DK2280962T5 - Pyridazinonderivater - Google Patents

Pyridazinonderivater

Info

Publication number
DK2280962T5
DK2280962T5 DK09734854.4T DK09734854T DK2280962T5 DK 2280962 T5 DK2280962 T5 DK 2280962T5 DK 09734854 T DK09734854 T DK 09734854T DK 2280962 T5 DK2280962 T5 DK 2280962T5
Authority
DK
Denmark
Prior art keywords
pyridazinone
Prior art date
Application number
DK09734854.4T
Other languages
Danish (da)
English (en)
Other versions
DK2280962T3 (da
Inventor
Dieter Dorsch
Oliver Schadt
Frank Stieber
Andree Blaukat
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of DK2280962T3 publication Critical patent/DK2280962T3/da
Application granted granted Critical
Publication of DK2280962T5 publication Critical patent/DK2280962T5/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK09734854.4T 2008-04-21 2009-03-24 Pyridazinonderivater DK2280962T5 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102008019907A DE102008019907A1 (de) 2008-04-21 2008-04-21 Pyridazinonderivate
PCT/EP2009/002137 WO2009129905A1 (de) 2008-04-21 2009-03-24 Pyridazinonderivate

Publications (2)

Publication Number Publication Date
DK2280962T3 DK2280962T3 (da) 2012-11-19
DK2280962T5 true DK2280962T5 (da) 2013-09-16

Family

ID=40639931

Family Applications (1)

Application Number Title Priority Date Filing Date
DK09734854.4T DK2280962T5 (da) 2008-04-21 2009-03-24 Pyridazinonderivater

Country Status (22)

Country Link
US (1) US8604036B2 (enExample)
EP (1) EP2280962B1 (enExample)
JP (1) JP5576358B2 (enExample)
KR (1) KR20100137564A (enExample)
CN (1) CN102015694A (enExample)
AR (1) AR071208A1 (enExample)
AU (1) AU2009240346B2 (enExample)
BR (1) BRPI0911161B8 (enExample)
CA (1) CA2721858C (enExample)
CY (1) CY1113443T1 (enExample)
DE (1) DE102008019907A1 (enExample)
DK (1) DK2280962T5 (enExample)
EA (1) EA018362B1 (enExample)
ES (1) ES2394147T3 (enExample)
HR (1) HRP20120884T1 (enExample)
IL (1) IL208336A (enExample)
MX (1) MX2010011454A (enExample)
PL (1) PL2280962T3 (enExample)
PT (1) PT2280962E (enExample)
SI (1) SI2280962T1 (enExample)
WO (1) WO2009129905A1 (enExample)
ZA (1) ZA201008330B (enExample)

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DE102007032507A1 (de) 2007-07-12 2009-04-02 Merck Patent Gmbh Pyridazinonderivate
DE102007038957A1 (de) * 2007-08-17 2009-02-19 Merck Patent Gmbh 6-Thioxo-pyridazinderivate
DE102007061963A1 (de) 2007-12-21 2009-06-25 Merck Patent Gmbh Pyridazinonderivate
DE102008019907A1 (de) 2008-04-21 2009-10-22 Merck Patent Gmbh Pyridazinonderivate
DE102008028905A1 (de) * 2008-06-18 2009-12-24 Merck Patent Gmbh 3-(3-Pyrimidin-2-yl-benzyl)-[1,2,4]triazolo[4,3-b]pyridazinderivate
DE102008037790A1 (de) * 2008-08-14 2010-02-18 Merck Patent Gmbh Bicyclische Triazolderivate
DK2361250T3 (da) 2008-12-22 2013-11-04 Merck Patent Gmbh Nye polymorfe former af 6-(1-methyl-1h-pyrazol-4-yl)-2-{3-[5-(2-morpholin-4-yl-ethoxy)-pyrimidin-2-yl]-benzyl}-2h-pyridazin-3-on-dihydrogenphosphat og fremgangsmåder til fremstilling deraf
CN102532126B (zh) * 2012-02-10 2014-06-18 贵州大学 2-取代-4-氯-5-[5-取代胺基-2-(1,3,4-噻二唑基)-巯基]-3(2h)-哒嗪酮类衍生物及其制备方法和用途
EP3532467A1 (en) * 2016-10-26 2019-09-04 Proteostasis Therapeutics, Inc. Pyridazine derivatives, compositions and methods for modulating cftr
JP7274473B2 (ja) 2017-10-17 2023-05-16 パラウ ファルマ，エス．エル．ユー． ４－アミノピリミジン化合物の合成
CN108752322A (zh) * 2018-09-12 2018-11-06 广州新民培林医药科技有限公司 一种新型Tepotinib衍生物和制备方法及其在抗肿瘤药物中的应用
CN113272014A (zh) 2018-11-06 2021-08-17 艾知怀斯治疗学公司 哒嗪酮化合物及其用途
JP7671245B2 (ja) 2018-11-06 2025-05-01 エッジワイズ セラピューティクス， インコーポレイテッド ピリダジノン化合物およびその使用
WO2020097266A1 (en) 2018-11-06 2020-05-14 Edgewise Therapeutics, Inc. Pyridazinone compounds and uses thereof
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
EP4053123A4 (en) 2019-11-01 2023-10-11 Unimatec Co., Ltd. FLUORINATED PYRIMIDINE COMPOUND AND METHOD FOR THE PRODUCTION THEREOF

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Also Published As

Publication number Publication date
EA201001648A1 (ru) 2011-06-30
BRPI0911161A2 (pt) 2015-10-06
CY1113443T1 (el) 2016-06-22
ZA201008330B (en) 2011-09-28
MX2010011454A (es) 2010-12-21
AU2009240346A1 (en) 2009-10-29
SI2280962T1 (sl) 2013-01-31
CA2721858C (en) 2016-07-19
PT2280962E (pt) 2012-12-17
DE102008019907A1 (de) 2009-10-22
CN102015694A (zh) 2011-04-13
EP2280962B1 (de) 2012-10-03
US20110034474A1 (en) 2011-02-10
HRP20120884T1 (hr) 2012-11-30
AR071208A1 (es) 2010-06-02
CA2721858A1 (en) 2009-10-29
IL208336A (en) 2016-07-31
EA018362B1 (ru) 2013-07-30
BRPI0911161B8 (pt) 2021-05-25
US8604036B2 (en) 2013-12-10
DK2280962T3 (da) 2012-11-19
ES2394147T3 (es) 2013-01-22
AU2009240346B2 (en) 2013-10-10
JP5576358B2 (ja) 2014-08-20
BRPI0911161B1 (pt) 2020-02-11
WO2009129905A1 (de) 2009-10-29
IL208336A0 (en) 2010-12-30
EP2280962A1 (de) 2011-02-09
PL2280962T3 (pl) 2013-02-28
KR20100137564A (ko) 2010-12-30
JP2011518202A (ja) 2011-06-23

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