DK172949B1 - Synergistinderivater, deres fremstilling og farmaceutiske præparater deraf - Google Patents

Synergistinderivater, deres fremstilling og farmaceutiske præparater deraf Download PDF

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Publication number
DK172949B1
DK172949B1 DK198702585A DK258587A DK172949B1 DK 172949 B1 DK172949 B1 DK 172949B1 DK 198702585 A DK198702585 A DK 198702585A DK 258587 A DK258587 A DK 258587A DK 172949 B1 DK172949 B1 DK 172949B1
Authority
DK
Denmark
Prior art keywords
group
pristinamycin
isomer
general formula
alkyl
Prior art date
Application number
DK198702585A
Other languages
Danish (da)
English (en)
Other versions
DK258587A (da
DK258587D0 (da
Inventor
Claude Cotrel
Jean-Claude Barriere
Jean-Marc Paris
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Publication of DK258587D0 publication Critical patent/DK258587D0/da
Publication of DK258587A publication Critical patent/DK258587A/da
Application granted granted Critical
Publication of DK172949B1 publication Critical patent/DK172949B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/19—Antibiotic
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/27—Cyclic peptide or cyclic protein

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Lubricants (AREA)
  • Vibration Prevention Devices (AREA)
  • Measurement Of Force In General (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Polarising Elements (AREA)
DK198702585A 1986-05-22 1987-05-21 Synergistinderivater, deres fremstilling og farmaceutiske præparater deraf DK172949B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8607270A FR2599036B1 (fr) 1986-05-22 1986-05-22 Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR8607270 1986-05-22

Publications (3)

Publication Number Publication Date
DK258587D0 DK258587D0 (da) 1987-05-21
DK258587A DK258587A (da) 1987-11-23
DK172949B1 true DK172949B1 (da) 1999-10-11

Family

ID=9335470

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198702585A DK172949B1 (da) 1986-05-22 1987-05-21 Synergistinderivater, deres fremstilling og farmaceutiske præparater deraf

Country Status (25)

Country Link
US (1) US4798827A (de)
EP (1) EP0248703B1 (de)
JP (2) JP2558282B2 (de)
KR (1) KR950001020B1 (de)
AT (1) ATE63563T1 (de)
AU (1) AU601426B2 (de)
BR (1) BR1101133A (de)
CA (1) CA1271297A (de)
DE (2) DE10075012I2 (de)
DK (1) DK172949B1 (de)
ES (1) ES2032457T3 (de)
FI (1) FI84355C (de)
FR (1) FR2599036B1 (de)
GE (1) GEP19960474B (de)
GR (1) GR3002558T3 (de)
IE (1) IE60656B1 (de)
IL (1) IL82564A (de)
LU (1) LU90732I2 (de)
LV (1) LV5268A3 (de)
MX (1) MX9203577A (de)
NL (1) NL300010I2 (de)
NZ (1) NZ220380A (de)
PT (1) PT84934B (de)
SU (1) SU1616520A3 (de)
ZA (1) ZA873639B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2664894A1 (fr) * 1990-07-19 1992-01-24 Rhone Poulenc Sante Nouveaux derives de streptogramines et leur preparation.
FR2689518B1 (fr) * 1992-04-01 1995-04-07 Rhone Poulenc Rorer Sa Microorganismes, procédé de préparation et utilisation.
US5242938A (en) * 1992-08-27 1993-09-07 Merck & Co., Inc. Derivatives of virginiamycin M1
IL121821A (en) * 1993-02-17 2000-02-17 Rhone Poulenc Rorer Sa Process for purifying a group A minority component of streptogramin some such purified components and their uses
FR2723373B1 (fr) 1994-08-02 1996-09-13 Rhone Poulenc Rorer Sa Forme purifiee de streptogramines, sa preparation et les compositions pharmaceutiques qui la contiennent
FR2755857B1 (fr) * 1996-11-19 1998-12-24 Rhone Poulenc Rorer Sa Compositions pharmaceutiques stabilisees, a base de quinupristine et de dalfopristine et leur preparation
FR2766489B1 (fr) 1997-07-28 1999-08-27 Rhone Poulenc Rorer Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
US6187746B1 (en) * 1997-12-16 2001-02-13 Rhone-Poulenc Rorer S.A. Pharmaceutical compositions based on dalfopristine and on quinupristine, and preparation thereof
FR2796949B1 (fr) * 1999-07-27 2001-09-21 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2549064B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines utiles pour la preparation de nouveaux medicaments antimicrobiens et leur preparation
FR2549065B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2549063B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2549062B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2576022B1 (fr) * 1985-01-11 1987-09-11 Rhone Poulenc Sante Nouveaux derives de la pristinamycine ii b, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
IL82564A (en) 1991-04-15
AU601426B2 (en) 1990-09-13
DK258587A (da) 1987-11-23
GR3002558T3 (en) 1993-01-25
ATE63563T1 (de) 1991-06-15
LV5268A3 (lv) 1993-10-10
FR2599036B1 (fr) 1988-09-09
MX9203577A (es) 1992-09-01
DE10075012I1 (de) 2000-08-31
JPH08319236A (ja) 1996-12-03
AU7323987A (en) 1987-11-26
EP0248703B1 (de) 1991-05-15
NL300010I2 (nl) 2001-01-02
NL300010I1 (nl) 2000-08-01
CA1271297A (fr) 1990-07-03
FI84355C (fi) 1991-11-25
LU90732I2 (en) 2001-04-17
IE871317L (en) 1987-11-22
FI872236A (fi) 1987-11-23
SU1616520A3 (ru) 1990-12-23
JPS6322095A (ja) 1988-01-29
GEP19960474B (en) 1996-07-22
BR1101133A (pt) 1999-12-07
IE60656B1 (en) 1994-08-10
DE10075012I2 (de) 2006-02-02
KR880013934A (ko) 1988-12-22
FI872236A0 (fi) 1987-05-21
US4798827A (en) 1989-01-17
KR950001020B1 (ko) 1995-02-07
DE3770048D1 (de) 1991-06-20
EP0248703A1 (de) 1987-12-09
JP2659531B2 (ja) 1997-09-30
IL82564A0 (en) 1987-11-30
DK258587D0 (da) 1987-05-21
ES2032457T3 (es) 1993-02-16
ZA873639B (en) 1987-11-17
PT84934A (fr) 1987-06-01
NZ220380A (en) 1989-02-24
JP2558282B2 (ja) 1996-11-27
FI84355B (fi) 1991-08-15
PT84934B (pt) 1990-02-08
FR2599036A1 (fr) 1987-11-27

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
CTFF Application for supplementary protection certificate (spc) filed

Free format text: CA 2000 00016, 20000818, EXPIRES: 20120521