DK120783A - Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner - Google Patents
Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner Download PDFInfo
- Publication number
- DK120783A DK120783A DK120783A DK120783A DK120783A DK 120783 A DK120783 A DK 120783A DK 120783 A DK120783 A DK 120783A DK 120783 A DK120783 A DK 120783A DK 120783 A DK120783 A DK 120783A
- Authority
- DK
- Denmark
- Prior art keywords
- pyrazolo
- pyrimidines
- preparing substituted
- substituted
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8207637 | 1982-03-16 | ||
| GB838303089A GB8303089D0 (en) | 1983-02-04 | 1983-02-04 | Substituted 1h-pyrazolo 1,5-a pyrimidines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK120783D0 DK120783D0 (da) | 1983-03-15 |
| DK120783A true DK120783A (da) | 1983-09-17 |
Family
ID=26282260
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK120783A DK120783A (da) | 1982-03-16 | 1983-03-15 | Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4482555A (de) |
| AU (1) | AU557300B2 (de) |
| CA (1) | CA1192546A (de) |
| CH (1) | CH654306A5 (de) |
| DE (1) | DE3309432A1 (de) |
| DK (1) | DK120783A (de) |
| FI (1) | FI74469C (de) |
| FR (1) | FR2523582B1 (de) |
| IL (1) | IL68133A (de) |
| IT (1) | IT1194555B (de) |
| NL (1) | NL8300934A (de) |
| SE (1) | SE450573B (de) |
| SU (1) | SU1366060A3 (de) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6245759B1 (en) | 1999-03-11 | 2001-06-12 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| MY125533A (en) | 1999-12-06 | 2006-08-30 | Bristol Myers Squibb Co | Heterocyclic dihydropyrimidine compounds |
| EP1782859A3 (de) * | 2003-04-11 | 2009-09-30 | High Point Pharmaceuticals, LLC | Pharmazeutische Verwendung von Pyrazolo [1,5- a] Pyrimidin-Derivaten |
| EP1615697A2 (de) * | 2003-04-11 | 2006-01-18 | Novo Nordisk A/S | Neue pyrazolo[1,5-a] pyrimidin-derivate und deren pharmazeutische verwendungen |
| US7772232B2 (en) | 2004-04-15 | 2010-08-10 | Bristol-Myers Squibb Company | Quinazolinyl compounds as inhibitors of potassium channel function |
| JP2008515956A (ja) * | 2004-10-12 | 2008-05-15 | ノボ ノルディスク アクティーゼルスカブ | １１β−ヒドロキシステロイドデヒドロゲナーゼ１型活性スピロ化合物 |
| US20090124598A1 (en) * | 2005-11-01 | 2009-05-14 | Henrik Sune Andersen | Pharmaceutical use of substituted amides |
| WO2007051811A2 (en) * | 2005-11-01 | 2007-05-10 | Transtech Pharma | Pharmaceutical use of substituted amides |
| WO2007107550A1 (en) * | 2006-03-21 | 2007-09-27 | High Point Pharmaceuticals, Llc | Adamantane derivatives for the treatment of the metabolic syndrome |
| JP2009532418A (ja) | 2006-04-07 | 2009-09-10 | ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー | １１β−ヒドロキシステロイドデヒドロゲナーゼ１型活性化合物 |
| CA2655282A1 (en) * | 2006-06-16 | 2007-12-21 | High Point Pharmaceuticals, Llc | Pharmaceutical use of substituted piperidine carboxamides |
| EP1878721A1 (de) * | 2006-07-13 | 2008-01-16 | Novo Nordisk A/S | 4-Piperidylbenzamide als Inhibitoren der 11-beta-hydroxysteroiddehydrogenase Typ 1 |
| CA2657078A1 (en) * | 2006-07-13 | 2008-01-17 | High Point Pharmaceuticals, Llc | 11beta-hydroxysteroid dehydrogenase type 1 active compounds |
| US20110003852A1 (en) * | 2007-02-23 | 2011-01-06 | Soren Ebdrup | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
| JP2010519240A (ja) * | 2007-02-23 | 2010-06-03 | ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー | １１−ベータ−ヒドロキシステロイドデヒドロゲナーゼの阻害剤としての、ｎ−アダマンチルベンズアミド |
| US8334305B2 (en) * | 2007-02-23 | 2012-12-18 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-β-hydroxysteroid dehydrogenase |
| AU2008219326B2 (en) * | 2007-02-23 | 2012-12-13 | Vtv Therapeutics Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
| US8153798B2 (en) * | 2007-03-09 | 2012-04-10 | High Point Pharmaceuticals, Llc | Indole- and benzimidazole amides as hydroxysteroid dehydrogenase inhibitors |
| WO2008119017A1 (en) * | 2007-03-28 | 2008-10-02 | High Point Pharmaceuticals, Llc | 11beta-hsd1 active compounds |
| CA2683852A1 (en) * | 2007-04-11 | 2008-10-23 | High Point Pharmaceuticals, Llc | Novel compounds |
| JP2010526777A (ja) * | 2007-04-24 | 2010-08-05 | ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー | 置換アミドの医薬用途 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3907799A (en) * | 1971-08-16 | 1975-09-23 | Icn Pharmaceuticals | Xanthine oxidase inhibitors |
| BE786611A (fr) * | 1971-08-16 | 1973-01-22 | Int Chem & Nuclear Corp | Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio |
| US3925385A (en) * | 1972-04-20 | 1975-12-09 | Icn Pharmaceuticals | 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines |
| BE792533A (fr) * | 1971-12-09 | 1973-06-08 | Int Chem & Nuclear Corp | Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation |
| US4093617A (en) * | 1974-11-12 | 1978-06-06 | Icn Pharmaceuticals, Inc. | 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines |
| US4048184A (en) * | 1976-11-15 | 1977-09-13 | E. R. Squibb & Sons, Inc. | 6-Phenyl-2H-pyrazolo[3,4-b]pyridines |
| US4281000A (en) * | 1979-07-09 | 1981-07-28 | American Cyanamid Company | Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents |
-
1983
- 1983-03-09 AU AU12304/83A patent/AU557300B2/en not_active Ceased
- 1983-03-10 US US06/474,205 patent/US4482555A/en not_active Expired - Fee Related
- 1983-03-11 IT IT20024/83A patent/IT1194555B/it active
- 1983-03-11 CH CH1325/83A patent/CH654306A5/de not_active IP Right Cessation
- 1983-03-15 DK DK120783A patent/DK120783A/da not_active Application Discontinuation
- 1983-03-15 FI FI830864A patent/FI74469C/fi not_active IP Right Cessation
- 1983-03-15 FR FR8304253A patent/FR2523582B1/fr not_active Expired
- 1983-03-15 SE SE8301412A patent/SE450573B/sv not_active IP Right Cessation
- 1983-03-15 SU SU833565748A patent/SU1366060A3/ru active
- 1983-03-15 IL IL68133A patent/IL68133A/xx unknown
- 1983-03-15 NL NL8300934A patent/NL8300934A/xx active Search and Examination
- 1983-03-15 CA CA000423644A patent/CA1192546A/en not_active Expired
- 1983-03-16 DE DE19833309432 patent/DE3309432A1/de not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| IL68133A (en) | 1985-12-31 |
| AU557300B2 (en) | 1986-12-18 |
| NL8300934A (nl) | 1983-10-17 |
| FI830864L (fi) | 1983-09-17 |
| FI74469C (fi) | 1988-02-08 |
| US4482555A (en) | 1984-11-13 |
| FR2523582A1 (fr) | 1983-09-23 |
| CH654306A5 (de) | 1986-02-14 |
| IT1194555B (it) | 1988-09-22 |
| IL68133A0 (en) | 1983-06-15 |
| FI74469B (fi) | 1987-10-30 |
| IT8320024A0 (it) | 1983-03-11 |
| SE8301412L (sv) | 1983-09-17 |
| AU1230483A (en) | 1983-09-22 |
| SE450573B (sv) | 1987-07-06 |
| FR2523582B1 (fr) | 1985-12-06 |
| FI830864A0 (fi) | 1983-03-15 |
| DK120783D0 (da) | 1983-03-15 |
| DE3309432A1 (de) | 1983-09-22 |
| SU1366060A3 (ru) | 1988-01-07 |
| CA1192546A (en) | 1985-08-27 |
| SE8301412D0 (sv) | 1983-03-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK120783A (da) | Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner | |
| DK350083A (da) | Fremgangsmaade til fremstilling af phenylethanolaminer | |
| DK194783D0 (da) | Fremgangsmade til fremstilling af bicycliske forbindelser | |
| DK29183D0 (da) | Fremgangsmade til fremstilling af purinderivater | |
| DK25081A (da) | Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner | |
| DK300883D0 (da) | Fremgangsmade til fremstilling af thromobolytiske midler | |
| DK227183A (da) | Fremgangsmaade til fremstilling af imidazo(1,2-c)-pyrazolo(3,4-e)pyrimidiner med den almene formel i | |
| DK173983D0 (da) | Fremgangsmade til fremstilling af imidazo (1,2-alfa)pyridiner | |
| DK210083A (da) | Fremgangsmaade til fremstilling af 6a,10a-trans-hexahydrodibenzopyranoner | |
| DK540984A (da) | Fremgangsmaade til fremstilling af 1,2,4-triazolo-(1,5-a)pyrimidin-2-sulfonylchlorider | |
| DK133482A (da) | Fremgangsmaade til fremstilling af imidazo(1,2-a)pyrimidiner | |
| DK390583A (da) | Fremgangsmaade til fremstilling af imidazo(1,2-a)pyrimidiner | |
| NO834711L (no) | Imidazo(1,5-a)pyridin-derivater | |
| DK457583A (da) | Fremgangsmaade til fremstilling af dihydropyrazolo(3,4-b)pyridin-derivater | |
| DK314682A (da) | Fremgangsmaade til fremstilling af substituerede thiazolo-(3,2-a)pyrimidiner | |
| DK200280A (da) | Fremgangsmaade til fremstilling af substituerede pyrido (1,2-a) pyrimidiner | |
| FI834664A0 (fi) | Substituerade imidazo(1,5-a)pyridiner | |
| DK44383D0 (da) | Fremgangsmade til fremstilling af substituerede 1,3,4-thiadiazolo(3,2-a)pyrimidiner | |
| DK40883A (da) | Fremgangsmaade til fremstilling af benzothienylallylaminer | |
| DK133883D0 (da) | Fremgangsmade til fremstilling af substituerede ethenylderivater af 1h-pyrazolo(1,5-a)pyrimidin | |
| DK162097C (da) | Fremgangsmaade til fremstilling af riboflavin | |
| DK446683D0 (da) | Fremgangsmade til fremstilling af 6-anilino-5,8-quinoxalindioner | |
| DK385983A (da) | Fremgangsmaade til fremstilling af 1-oxacephamer | |
| DK219483D0 (da) | Fremgangsmade til fremstilling af anthracyclinglycosider | |
| DK158726C (da) | Fremgangsmaade til fremstilling af pyrimidintrionderivater |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |