DK155048C - Analogifremgangsmaade til fremstilling af 1,8-naphthyridinforbindelser - Google Patents

Analogifremgangsmaade til fremstilling af 1,8-naphthyridinforbindelser

Info

Publication number
DK155048C
DK155048C DK408580A DK408580A DK155048C DK 155048 C DK155048 C DK 155048C DK 408580 A DK408580 A DK 408580A DK 408580 A DK408580 A DK 408580A DK 155048 C DK155048 C DK 155048C
Authority
DK
Denmark
Prior art keywords
naphthyride
analogue
preparing
compounds
naphthyride compounds
Prior art date
Application number
DK408580A
Other languages
Danish (da)
English (en)
Other versions
DK408580A (da
DK155048B (da
Inventor
Jun-Ichi Matsumoto
Yoshiyuki Takase
Yoshiro Nishimura
Original Assignee
Dainippon Pharmaceutical Co
Bellon Labor Sa Roger
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dainippon Pharmaceutical Co, Bellon Labor Sa Roger filed Critical Dainippon Pharmaceutical Co
Publication of DK408580A publication Critical patent/DK408580A/da
Publication of DK155048B publication Critical patent/DK155048B/da
Application granted granted Critical
Publication of DK155048C publication Critical patent/DK155048C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK408580A 1979-09-28 1980-09-26 Analogifremgangsmaade til fremstilling af 1,8-naphthyridinforbindelser DK155048C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP12622379 1979-09-28
JP12622379A JPS5649382A (en) 1979-09-28 1979-09-28 6-fluoro-7-cyclic amino-1,8-naphthylidine derivative and its salt

Publications (3)

Publication Number Publication Date
DK408580A DK408580A (da) 1981-03-29
DK155048B DK155048B (da) 1989-01-30
DK155048C true DK155048C (da) 1989-06-26

Family

ID=14929790

Family Applications (1)

Application Number Title Priority Date Filing Date
DK408580A DK155048C (da) 1979-09-28 1980-09-26 Analogifremgangsmaade til fremstilling af 1,8-naphthyridinforbindelser

Country Status (18)

