DK142852B - Analogifremgangsmåde til fremstilling af fusida-13(17)-en-21-carboxylsyrederivater. - Google Patents

Analogifremgangsmåde til fremstilling af fusida-13(17)-en-21-carboxylsyrederivater. Download PDF

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Publication number
DK142852B
DK142852B DK539476AA DK539476A DK142852B DK 142852 B DK142852 B DK 142852B DK 539476A A DK539476A A DK 539476AA DK 539476 A DK539476 A DK 539476A DK 142852 B DK142852 B DK 142852B
Authority
DK
Denmark
Prior art keywords
carboxylic acid
dihydroxy
diene
acid
fusida
Prior art date
Application number
DK539476AA
Other languages
Danish (da)
English (en)
Other versions
DK142852C (it
DK539476A (it
Inventor
Welf Von Daehne
Poul Roedbroe Rasmussen
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB49714/75A external-priority patent/GB1565954A/en
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of DK539476A publication Critical patent/DK539476A/da
Publication of DK142852B publication Critical patent/DK142852B/da
Application granted granted Critical
Publication of DK142852C publication Critical patent/DK142852C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J13/00Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/003Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0088Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing unsubstituted amino radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
DK539476AA 1975-12-03 1976-12-01 Analogifremgangsmåde til fremstilling af fusida-13(17)-en-21-carboxylsyrederivater. DK142852B (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB4971475 1975-12-03
GB49714/75A GB1565954A (en) 1975-12-03 1975-12-03 Fusidic acid derivatives
GB1601576 1976-04-20
GB1601576 1976-04-20

Publications (3)

Publication Number Publication Date
DK539476A DK539476A (it) 1977-06-04
DK142852B true DK142852B (da) 1981-02-09
DK142852C DK142852C (it) 1981-09-21

Family

ID=26251702

Family Applications (1)

Application Number Title Priority Date Filing Date
DK539476AA DK142852B (da) 1975-12-03 1976-12-01 Analogifremgangsmåde til fremstilling af fusida-13(17)-en-21-carboxylsyrederivater.

Country Status (20)

Country Link
US (2) US4100276A (it)
JP (1) JPS5271459A (it)
AT (1) AT343810B (it)
AU (1) AU501066B2 (it)
CA (1) CA1079267A (it)
DE (1) DE2654508A1 (it)
DK (1) DK142852B (it)
ES (1) ES453853A1 (it)
FI (1) FI57599C (it)
FR (1) FR2333807A1 (it)
GR (1) GR62007B (it)
IE (1) IE44263B1 (it)
IT (1) IT1074295B (it)
LU (1) LU76313A1 (it)
NL (1) NL7613445A (it)
NZ (1) NZ182661A (it)
PT (1) PT65925B (it)
SE (1) SE410859B (it)
SU (1) SU679146A3 (it)
YU (1) YU291176A (it)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE44263B1 (en) * 1975-12-03 1981-09-23 Leo Pharm Prod Ltd New fusidic acid derivatives
US4162259A (en) * 1975-12-03 1979-07-24 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske fabrik Produktionsaktienselskab) Fusidic acid derivatives
US4959358A (en) * 1983-06-06 1990-09-25 Beth Israel Hospital Assn. Drug administration
US4548922A (en) * 1983-06-06 1985-10-22 Beth Israel Hospital Drug administration
US4746508A (en) * 1983-06-06 1988-05-24 Beth Israel Hospital Assn. Drug administration
US6255299B1 (en) * 1985-01-07 2001-07-03 Leo Pharmaceutical Products Ltd. Opthalmic gel composition and method of treating eye infections
GB8500310D0 (en) * 1985-01-07 1985-02-13 Leo Pharm Prod Ltd Pharmaceutical preparation
GB8706313D0 (en) * 1987-03-17 1987-04-23 Health Lab Service Board Treatment & prevention of viral infections
US4994439A (en) * 1989-01-19 1991-02-19 California Biotechnology Inc. Transmembrane formulations for drug administration
US5372996A (en) * 1989-03-10 1994-12-13 Endorecherche, Inc. Method of treatment of androgen-related diseases
ATE170753T1 (de) * 1989-07-07 1998-09-15 Endorecherche Inc Androgenderivate zur hemming der aktivität der sexualsteroide
JP3350048B2 (ja) * 1989-07-07 2002-11-25 アンドルシェルシュ・インコーポレイテッド アンドロゲン関連疾患の治療方法
CZ286894A3 (en) * 1992-05-21 1995-09-13 Endorecherche Inc Pharmaceutical preparation
US5454801A (en) * 1992-10-09 1995-10-03 Mcneil-Ppc, Inc. Printed polymer coatings and method for making same
US5658560A (en) * 1994-01-18 1997-08-19 Serikov; Vladimir B. Method of treating endotoxemia by administering tyloxapol
MY140194A (en) * 2003-07-16 2009-11-30 Leo Pharma As Novel fusidic acid derivatives
US20080161324A1 (en) * 2006-09-14 2008-07-03 Johansen Lisa M Compositions and methods for treatment of viral diseases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1447489A (en) * 1972-10-06 1976-08-25 Leo Pharm Prod Ltd Fusidic acid conjugates
GB1490852A (en) * 1974-09-12 1977-11-02 Leo Pharm Prod Ltd Fusidic acid derivatives
IE44263B1 (en) * 1975-12-03 1981-09-23 Leo Pharm Prod Ltd New fusidic acid derivatives

Also Published As

Publication number Publication date
SE7613565L (sv) 1977-06-04
SU679146A3 (ru) 1979-08-05
PT65925B (en) 1978-06-13
AU1986876A (en) 1978-06-01
PT65925A (en) 1977-01-01
IT1074295B (it) 1985-04-20
NZ182661A (en) 1979-07-11
ATA887576A (de) 1977-10-15
US4100276A (en) 1978-07-11
FI57599B (fi) 1980-05-30
SE410859B (sv) 1979-11-12
ES453853A1 (es) 1978-01-16
AT343810B (de) 1978-06-26
LU76313A1 (it) 1977-06-21
US4315004A (en) 1982-02-09
GR62007B (en) 1979-02-15
NL7613445A (nl) 1977-06-07
DE2654508A1 (de) 1977-06-08
CA1079267A (en) 1980-06-10
DK142852C (it) 1981-09-21
AU501066B2 (en) 1979-06-07
IE44263L (en) 1977-06-03
FR2333807B1 (it) 1980-11-07
IE44263B1 (en) 1981-09-23
YU291176A (en) 1982-05-31
FI763473A (it) 1977-06-04
FI57599C (fi) 1980-09-10
JPS5271459A (en) 1977-06-14
FR2333807A1 (fr) 1977-07-01
DK539476A (it) 1977-06-04

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