DK120783A - Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner - Google Patents
Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner Download PDFInfo
- Publication number
- DK120783A DK120783A DK120783A DK120783A DK120783A DK 120783 A DK120783 A DK 120783A DK 120783 A DK120783 A DK 120783A DK 120783 A DK120783 A DK 120783A DK 120783 A DK120783 A DK 120783A
- Authority
- DK
- Denmark
- Prior art keywords
- pyrazolo
- pyrimidines
- preparing substituted
- substituted
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8207637 | 1982-03-16 | ||
GB838303089A GB8303089D0 (en) | 1983-02-04 | 1983-02-04 | Substituted 1h-pyrazolo 1,5-a pyrimidines |
Publications (2)
Publication Number | Publication Date |
---|---|
DK120783D0 DK120783D0 (da) | 1983-03-15 |
DK120783A true DK120783A (da) | 1983-09-17 |
Family
ID=26282260
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK120783A DK120783A (da) | 1982-03-16 | 1983-03-15 | Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner |
Country Status (13)
Country | Link |
---|---|
US (1) | US4482555A (de) |
AU (1) | AU557300B2 (de) |
CA (1) | CA1192546A (de) |
CH (1) | CH654306A5 (de) |
DE (1) | DE3309432A1 (de) |
DK (1) | DK120783A (de) |
FI (1) | FI74469C (de) |
FR (1) | FR2523582B1 (de) |
IL (1) | IL68133A (de) |
IT (1) | IT1194555B (de) |
NL (1) | NL8300934A (de) |
SE (1) | SE450573B (de) |
SU (1) | SU1366060A3 (de) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6245759B1 (en) * | 1999-03-11 | 2001-06-12 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
MY125533A (en) | 1999-12-06 | 2006-08-30 | Bristol Myers Squibb Co | Heterocyclic dihydropyrimidine compounds |
EP1782859A3 (de) * | 2003-04-11 | 2009-09-30 | High Point Pharmaceuticals, LLC | Pharmazeutische Verwendung von Pyrazolo [1,5- a] Pyrimidin-Derivaten |
EP1615697A2 (de) * | 2003-04-11 | 2006-01-18 | Novo Nordisk A/S | Neue pyrazolo[1,5-a] pyrimidin-derivate und deren pharmazeutische verwendungen |
US7772232B2 (en) | 2004-04-15 | 2010-08-10 | Bristol-Myers Squibb Company | Quinazolinyl compounds as inhibitors of potassium channel function |
WO2006040329A1 (en) * | 2004-10-12 | 2006-04-20 | Novo Nordisk A/S | 1 ibeta- hydroxysteroid dehydrogenase type 1 active spiro compounds |
JP2009513611A (ja) * | 2005-11-01 | 2009-04-02 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 置換アミドの医薬用途 |
WO2007051810A2 (en) * | 2005-11-01 | 2007-05-10 | Transtech Pharma | Pharmaceutical use of substituted amides |
JP2009530346A (ja) * | 2006-03-21 | 2009-08-27 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | メタボリックシンドロームの治療用のアダマンタン誘導体 |
KR20090014347A (ko) | 2006-04-07 | 2009-02-10 | 하이 포인트 파마슈티칼스, 엘엘씨 | 11β-히드록시스테로이드 탈수소효소 타입 1 활성 화합물 |
JP2009539937A (ja) * | 2006-06-16 | 2009-11-19 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 置換型ピペリジンカルボキサミドの医薬的使用 |
US8048908B2 (en) * | 2006-07-13 | 2011-11-01 | High Point Pharmaceuticals, Llc | 11β-hydroxysteroid dehydrogenase type 1 active compounds |
EP1878721A1 (de) * | 2006-07-13 | 2008-01-16 | Novo Nordisk A/S | 4-Piperidylbenzamide als Inhibitoren der 11-beta-hydroxysteroiddehydrogenase Typ 1 |
US20110003852A1 (en) * | 2007-02-23 | 2011-01-06 | Soren Ebdrup | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
AU2008219326B2 (en) * | 2007-02-23 | 2012-12-13 | Vtv Therapeutics Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
WO2008101886A1 (en) * | 2007-02-23 | 2008-08-28 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
JP2010519242A (ja) * | 2007-02-23 | 2010-06-03 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 新規化合物 |
CA2679866A1 (en) * | 2007-03-09 | 2008-09-18 | High Point Pharmaceuticals, Llc | Indole- and benzimidazole amides as hydroxysteroid dehydrogenase inhibitors |
CA2681934A1 (en) * | 2007-03-28 | 2008-10-02 | High Point Pharmaceuticals, Llc | 11beta-hsd1 active compounds |
CN101677562A (zh) * | 2007-04-11 | 2010-03-24 | 高点制药有限责任公司 | 新化合物 |
EP2150109B1 (de) * | 2007-04-24 | 2012-09-19 | High Point Pharmaceuticals, LLC | Pharmazeutische verwendung von substituierten amiden |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE786611A (fr) * | 1971-08-16 | 1973-01-22 | Int Chem & Nuclear Corp | Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio |
US3907799A (en) * | 1971-08-16 | 1975-09-23 | Icn Pharmaceuticals | Xanthine oxidase inhibitors |
US3925385A (en) * | 1972-04-20 | 1975-12-09 | Icn Pharmaceuticals | 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines |
BE792533A (fr) * | 1971-12-09 | 1973-06-08 | Int Chem & Nuclear Corp | Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation |
US4093617A (en) * | 1974-11-12 | 1978-06-06 | Icn Pharmaceuticals, Inc. | 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines |
US4048184A (en) * | 1976-11-15 | 1977-09-13 | E. R. Squibb & Sons, Inc. | 6-Phenyl-2H-pyrazolo[3,4-b]pyridines |
US4281000A (en) * | 1979-07-09 | 1981-07-28 | American Cyanamid Company | Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents |
-
1983
- 1983-03-09 AU AU12304/83A patent/AU557300B2/en not_active Ceased
- 1983-03-10 US US06/474,205 patent/US4482555A/en not_active Expired - Fee Related
- 1983-03-11 CH CH1325/83A patent/CH654306A5/de not_active IP Right Cessation
- 1983-03-11 IT IT20024/83A patent/IT1194555B/it active
- 1983-03-15 SU SU833565748A patent/SU1366060A3/ru active
- 1983-03-15 FI FI830864A patent/FI74469C/fi not_active IP Right Cessation
- 1983-03-15 CA CA000423644A patent/CA1192546A/en not_active Expired
- 1983-03-15 IL IL68133A patent/IL68133A/xx unknown
- 1983-03-15 NL NL8300934A patent/NL8300934A/xx active Search and Examination
- 1983-03-15 FR FR8304253A patent/FR2523582B1/fr not_active Expired
- 1983-03-15 DK DK120783A patent/DK120783A/da not_active Application Discontinuation
- 1983-03-15 SE SE8301412A patent/SE450573B/sv not_active IP Right Cessation
- 1983-03-16 DE DE19833309432 patent/DE3309432A1/de not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
US4482555A (en) | 1984-11-13 |
SE450573B (sv) | 1987-07-06 |
FI830864A0 (fi) | 1983-03-15 |
CH654306A5 (de) | 1986-02-14 |
AU1230483A (en) | 1983-09-22 |
CA1192546A (en) | 1985-08-27 |
IT8320024A0 (it) | 1983-03-11 |
NL8300934A (nl) | 1983-10-17 |
FI74469C (fi) | 1988-02-08 |
FR2523582B1 (fr) | 1985-12-06 |
AU557300B2 (en) | 1986-12-18 |
SE8301412L (sv) | 1983-09-17 |
IL68133A (en) | 1985-12-31 |
FI830864L (fi) | 1983-09-17 |
SU1366060A3 (ru) | 1988-01-07 |
FI74469B (fi) | 1987-10-30 |
DE3309432A1 (de) | 1983-09-22 |
IL68133A0 (en) | 1983-06-15 |
IT1194555B (it) | 1988-09-22 |
DK120783D0 (da) | 1983-03-15 |
SE8301412D0 (sv) | 1983-03-15 |
FR2523582A1 (fr) | 1983-09-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |