DK2076491T3 - Nye benzamidderivater som bradykininantagonister - Google Patents

Nye benzamidderivater som bradykininantagonister

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Publication number
DK2076491T3
DK2076491T3 DK07824994.3T DK07824994T DK2076491T3 DK 2076491 T3 DK2076491 T3 DK 2076491T3 DK 07824994 T DK07824994 T DK 07824994T DK 2076491 T3 DK2076491 T3 DK 2076491T3
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Prior art keywords
benzamide derivatives
bradykinin antagonists
new benzamide
new
bradykinin
Prior art date
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DK07824994.3T
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English (en)
Inventor
Istvan Vago
Eva Bozo
Sandor Farkas
Katalin Hornok
Monika Vastag
Gyula Beke
Gyoergy Keserue
Eva Schmidt
Eva Szentirmay
Original Assignee
Richter Gedeon Nyrt
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Publication of DK2076491T3 publication Critical patent/DK2076491T3/da

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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DK07824994.3T 2006-10-27 2007-10-27 Nye benzamidderivater som bradykininantagonister DK2076491T3 (da)

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HUP0600810A3 (en) * 2006-10-27 2008-09-29 Richter Gedeon Nyrt New sulfonamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them
US20100298299A1 (en) * 2007-10-27 2010-11-25 Istvan Vago non-peptide derivatives as bradykinin b1 antagonists
AU2009282822A1 (en) * 2008-08-21 2010-02-25 Richter Gedeon Nyrt. Methods for treating CNS disorders
US20100048629A1 (en) * 2008-08-21 2010-02-25 Allyson Gage Methods for treating neuropathic pain
JP5629274B2 (ja) * 2009-02-26 2014-11-19 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ブラジキニンｂ１アンタゴニストとしての化合物
ES2350077B1 (es) 2009-06-04 2011-11-04 Laboratorios Salvat, S.A. Compuestos inhibidores de 11beta-hidroxiesteroide deshidrogenasa de tipo 1.
US8912221B2 (en) * 2010-12-27 2014-12-16 Hoffmann-La Roche Inc. Biaryl amide derivatives
JP6592008B2 (ja) * 2014-04-23 2019-10-16 エックス−アールエックス， インコーポレイテッド オートタキシンの置換ｎ−（２−アミノ）−２−オキソエチルベンズアミド阻害剤およびそれらの調製、ならびにｌｐａ依存性またはｌｐａ媒介性疾患の処置における使用
KR101676850B1 (ko) 2015-04-23 2016-11-18 한일화섬 주식회사 내구성이 우수한 스피커용 댐퍼 및 그 제조 방법
TW202202495A (zh) 2020-03-26 2022-01-16 匈牙利商羅特格登公司 作為ｇａｍｍａ－胺基丁酸Ａ受體次單元ａｌｐｈａ ５受體調節劑之㖠啶及吡啶并〔３，４－ｃ〕嗒𠯤衍生物
HUP2100338A1 (hu) 2021-09-29 2023-04-28 Richter Gedeon Nyrt GABAA ALFA5 receptor modulátor hatású biciklusos aminszármazékok

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HUP0600809A3 (en) 2006-10-27 2008-09-29 Richter Gedeon Nyrt New phenylsulfamoyl-benzamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them
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US20100048629A1 (en) 2008-08-21 2010-02-25 Allyson Gage Methods for treating neuropathic pain
CN102884428A (zh) 2010-01-26 2013-01-16 里奇诊断学股份有限公司 对疾病严重度分级和检测抑郁治疗的多个生物标记组

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HUP0600808A2 (en) 2008-08-28
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