FR2840303B1 - Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile - Google Patents

Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile

Info

Publication number
FR2840303B1
FR2840303B1 FR0206717A FR0206717A FR2840303B1 FR 2840303 B1 FR2840303 B1 FR 2840303B1 FR 0206717 A FR0206717 A FR 0206717A FR 0206717 A FR0206717 A FR 0206717A FR 2840303 B1 FR2840303 B1 FR 2840303B1
Authority
FR
France
Prior art keywords
vinylation
arylation
alkylation
nucleophilic compound
nucleophilic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0206717A
Other languages
English (en)
Other versions
FR2840303A1 (fr
Inventor
Marc Taillefer
Henri Jean Cristau
Pascal Cellier
Jean Francis Spindler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhodia Chimie SAS
Original Assignee
Rhodia Chimie SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US10/159,829 priority Critical patent/US7202367B2/en
Application filed by Rhodia Chimie SAS filed Critical Rhodia Chimie SAS
Priority to FR0206717A priority patent/FR2840303B1/fr
Priority to EP03756038A priority patent/EP1509502A1/fr
Priority to JP2004509659A priority patent/JP2006501159A/ja
Priority to AU2003255620A priority patent/AU2003255620A1/en
Priority to CNA038166712A priority patent/CN1668595A/zh
Priority to US10/515,856 priority patent/US20050234239A1/en
Priority to PCT/FR2003/001647 priority patent/WO2003101966A1/fr
Priority to CA002487475A priority patent/CA2487475A1/fr
Publication of FR2840303A1 publication Critical patent/FR2840303A1/fr
Application granted granted Critical
Publication of FR2840303B1 publication Critical patent/FR2840303B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
    • C07D213/53—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FR0206717A 2002-03-31 2002-05-31 Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile Expired - Fee Related FR2840303B1 (fr)

Priority Applications (9)

Application Number Priority Date Filing Date Title
FR0206717A FR2840303B1 (fr) 2002-05-31 2002-05-31 Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile
US10/159,829 US7202367B2 (en) 2002-05-31 2002-05-31 Process for arylating or vinylating or alkynating a nucleophilic compound
JP2004509659A JP2006501159A (ja) 2002-05-31 2003-06-02 炭素−炭素結合又は炭素−ヘテロ原子結合の形成方法
AU2003255620A AU2003255620A1 (en) 2002-05-31 2003-06-02 Method of forming a carbon-carbon or carbon-heteroatom linkage
EP03756038A EP1509502A1 (fr) 2002-05-31 2003-06-02 Procede de formation d une liaison carbone-carbone ou carbone-heteroatome
CNA038166712A CN1668595A (zh) 2002-05-31 2003-06-02 形成碳－碳或碳－杂原子键的方法
US10/515,856 US20050234239A1 (en) 2002-03-31 2003-06-02 Method of forming a carbon-carbon or carbon-heteroatom linkage
PCT/FR2003/001647 WO2003101966A1 (fr) 2002-05-31 2003-06-02 Procede de formation d'une liaison carbone-carbone ou carbone-heteroatome
CA002487475A CA2487475A1 (fr) 2002-05-31 2003-06-02 Procede de formation d'une liaison carbone-carbone ou carbone-heteroatome

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0206717A FR2840303B1 (fr) 2002-05-31 2002-05-31 Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile
US10/159,829 US7202367B2 (en) 2002-05-31 2002-05-31 Process for arylating or vinylating or alkynating a nucleophilic compound

Publications (2)

Publication Number Publication Date
FR2840303A1 FR2840303A1 (fr) 2003-12-05
FR2840303B1 true FR2840303B1 (fr) 2005-07-15

Family

ID=32232264

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0206717A Expired - Fee Related FR2840303B1 (fr) 2002-03-31 2002-05-31 Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile

Country Status (3)

