DK142767B - Analogifremgangsmåde til fremstilling af 1- og dl-(racem-)formerne af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol. - Google Patents

Analogifremgangsmåde til fremstilling af 1- og dl-(racem-)formerne af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol. Download PDF

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Publication number
DK142767B
DK142767B DK467977AA DK467977A DK142767B DK 142767 B DK142767 B DK 142767B DK 467977A A DK467977A A DK 467977AA DK 467977 A DK467977 A DK 467977A DK 142767 B DK142767 B DK 142767B
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Prior art keywords
tetrahydroimidazo
thiazole
compounds
product
compound
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Application number
DK467977AA
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Danish (da)
English (en)
Other versions
DK467977A (de
DK142767C (de
Inventor
John Kendrick Stubbs
Michael Raymond Graves Leeming
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK467977A publication Critical patent/DK467977A/da
Publication of DK142767B publication Critical patent/DK142767B/da
Application granted granted Critical
Publication of DK142767C publication Critical patent/DK142767C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK467977AA 1976-10-22 1977-10-20 Analogifremgangsmåde til fremstilling af 1- og dl-(racem-)formerne af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol. DK142767B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB44060/76A GB1533347A (en) 1976-10-22 1976-10-22 Anthelmintic compounds
GB4406076 1976-10-22

Publications (3)

Publication Number Publication Date
DK467977A DK467977A (de) 1978-04-23
DK142767B true DK142767B (da) 1981-01-19
DK142767C DK142767C (de) 1981-08-17

Family

ID=10431568

Family Applications (1)

Application Number Title Priority Date Filing Date
DK467977AA DK142767B (da) 1976-10-22 1977-10-20 Analogifremgangsmåde til fremstilling af 1- og dl-(racem-)formerne af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol.

Country Status (25)

Country Link
US (1) US4137321A (de)
JP (1) JPS5353692A (de)
AR (1) AR213981A1 (de)
AT (1) AT360518B (de)
BE (1) BE859949A (de)
BG (1) BG28421A3 (de)
CA (1) CA1088546A (de)
CH (1) CH627473A5 (de)
CS (1) CS191897B2 (de)
DD (1) DD133439A5 (de)
DE (1) DE2747122A1 (de)
DK (1) DK142767B (de)
ES (1) ES463414A1 (de)
FI (1) FI62095C (de)
FR (1) FR2368493A1 (de)
GB (1) GB1533347A (de)
IE (1) IE45811B1 (de)
IL (1) IL53093A (de)
LU (1) LU78358A1 (de)
NL (1) NL168229C (de)
NZ (1) NZ185339A (de)
PL (1) PL201668A1 (de)
PT (1) PT67178B (de)
SE (1) SE7711897L (de)
ZA (1) ZA775876B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS573376Y2 (de) * 1978-09-06 1982-01-21
EP0041322A1 (de) 1980-05-30 1981-12-09 Beecham Group Plc m-Pyrazolylamidotetramisol-Derivate, Verfahren zur Herstellung dieser Verbindungen, sie enthaltende Zusammensetzungen sowie ihre Verwendung bei der Behandlung der Helminthiasis
US4636517A (en) * 1985-10-18 1987-01-13 International Minerals & Chemical Corp. 3-tolylthio-4-amino-4,5-dihydro isoxazole as anthelmintic
US5516647A (en) * 1993-11-05 1996-05-14 Abbott Laboratories Compounds useful as alkaline phosphatase inhibitors and therapeutic agents
US6727272B1 (en) * 2002-07-15 2004-04-27 Unitech Pharmaceuticals, Inc. Leflunomide analogs for treating rheumatoid arthritis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL131034C (de) * 1964-05-11
AU409983B2 (en) * 1965-07-19 1970-12-31 Imperial Chemical Industries Of Australia New Zealand Limited Process for the manufacture of thia zolidines and thiazolidines produced thereby
US3708490A (en) * 1970-11-16 1973-01-02 L Spicer Imidazothiazolium compounds,preparation and method of use
US4014892A (en) * 1972-09-14 1977-03-29 American Cyanamid Company 6-Substituted amino phenyl-2,3,5,6-tetrahydro[2,1-b]thiazoles
ZA735753B (en) * 1972-09-14 1974-07-31 American Cyanamid Co Resolution of 6-substituted amino phenyl-2,3,5,6-tetrahydro(2,1-b)thiadiazoles

Also Published As

Publication number Publication date
CA1088546A (en) 1980-10-28
CH627473A5 (fr) 1982-01-15
NL168229C (nl) 1982-03-16
IL53093A (en) 1980-01-31
SE7711897L (sv) 1978-04-23
ZA775876B (en) 1978-05-30
DE2747122A1 (de) 1978-04-27
NL7711520A (nl) 1978-04-25
FI62095C (fi) 1982-11-10
PL201668A1 (pl) 1978-08-28
LU78358A1 (de) 1978-01-24
FR2368493B1 (de) 1981-11-27
GB1533347A (en) 1978-11-22
ES463414A1 (es) 1979-07-01
US4137321A (en) 1979-01-30
JPS5353692A (en) 1978-05-16
FR2368493A1 (fr) 1978-05-19
IE45811L (en) 1978-04-22
AU2943077A (en) 1978-09-28
DK467977A (de) 1978-04-23
IL53093A0 (en) 1977-12-30
DD133439A5 (de) 1979-01-03
AT360518B (de) 1981-01-12
JPS5531158B2 (de) 1980-08-15
IE45811B1 (en) 1982-12-01
DK142767C (de) 1981-08-17
NL168229B (nl) 1981-10-16
NZ185339A (en) 1979-03-16
AR213981A1 (es) 1979-04-11
PT67178A (en) 1977-11-01
FI62095B (fi) 1982-07-30
FI773118A (fi) 1978-04-23
CS191897B2 (en) 1979-07-31
BG28421A3 (en) 1980-04-15
ATA749177A (de) 1980-06-15
PT67178B (en) 1979-03-21
BE859949A (fr) 1978-04-20

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