DK175824B1 - Styrylpyrazoler,-isoxazoler og analoge forbindelser farmaceutiske præparater med aktivitet mod 5-lipoxygenase eller cyclooxygenase eller............ - Google Patents

Styrylpyrazoler,-isoxazoler og analoge forbindelser farmaceutiske præparater med aktivitet mod 5-lipoxygenase eller cyclooxygenase eller............ Download PDF

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Publication number
DK175824B1
DK175824B1 DK198702269A DK226987A DK175824B1 DK 175824 B1 DK175824 B1 DK 175824B1 DK 198702269 A DK198702269 A DK 198702269A DK 226987 A DK226987 A DK 226987A DK 175824 B1 DK175824 B1 DK 175824B1
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defined above
hydroxy
compound
ethenyl
independently
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DK198702269A
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Danish (da)
English (en)
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DK226987D0 (da
DK226987A (da
Inventor
Daniel L Flynn
David T Connor
Thomas R Belliotti
Catherine R Kostlan
Donald E Nies
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Warner Lambert Co
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Publication of DK226987A publication Critical patent/DK226987A/da
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07F9/653—Five-membered rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
DK198702269A 1986-05-09 1987-05-04 Styrylpyrazoler,-isoxazoler og analoge forbindelser farmaceutiske præparater med aktivitet mod 5-lipoxygenase eller cyclooxygenase eller............ DK175824B1 (da)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US86117986A 1986-05-09 1986-05-09
US86117986 1986-05-09
US91069286A 1986-09-22 1986-09-22
US91069286 1986-09-22
US3273087A 1987-04-06 1987-04-06
US3273087 1987-04-06

Publications (3)

Publication Number Publication Date
DK226987D0 DK226987D0 (da) 1987-05-04
DK226987A DK226987A (da) 1987-11-10
DK175824B1 true DK175824B1 (da) 2005-03-14

Family

ID=27364200

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198702269A DK175824B1 (da) 1986-05-09 1987-05-04 Styrylpyrazoler,-isoxazoler og analoge forbindelser farmaceutiske præparater med aktivitet mod 5-lipoxygenase eller cyclooxygenase eller............

Country Status (15)

Country Link
US (1) US5208251A (xx)
EP (1) EP0245825B1 (xx)
JP (1) JP2656035B2 (xx)
KR (1) KR870011113A (xx)
AT (1) ATE61582T1 (xx)
AU (1) AU613579B2 (xx)
DE (1) DE3768553D1 (xx)
DK (1) DK175824B1 (xx)
ES (1) ES2037681T3 (xx)
FI (1) FI872015A (xx)
GR (1) GR3001831T3 (xx)
IE (1) IE59813B1 (xx)
NO (1) NO871917L (xx)
NZ (1) NZ220248A (xx)
PT (1) PT84840B (xx)

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JP5063351B2 (ja) * 2004-09-17 2012-10-31 エグゼリクシス， インコーポレイテッド ピラゾールキナーゼモジュレーターおよび使用方法
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Also Published As

Publication number Publication date
PT84840B (pt) 1990-02-08
ES2037681T3 (es) 1993-07-01
DK226987D0 (da) 1987-05-04
FI872015A (fi) 1987-11-10
DK226987A (da) 1987-11-10
EP0245825B1 (en) 1991-03-13
GR3001831T3 (en) 1992-11-23
US5208251A (en) 1993-05-04
IE871041L (en) 1987-11-09
KR870011113A (ko) 1987-12-21
AU613579B2 (en) 1991-08-08
ATE61582T1 (de) 1991-03-15
NO871917L (no) 1987-11-10
PT84840A (en) 1987-06-01
JP2656035B2 (ja) 1997-09-24
FI872015A0 (fi) 1987-05-06
DE3768553D1 (de) 1991-04-18
AU7197387A (en) 1987-11-12
NO871917D0 (no) 1987-05-08
EP0245825A1 (en) 1987-11-19
JPS6322079A (ja) 1988-01-29
NZ220248A (en) 1989-05-29
IE59813B1 (en) 1994-04-06

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