyrederivater DK154976C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/583,065 US3998844A (en) 1975-06-02 1975-06-02 Uncatalyzed aroylation of 1-alkylpyrrole-2-acetic acid derivatives
US58306575 1975-06-02

Publications (3)

Publication Number Publication Date
DK243676A true DK243676A (da) 1976-12-03
DK154976B DK154976B (da) 1989-01-16
DK154976C DK154976C (da) 1989-06-05

Family

ID=24331553

Family Applications (1)

Application Number Title Priority Date Filing Date
DK243676A DK154976C (da) 1975-06-02 1976-06-02 Fremgangsmaade til fremstilling af 5-aroyl-1-laverealkylpyrrol-2-eddikesyrederivater

Country Status (24)

Country Link
US (1) US3998844A (da)
JP (1) JPS5919536B2 (da)
AT (1) AT358572B (da)
AU (1) AU497557B2 (da)
BE (1) BE842458A (da)
CA (1) CA1066297A (da)
CH (1) CH603578A5 (da)
CS (1) CS220310B2 (da)
DE (2) DE2624557C2 (da)
DK (1) DK154976C (da)
ES (1) ES448408A1 (da)
FR (1) FR2313364A1 (da)
GB (1) GB1477998A (da)
HU (1) HU172047B (da)
IL (1) IL49687A (da)
IN (1) IN141746B (da)
NL (1) NL7605958A (da)
NZ (1) NZ180785A (da)
PL (1) PL101700B1 (da)
PT (1) PT65161B (da)
RO (1) RO69252A (da)
SE (1) SE414765B (da)
YU (1) YU40648B (da)
ZA (1) ZA763191B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4048191A (en) * 1975-06-27 1977-09-13 Mcneil Laboratories, Incorporated Halo-substituted 1-loweralkyl-5-aroylpyrrole-2-acetic acid compounds
US4207237A (en) * 1977-04-20 1980-06-10 Mcneilab, Inc. Preparation of pyrrole-2-acetates
US4200645A (en) * 1977-05-10 1980-04-29 Beecham Group Limited Pyrrole derivatives
US4119639A (en) * 1977-06-27 1978-10-10 Mcneil Laboratories, Incorporated Preparation of 5-aroylpyrrole-2-acetic acid derivatives
GB1592996A (en) * 1977-10-10 1981-07-15 Rolland Sa A Acylated pyrrole carboxylic acids and derivatives thereof
JPS5481264A (en) * 1977-12-08 1979-06-28 Sagami Chem Res Center Preparation of 1-methyl-5-aroylpryrrole-2-acetic acid
SE435278B (sv) * 1977-12-08 1984-09-17 Sagami Chem Res 5-cyano-1-legre(c?711?71-?714)alkyl-pyrrol-2-ettiksyra, framstellning derav och anvendningen som mellanprodukt vid framstellning av terapeutiskt verksamma pyrrolderivat
US4216150A (en) * 1978-10-16 1980-08-05 Mcneil Lab, Inc. Preparation of pyrrole-2-acetates
US4213905A (en) * 1979-06-25 1980-07-22 Mcneilab, Inc. Preparation of 5-aroyl-1-loweralkylpyrrole-2-acetic acid salts
US4284562A (en) * 1979-11-27 1981-08-18 Mcneilab, Inc. Process for preparing pyrrole-2-acetic acids
US4255335A (en) * 1980-04-03 1981-03-10 Mcneilab, Inc. Preparation of 5-aroyl-1-loweralkylpyrrole-2-acetic acid derivatives
US4299770A (en) * 1980-05-29 1981-11-10 Mallinckrodt, Inc. Recovery of substituted pyrrole acetate
NZ201468A (en) * 1981-08-10 1986-02-21 Merck & Co Inc 5-aroyl-4-pyrrolyl-alkanoic acid derivatives and pharmaceutical compositions
US5418236A (en) * 1993-12-23 1995-05-23 Ortho Pharmaceutical Corporation Anxiolytic aroyl piperidinyl and piperazinylacyl pyrroles
US6441194B1 (en) 1999-10-21 2002-08-27 Emory University Synthesis of 4-substituted pyrrole-2-carbaldehyde compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3752826A (en) * 1970-01-26 1973-08-14 Mcneilab Inc Aroyl substituted pyrroles
US3846447A (en) * 1972-08-03 1974-11-05 Mcneilab Inc Preparation of 5-aroyl-pyrroles and intermediates therefor

Also Published As

Publication number Publication date
NZ180785A (en) 1978-03-06
PT65161B (en) 1978-07-03
BE842458A (fr) 1976-12-01
DK154976C (da) 1989-06-05
US3998844A (en) 1976-12-27
RO69252A (ro) 1981-08-30
DE2624557A1 (de) 1976-12-23
GB1477998A (en) 1977-06-29
DE2624557C2 (de) 1984-04-05
PT65161A (en) 1976-06-01
YU40648B (en) 1986-04-30
JPS5919536B2 (ja) 1984-05-07
ES448408A1 (es) 1977-11-16
DE2624558A1 (de) 1976-12-23
FR2313364A1 (fr) 1976-12-31
SE414765B (sv) 1980-08-18
IL49687A (en) 1978-10-31
YU136076A (en) 1982-05-31
JPS51143664A (en) 1976-12-10
CA1066297A (en) 1979-11-13
HU172047B (hu) 1978-05-28
AU1440576A (en) 1977-12-01
FR2313364B1 (da) 1980-09-12
PL101700B1 (pl) 1979-01-31
ATA401476A (de) 1980-02-15
NL7605958A (nl) 1976-12-06
SE7606165L (sv) 1976-12-03
AT358572B (de) 1980-09-25
DK154976B (da) 1989-01-16
IL49687A0 (en) 1976-07-30
ZA763191B (en) 1978-01-25
CH603578A5 (da) 1978-08-31
CS220310B2 (en) 1983-03-25
AU497557B2 (en) 1978-12-14
IN141746B (da) 1977-04-09

Similar Documents

Publication Publication Date Title
DK143706C (da) Fremgangsmaade til fremstilling af svovlholdige organosiliciumforbindelser
DK494876A (da) Fremgangsmade til fremstilling af piperidinderivater
DK365176A (da) Fremgangsmade til fremstilling af pyrrolidinderivater
DK484576A (da) Fremgangsmade til fremstilling af 2-aroyl-3-phenyl-benzothiophenforbindelser
DK562376A (da) Fremgangsmade til fremstilling af ergolinderivater
DK442476A (da) Fremgangsmade til fremstilling af pyrimidinforbindelser
DK462376A (da) Fremgangsmade til fremstilling af 5-halogenpyrimidinderivater
DK517776A (da) Fremgangsmade til femstilling af heterocycliske forbindelser
DK243176A (da) Fremgangsmade til fremstilling af polycliske forbindelser
DK243676A (da) Fremgangsmade til fremstilling af pyrrolforbindelser
DK415676A (da) Fremgangsmade til fremstilling af pilocarpiniumsalte
DK473976A (da) Fremgangsmade til fremstilling af partikelformede detergenter
DK272676A (da) Fremgangsmade til fremstilling af cephalosporinforbindelser
DK164476A (da) Fremgangsmade til fremstilling af piperazinylpyrazinforbindelser
DK215676A (da) Fremgangsmade til fremstilling af rifamycinforbindelser
DK324776A (da) Fremgangsmade til fremstilling af 3-cyanoimino-3-aminopropionitriler
DK372576A (da) Fremgangsmade til fremstilling af polyaminforbindelser
DK305876A (da) Fremgangsmade til fremstilling af l-pyroglutamyl-l-prolinamid
DK220276A (da) Fremgangsmade til fremstilling af rifamycinforbindelser
DK155598C (da) Fremgangsmaade til fremstilling af ethylchlorthioformiat
DK143281C (da) Fremgangsmaade til fremstilling af phosphitchlorider
DK143137C (da) Fremgangsmaade til fremstilling af phosphitchlorider
DK511376A (da) Fremgangsmade til fremstilling af imidazolforbindelser
DK527476A (da) Fremgangsmade til fremstilling af organiske forbindelser
DK509076A (da) Fremgangsmade til fremstilling af rifamycinforbindelser