Country Link
US (1) US7202367B2 (fr)
FR (1) FR2840303B1 (fr)
WO (1) WO2003101966A1 (fr)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004039280A1 (de) * 2004-08-13 2006-02-23 Merck Patent Gmbh 1,5-Diphenyl-pyrazole
GT200600207A (es) * 2005-06-09 2007-01-15 Novartis Ag Proceso para la síntesis de compuestos orgánicos
SA06270147B1 (ar) 2005-06-09 2009-12-22 نوفارتيس ايه جي عملية لتخليق 5-(مثيل–1h–إيميدازول–1-يل )–3-(ثلاثي فلـورو مثيل)–بنزامـين
JP2006342127A (ja) * 2005-06-10 2006-12-21 Koei Chem Co Ltd アリールピラゾール類の製造法
US9162953B2 (en) * 2006-07-05 2015-10-20 Centre Nationale De Recherche Scientifique Iron-copper co-catalyzed process for carbon-carbon or carbon-heteroatom bonding
US8034815B2 (en) 2007-01-11 2011-10-11 Critical Outcome Technologies, Inc. Compounds and method for treatment of cancer
FR2915200B1 (fr) * 2007-04-20 2009-07-03 Centre Nat Rech Scient Procede de preparation de ligands de type phosphines butadieniques,leurs complexes avec le cuivre,et leurs applications en catalyse
FR2921659B1 (fr) * 2007-09-28 2013-01-18 Centre Nat Rech Scient Utilisation de complexes cuivre/phosphines cyclovinyliques comme catalyseurs d'arylation
WO2009071997A2 (fr) 2007-12-06 2009-06-11 Centre National De La Recherche Scientifique (C.N.R.S.) Nouveau système catalytique pour réaction de couplage croisé
CA2710039C (fr) 2007-12-26 2018-07-03 Critical Outcome Technologies, Inc. Semicarbazones, thiosemicarnazones et composes associes, et methodes de traitement du cancer
CA2730890C (fr) 2008-07-17 2018-05-15 Critical Outcome Technologies Inc. Composes inhibiteurs et procedes de traitement du cancer
WO2010072632A1 (fr) * 2008-12-24 2010-07-01 Syngenta Limited Procedes de preparation d'arylamides
CA2794952C (fr) 2010-04-01 2018-05-15 Critical Outcome Technologies Inc. Composes et methodes pour le traitement du vih
WO2012114285A1 (fr) 2011-02-23 2012-08-30 Lupin Limited Dérivés hétéroaryle à titre de modulateurs des nachr alpha 7
US9388196B2 (en) 2012-03-06 2016-07-12 Lupin Limited Thiazole derivatives as alpha 7 nAChR modulators
WO2014060381A1 (fr) 2012-10-18 2014-04-24 Bayer Cropscience Ag Composés hétérocycliques pour la lutte contre les nuisibles
WO2014067962A1 (fr) 2012-10-31 2014-05-08 Bayer Cropscience Ag Nouveaux composés hétérocycliques utilisés comme agents de lutte contre les nuisibles
US9231217B2 (en) * 2013-11-28 2016-01-05 Semiconductor Energy Laboratory Co., Ltd. Synthesis method of organometallic complex, synthesis method of pyrazine derivative, 5,6-diaryl-2-pyrazyl triflate, light-emitting element, light-emitting device, electronic device, and lighting device
CN116969925A (zh) 2018-04-12 2023-10-31 拜耳公司 杂芳基-三唑化合物
CN112645909A (zh) * 2021-01-25 2021-04-13 苏州大学 一种合成α-苄基苯并呋喃类化合物的方法
CN114149364A (zh) * 2021-12-21 2022-03-08 无锡捷化医药科技有限公司 一种n-(6-甲氧基吡啶-3-基)-3-甲基吡啶-2-磺酰胺的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002085838A1 (fr) * 2001-04-24 2002-10-31 Massachusetts Institute Of Technology Formation par catalyse de cuivre de liaisons carbone-heteroatome et carbone-carbone

Also Published As

Publication number Publication date
WO2003101966A1 (fr) 2003-12-11
FR2840303A1 (fr) 2003-12-05
US20030236413A1 (en) 2003-12-25
US7202367B2 (en) 2007-04-10

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Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20080131