DK169073B1 - (4-piperidinylmethyl og -hetero)puriner, præparater indeholdende disse samt fremgangsmåde til fremstilling af disse purinforbindelser - Google Patents

(4-piperidinylmethyl og -hetero)puriner, præparater indeholdende disse samt fremgangsmåde til fremstilling af disse purinforbindelser Download PDF

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Publication number
DK169073B1
DK169073B1 DK295286A DK295286A DK169073B1 DK 169073 B1 DK169073 B1 DK 169073B1 DK 295286 A DK295286 A DK 295286A DK 295286 A DK295286 A DK 295286A DK 169073 B1 DK169073 B1 DK 169073B1
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Prior art keywords
formula
compound
parts
methyl
group
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DK295286A
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Danish (da)
English (en)
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DK295286D0 (da
DK295286A (da
Inventor
Frans Eduard Janssens
Gaston Stanislas Marcell Diels
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Janssen Pharmaceutica Nv
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Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DK295286D0 publication Critical patent/DK295286D0/da
Publication of DK295286A publication Critical patent/DK295286A/da
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Publication of DK169073B1 publication Critical patent/DK169073B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/28—Oxygen atom
    • C07D473/30—Oxygen atom attached in position 6, e.g. hypoxanthine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK295286A 1985-06-24 1986-06-23 (4-piperidinylmethyl og -hetero)puriner, præparater indeholdende disse samt fremgangsmåde til fremstilling af disse purinforbindelser DK169073B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8515934 1985-06-24
GB858515934A GB8515934D0 (en) 1985-06-24 1985-06-24 (4-piperidinomethyl and-hetero)purines

Publications (3)

Publication Number Publication Date
DK295286D0 DK295286D0 (da) 1986-06-23
DK295286A DK295286A (da) 1986-12-25
DK169073B1 true DK169073B1 (da) 1994-08-08

Family

ID=10581240

Family Applications (1)

Application Number Title Priority Date Filing Date
DK295286A DK169073B1 (da) 1985-06-24 1986-06-23 (4-piperidinylmethyl og -hetero)puriner, præparater indeholdende disse samt fremgangsmåde til fremstilling af disse purinforbindelser

Country Status (21)

Country Link
US (1) US5041448A (el)
EP (1) EP0206415B1 (el)
JP (1) JPS62487A (el)
KR (1) KR930009356B1 (el)
AT (1) ATE85055T1 (el)
AU (1) AU588890B2 (el)
CA (1) CA1267889A (el)
DE (1) DE3687601T2 (el)
DK (1) DK169073B1 (el)
ES (1) ES8800682A1 (el)
FI (1) FI85704C (el)
GB (1) GB8515934D0 (el)
GR (1) GR861580B (el)
HU (1) HU199143B (el)
IE (1) IE59658B1 (el)
IL (1) IL79193A0 (el)
NO (1) NO163956C (el)
NZ (1) NZ216536A (el)
PT (1) PT82824B (el)
SU (1) SU1581221A3 (el)
ZA (1) ZA864677B (el)

Families Citing this family (69)

* Cited by examiner, † Cited by third party
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US4988689A (en) * 1987-07-01 1991-01-29 Janssen Pharmaceutica N.V. ((Pharmacologically active bicyclic heterocyclic)methyl and -heteroatom) substituted hexahydro-1H-azepines and pyrrolidines
CA1317939C (en) * 1987-07-01 1993-05-18 Janssen Pharmaceutica Naamloze Vennootschap ¬(bicyclic heterocyclyl)methyl and -hetero| substituted hexahydro-1h-azepines and pyrrolidines
US5151424A (en) * 1987-07-01 1992-09-29 Janssen Pharmaceutica N.V. Pharmacologically active (Bicyclic heterocyclyl)methyl and -hetero) substituted hexahydro-1H-azepines and pyrrolidines
GB8716313D0 (en) * 1987-07-10 1987-08-19 Janssen Pharmaceutica Nv 2-(heterocyclylalkyl)imidazopyridines
GB8900380D0 (en) * 1989-01-09 1989-03-08 Janssen Pharmaceutica Nv 2-aminopyrimidinone derivatives
PH30434A (en) * 1989-04-07 1997-05-09 Janssen Pharmaceutica Nv Hydroxyalkylfuranyl derivatives
US5272150A (en) * 1989-04-07 1993-12-21 Janssen Pharmaceutica N.V. Hydroxyalkylfuranyl derivatives
US5360807A (en) * 1990-07-19 1994-11-01 Janssen Pharmaceutica N.V. Substituted thiazolyl and substituted pyridinyl derivatives
NZ238863A (en) * 1990-07-19 1993-03-26 Janssen Pharmaceutica Nv Substituted thiazolyl and pyridinyl derivatives
KR100190299B1 (ko) * 1990-07-19 1999-06-01 디르크 반테 신규한 옥사졸릴 유도체
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AU8506791A (en) * 1990-10-01 1992-04-28 Janssen Pharmaceutica N.V. Novel 4-piperidinylcarbonyl derivatives
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US7179809B2 (en) * 2004-04-10 2007-02-20 Boehringer Ingelheim International Gmbh 2-Amino-imidazo[4,5-d]pyridazin-4-ones, their preparation and their use as pharmaceutical compositions
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WO2008017670A1 (en) * 2006-08-08 2008-02-14 Boehringer Ingelheim International Gmbh Pyrrolo [3, 2 -d] pyrimidines as dpp-iv inhibitors for the treatment of diabetes mellitus
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Also Published As

Publication number Publication date
JPS62487A (ja) 1987-01-06
NO862504L (no) 1986-12-29
FI85704C (fi) 1992-05-25
HU199143B (en) 1990-01-29
ES8800682A1 (es) 1987-11-16
GB8515934D0 (en) 1985-07-24
DK295286D0 (da) 1986-06-23
DE3687601T2 (de) 1993-06-03
NZ216536A (en) 1988-10-28
US5041448A (en) 1991-08-20
EP0206415B1 (en) 1993-01-27
GR861580B (en) 1986-10-21
KR930009356B1 (ko) 1993-09-28
ZA864677B (en) 1988-02-24
PT82824B (pt) 1988-07-29
NO163956C (no) 1990-08-15
HUT42095A (en) 1987-06-29
SU1581221A3 (ru) 1990-07-23
FI85704B (fi) 1992-02-14
DK295286A (da) 1986-12-25
AU5919186A (en) 1987-01-08
DE3687601D1 (de) 1993-03-11
AU588890B2 (en) 1989-09-28
PT82824A (en) 1986-07-01
ATE85055T1 (de) 1993-02-15
EP0206415A2 (en) 1986-12-30
IE59658B1 (en) 1994-03-09
IL79193A0 (en) 1986-09-30
IE861674L (en) 1986-12-24
FI862655A (fi) 1986-12-25
NO862504D0 (no) 1986-06-23
CA1267889A (en) 1990-04-17
FI862655A0 (fi) 1986-06-23
KR870000335A (ko) 1987-02-17
NO163956B (no) 1990-05-07
EP0206415A3 (en) 1988-03-16
ES556381A0 (es) 1987-11-16

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Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed