DK1458723T3 - Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nuklear hormonreceptorfunktion - Google Patents

Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nuklear hormonreceptorfunktion

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Publication number
DK1458723T3
DK1458723T3 DK02797421T DK02797421T DK1458723T3 DK 1458723 T3 DK1458723 T3 DK 1458723T3 DK 02797421 T DK02797421 T DK 02797421T DK 02797421 T DK02797421 T DK 02797421T DK 1458723 T3 DK1458723 T3 DK 1458723T3
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Prior art keywords
modulators
analogs
hormone receptor
receptor function
condensed heterocyclic
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Application number
DK02797421T
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Danish (da)
English (en)
Inventor
Mark E Salvati
James Aaron Balog
Soren Giese
Aberra Fura
Wenying Li
Toomas Mitt
Jacques Roberge
James R Corte
Steven H Spergel
Richard A Rampulla
Raj Misra
Hai-Yun Xiao
Dacia A Pickering
Ramesh N Patel
Ronald L Hanson
Original Assignee
Bristol Myers Squibb Co
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Publication of DK1458723T3 publication Critical patent/DK1458723T3/da

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    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/18—Bridged systems
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Urology & Nephrology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK02797421T 2001-12-19 2002-12-18 Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nuklear hormonreceptorfunktion DK1458723T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2511601A 2001-12-19 2001-12-19
PCT/US2002/040598 WO2003062241A1 (en) 2001-12-19 2002-12-18 Fused heterocyclic succinimidecompounds and analogs thereof, modulators of nuclear hormone receptor function

Publications (1)

Publication Number Publication Date
DK1458723T3 true DK1458723T3 (da) 2009-02-09

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DK02797421T DK1458723T3 (da) 2001-12-19 2002-12-18 Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nuklear hormonreceptorfunktion

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Country Link
EP (1) EP1458723B1 (xx)
JP (1) JP2005523257A (xx)
KR (1) KR20040086248A (xx)
CN (1) CN1589271A (xx)
AR (1) AR037950A1 (xx)
AT (1) ATE411319T1 (xx)
AU (1) AU2002361785B2 (xx)
BR (1) BR0215281A (xx)
CA (1) CA2471342A1 (xx)
CO (1) CO5640082A2 (xx)
DE (1) DE60229435D1 (xx)
DK (1) DK1458723T3 (xx)
ES (1) ES2314127T3 (xx)
GE (1) GEP20063817B (xx)
HR (1) HRP20040567A2 (xx)
HU (1) HUP0402554A3 (xx)
IL (1) IL162547A0 (xx)
IS (1) IS7324A (xx)
MX (1) MXPA04005876A (xx)
NO (1) NO20043068L (xx)
NZ (1) NZ533471A (xx)
PL (1) PL370904A1 (xx)
PT (1) PT1458723E (xx)
RU (1) RU2330038C2 (xx)
SI (1) SI1458723T1 (xx)
TW (1) TWI263640B (xx)
UA (1) UA78265C2 (xx)
UY (1) UY27595A1 (xx)
WO (1) WO2003062241A1 (xx)
YU (1) YU53604A (xx)
ZA (1) ZA200404812B (xx)

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AU2002361785B2 (en) 2008-05-22
EP1458723B1 (en) 2008-10-15
CA2471342A1 (en) 2003-07-31
EP1458723A1 (en) 2004-09-22
ATE411319T1 (de) 2008-10-15
HUP0402554A2 (hu) 2005-03-29
DE60229435D1 (de) 2008-11-27
JP2005523257A (ja) 2005-08-04
EP1458723A4 (en) 2005-12-21
GEP20063817B (en) 2006-05-10
IL162547A0 (en) 2005-11-20
RU2330038C2 (ru) 2008-07-27
HUP0402554A3 (en) 2009-01-28
SI1458723T1 (sl) 2009-02-28
RU2004122403A (ru) 2005-05-27
TW200304810A (en) 2003-10-16
BR0215281A (pt) 2004-10-19
NZ533471A (en) 2007-05-31
KR20040086248A (ko) 2004-10-08
ZA200404812B (en) 2005-08-26
YU53604A (sh) 2006-08-17
UY27595A1 (es) 2003-07-31
AR037950A1 (es) 2004-12-22
ES2314127T3 (es) 2009-03-16
WO2003062241A1 (en) 2003-07-31
MXPA04005876A (es) 2005-05-16
CN1589271A (zh) 2005-03-02
PL370904A1 (en) 2005-05-30
NO20043068L (no) 2004-09-08
PT1458723E (pt) 2008-12-26
WO2003062241A8 (en) 2004-10-21
IS7324A (is) 2004-06-18
HRP20040567A2 (en) 2005-06-30
TWI263640B (en) 2006-10-11
UA78265C2 (en) 2007-03-15

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