Country Link
US (1) US4341784A (es)
EP (1) EP0027752B1 (es)
JP (1) JPS5649382A (es)
AR (1) AR226320A1 (es)
AU (1) AU534288B2 (es)
CA (1) CA1147731A (es)
CS (1) CS215139B2 (es)
DD (1) DD155990A5 (es)
DE (1) DE3065949D1 (es)
DK (1) DK155048C (es)
ES (1) ES8107217A1 (es)
FI (1) FI70216C (es)
HU (1) HU183218B (es)
PH (1) PH15907A (es)
PL (1) PL127762B1 (es)
SU (1) SU1060112A3 (es)
YU (1) YU42983B (es)
ZA (1) ZA806007B (es)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4382937A (en) * 1981-02-27 1983-05-10 Dainippon Pharmaceutical Co., Ltd. Naphthyridine derivatives and their use as anti-bacterials
JPS57146775A (en) * 1981-03-06 1982-09-10 Dainippon Pharmaceut Co Ltd 1,8-naphthyridine derivative and its salt
JPS5925391A (ja) * 1982-07-30 1984-02-09 Dainippon Pharmaceut Co Ltd ピリジルナフチリジン誘導体およびその塩
US5281612A (en) * 1982-09-09 1994-01-25 Warner-Lambert Company Naphthyridine antibacterial agents
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
US4777175A (en) * 1982-09-09 1988-10-11 Warner-Lambert Company Antibacterial agents
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
FR2559484B2 (fr) * 1983-07-06 1986-09-26 Provesan Sa Nouveau derive 7-(pyrrol-1-yl) de l'acide 1-ethyl-1,4-dihydro-4-oxo-(1,8-naphtyridin)-3-carboxylique, sa preparation et son application en tant que medicament
CS274601B2 (en) 1983-07-27 1991-09-15 Dainippon Pharmaceutical Co Method of 1,8-naphthyridine derivative production
JPS60260577A (ja) * 1984-06-06 1985-12-23 Dainippon Pharmaceut Co Ltd １，８−ナフチリジン誘導体
JPS60112790A (ja) * 1983-11-21 1985-06-19 Dainippon Pharmaceut Co Ltd ピリジルナフチリジン誘導体
NZ210847A (en) * 1984-01-26 1988-02-29 Abbott Lab Naphthyridine and pyridopyrimidine derivatives and pharmaceutical compositions
DE3409922A1 (de) * 1984-03-17 1985-09-26 Bayer Ag, 5090 Leverkusen 1,7-diamino-1,4-dihydro-4-oxo-3-(aza)chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie ihre verwendung bei der bekaempfung bakterieller erkrankungen
US4571396A (en) * 1984-04-16 1986-02-18 Warner-Lambert Company Antibacterial agents
US4604401A (en) * 1984-07-20 1986-08-05 Warner-Lambert Company Antibacterial agents III
DE3508816A1 (de) * 1985-01-10 1986-07-10 Bayer Ag, 5090 Leverkusen 6,7-disubstituierte 1-cyclopropyl-1,4-dihydro-4-oxo-1,8-naphtyridin-3-carbonsaeuren
US4851535A (en) * 1985-01-23 1989-07-25 Toyama Chemical Co., Ltd. Nicotinic acid derivatives
DE3525108A1 (de) * 1985-06-07 1986-12-11 Bayer Ag, 5090 Leverkusen Antibakteriell wirksame chinoloncarbonsaeureester
US4692454A (en) * 1986-02-03 1987-09-08 Warner-Lambert Company Opthalmic use of quinolone antibiotics
US4954507A (en) * 1986-10-08 1990-09-04 Bristol-Myers Company 1-tertiary-alkyl-substituted naphthyridine carboxylic acid antibacterial agents
ZA877471B (en) * 1986-10-08 1988-04-05 Bristol-Myers Company 1-tertiary-alkyl-substituted naphthyridine-and quinoline-carboxylic acid antibacterial agents
US4962108A (en) * 1987-07-31 1990-10-09 Warner-Lambert Company Antibacterial quinoline compounds
US4923879A (en) * 1987-07-31 1990-05-08 Warner-Lambert Company 1,8-Naphthyridines and their use as antibacterial agents
US4920120A (en) * 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents
US5585491A (en) * 1988-01-25 1996-12-17 Otsuka Pharmaceutical Co., Ltd. Antibacterial agents
KR910003630B1 (ko) * 1988-06-17 1991-06-07 한국과학기술원 벤조일 아세틱 에스테르 유도체 및 그 제조방법
US5151267A (en) * 1988-07-15 1992-09-29 University Of Saskatchewan Bovine herpesvirus type 1 polypeptides and vaccines
US5585264A (en) * 1988-07-15 1996-12-17 University Of Saskatchewan Nucleotide sequences encoding recombinant bovine herpesvirus type-1 GI, GIII and GIV polypeptides
IE76284B1 (en) * 1988-09-22 1997-10-08 Abbott Lab Amino acid quinoline and naphthyridine derivatives
US5262417A (en) * 1988-12-06 1993-11-16 The Upjohn Company Antibacterial quinolone compounds
US5527910A (en) * 1992-12-30 1996-06-18 Cheil Foods & Chemicals, Inc. Pyridone carboxylic acid compounds and their uses for treating infectious diseases caused by bacteria
JPH08213881A (ja) * 1995-02-02 1996-08-20 Fujitsu Ltd 周波数制御回路
US5994365A (en) * 1997-02-25 1999-11-30 Diazans Limited Substituted diazaanthracene compounds having pharmaceutical utility
HUP0100051A3 (en) * 1997-09-15 2002-08-28 Procter & Gamble Antimicrobial quinolones, their compositions and uses
US6387928B1 (en) * 1997-09-15 2002-05-14 The Procter & Gamble Co. Antimicrobial quinolones, their compositions and uses
JP4876165B2 (ja) * 2006-03-28 2012-02-15 ザ プロクター アンド ギャンブル カンパニー キノロン中間体を調製するための水素化物還元法
JP2009531418A (ja) * 2006-03-28 2009-09-03 ザ プロクター アンド ギャンブル カンパニー キノロン中間体調製のためのカップリング方法
WO2007110834A2 (en) * 2006-03-28 2007-10-04 The Procter & Gamble Company Malate salts, and polymorphs of (3s,5s)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
AR096135A1 (es) 2013-05-02 2015-12-09 Actelion Pharmaceuticals Ltd Derivados de la quinolona

