DK2678327T3 - Heteroaryl derivatives which ALFA7 nAChR modulators - Google Patents

Heteroaryl derivatives which ALFA7 nAChR modulators Download PDF

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Publication number
DK2678327T3
DK2678327T3 DK12709965.3T DK12709965T DK2678327T3 DK 2678327 T3 DK2678327 T3 DK 2678327T3 DK 12709965 T DK12709965 T DK 12709965T DK 2678327 T3 DK2678327 T3 DK 2678327T3
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alkyl
methyl
optionally substituted
group
benzenesulfonamide
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DK12709965.3T
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Danish (da)
English (en)
Inventor
Neelima Sinha
Gourhari Jana
Sachchidanand Sachchidanand
Sanjay Pralhad Kurhade
Navnath Popat Karche
Anil Kashiram Hajare
Ajay Ramchandra Tilekar
Venkata P Palle
Rajender Kumar Kamboj
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Lupin Ltd
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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DK12709965.3T 2011-02-23 2012-02-22 Heteroaryl derivatives which ALFA7 nAChR modulators DK2678327T3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN242KO2011 2011-02-23
IN1184KO2011 2011-09-09
PCT/IB2012/050806 WO2012114285A1 (en) 2011-02-23 2012-02-22 Heteroaryl derivatives as alpha7 nachr modulators

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DK2678327T3 true DK2678327T3 (en) 2016-12-12

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US (2) US9072731B2 (enExample)
EP (1) EP2678327B9 (enExample)
JP (1) JP6118270B2 (enExample)
KR (1) KR20140026378A (enExample)
CN (1) CN103402994B (enExample)
AP (1) AP3649A (enExample)
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