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3149104A (en) * 1961-01-03 1964-09-15 Sterling Drug Inc 4-hydroxy-7-styryl-1, 8-naphthyridine-3-carboxylic acids and esters
US3673193A (en) * 1970-05-11 1972-06-27 Sterling Drug Inc 4-oxo-1,8-naphthyridine-3-carboxylates and derivatives thereof
US3786043A (en) * 1972-06-19 1974-01-15 Sterling Drug Inc 7-methyl-4-chloro (or -4-lower-alkoxy)-1,8-naphthyridine-3-carboxylates
JPS5637232B2 (es) * 1973-04-17 1981-08-29
US4024255A (en) * 1973-04-05 1977-05-17 Allen & Hanburys Limited Tetrazole containing naphthyridine-3-carboxamides
JPS587626B2 (ja) * 1974-02-13 1983-02-10 大日本製薬株式会社 ナフチリジン オヨビ キノリンユウドウタイノセイホウ
HU173573B (hu) * 1975-02-18 1979-06-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh 1,8-naftridina
DE2607012A1 (de) * 1976-02-18 1977-08-25 Schering Ag Neue 1,5-naphthyridincarbonsaeurederivate und verfahren zu ihrer herstellung
IL51092A0 (en) * 1976-12-10 1977-02-28 Abic Ltd Naphthyridine derivatives and their preparation
JPS543095A (en) * 1977-06-09 1979-01-11 Daito Koeki Preparation of 1*88naphthyridine derivative
SE444566B (sv) * 1977-09-20 1986-04-21 Bellon Labor Sa Roger 7-dialkylamin-6-halogen-4-oxo-1,4-dihydrokinolin-3-karboxylsyra, forfarande for framstellning derav och farmaceutiskt preparat derav
AR223983A1 (es) * 1978-08-25 1981-10-15 Dainippon Pharmaceutical Co Un procedimiento para-preparar derivados de acido 6-halogeno-4-oxo-7-(1-piperazinil)-1,8-naftiridin-3-carboxilico

Also Published As

Publication number Publication date
CS215139B2 (en) 1982-07-30
FI803042A (fi) 1981-03-29
FI70216B (fi) 1986-02-28
EP0027752B1 (en) 1983-12-21
SU1060112A3 (ru) 1983-12-07
PH15907A (en) 1983-04-15
HU183218B (en) 1984-04-28
EP0027752A1 (en) 1981-04-29
ZA806007B (en) 1981-10-28
FI70216C (fi) 1986-09-15
PL127762B1 (en) 1983-11-30
ES495376A0 (es) 1981-10-01
DE3065949D1 (en) 1984-01-26
DK408580A (da) 1981-03-29
YU236480A (en) 1983-02-28
DD155990A5 (de) 1982-07-21
PL226951A1 (es) 1981-10-16
CA1147731A (en) 1983-06-07
JPS5649382A (en) 1981-05-02
AU6257080A (en) 1981-04-09
AR226320A1 (es) 1982-06-30
US4341784A (en) 1982-07-27
YU42983B (en) 1989-02-28
JPS6113717B2 (es) 1986-04-15
ES8107217A1 (es) 1981-10-01
AU534288B2 (en) 1984-01-19
DK155048B (da) 1989-01-30

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Legal Events

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PBP Patent lapsed