DK25081A - Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner - Google Patents

Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner

Info

Publication number
DK25081A
DK25081A DK25081A DK25081A DK25081A DK 25081 A DK25081 A DK 25081A DK 25081 A DK25081 A DK 25081A DK 25081 A DK25081 A DK 25081A DK 25081 A DK25081 A DK 25081A
Authority
DK
Denmark
Prior art keywords
pyridines
preparing imidazo
imidazo
preparing
Prior art date
Application number
DK25081A
Other languages
English (en)
Inventor
J A Bristol
C Puchalski
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of DK25081A publication Critical patent/DK25081A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK25081A 1980-01-23 1981-01-20 Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner DK25081A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11447380A 1980-01-23 1980-01-23

Publications (1)

Publication Number Publication Date
DK25081A true DK25081A (da) 1981-07-24

Family

ID=22355431

Family Applications (1)

Application Number Title Priority Date Filing Date
DK25081A DK25081A (da) 1980-01-23 1981-01-20 Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner

Country Status (21)

Country Link
EP (1) EP0033094B1 (da)
JP (1) JPS56113782A (da)
KR (1) KR850000240B1 (da)
AU (1) AU540840B2 (da)
CA (1) CA1167845A (da)
DE (1) DE3166531D1 (da)
DK (1) DK25081A (da)
FI (1) FI810147L (da)
GR (1) GR72960B (da)
HK (1) HK94187A (da)
HU (1) HU185857B (da)
IE (1) IE50682B1 (da)
IL (1) IL61939A (da)
MA (1) MA19048A1 (da)
MY (1) MY8700760A (da)
NO (1) NO157781C (da)
NZ (1) NZ196071A (da)
OA (1) OA06727A (da)
PT (1) PT72370B (da)
SG (1) SG70887G (da)
ZA (1) ZA81219B (da)

Families Citing this family (52)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4460584A (en) * 1981-03-13 1984-07-17 Imperial Chemical Industries Plc Nitrogen heterocycles
US4463005A (en) * 1981-03-18 1984-07-31 Imperial Chemical Industries Plc Bicyclic guanidines
DE3269604D1 (en) * 1981-06-26 1986-04-10 Schering Corp Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
JPS61218589A (ja) * 1985-03-26 1986-09-29 Eisai Co Ltd ５―（６―イミダゾ〔１，２―ａ〕ピリジニル）ピリジン誘導体
GB8530878D0 (en) * 1985-12-16 1986-01-29 Fujisawa Pharmaceutical Co Imidazopyridine compounds
GB8514080D0 (en) * 1985-06-04 1985-07-10 Fujisawa Pharmaceutical Co Imidazopyridine compounds
US4725601A (en) * 1985-06-04 1988-02-16 Fujisawa Pharmaceutical Co., Ltd. Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers
EP0228006A1 (en) * 1985-12-16 1987-07-08 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
ES2032455T3 (es) * 1986-01-22 1993-02-16 Synthelabo Procedimiento para preparar derivados de 3-acilaminometil-imidazo (-1,2-a)piridinas.
FR2593818B1 (fr) * 1986-02-05 1988-04-29 Synthelabo Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
US4831041A (en) * 1986-11-26 1989-05-16 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
IL86269A0 (en) * 1987-05-08 1988-11-15 Byk Gulden Lomberg Chem Fab Imidazole derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
PT87988B (pt) * 1987-07-16 1995-05-04 Byk Gulden Lomberg Chem Fab Processo para a preparacao de diazois e de composicoes farmaceuticas que os contem
GB8722488D0 (en) * 1987-09-24 1987-10-28 Fujisawa Pharmaceutical Co Imidazopyridine compound
AT390438B (de) * 1987-10-08 1990-05-10 Yamanouchi Pharma Co Ltd Neue imidazo(1,2-a)pyridinderivate und deren herstellung und diese enthaltende pharmazeutische zubereitungen
WO1990005136A1 (de) * 1988-11-07 1990-05-17 Byk Gulden Lomberg Chemische Fabrik Gmbh Neue imidazopyridine
US5716964A (en) * 1989-12-04 1998-02-10 G.D. Searle & Co. Tetrazolyl substituted imidazo 1,2-a!pyridinylalkyl compounds for treatment of neurotoxic injury
KR910011852A (ko) * 1989-12-04 1991-08-07 폴 디. 매튜카이티스 신경독 장해 치료용 이미다조[1,2-a]피리디닐알킬 화합물
IE904346A1 (en) * 1989-12-04 1991-06-05 Searle & Co IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF¹NEUROTOXIC INJURY
DE4010797A1 (de) * 1990-04-04 1991-10-10 Hoechst Ag Substituierte azole, verfahren zu deren herstellung, diese enthaltende mittel und deren verwendung
US5464843A (en) * 1992-06-23 1995-11-07 G.D. Searle & Co. Imidazo[1,2-a]pyridinyldiacid compounds for cognitive enhancement and for treatment of cognitive disorders and neutrotoxic injury
US5574042A (en) * 1992-11-02 1996-11-12 Fujisawa Pharmaceutical Co., Ltd Imidazo [1,2-a] pyridines and their pharmaceutical use
IL108520A (en) * 1993-02-15 1997-09-30 Byk Gulden Lomberg Chem Fab 2, 3, 8-TRISUBSTITUTED IMIDAZO £1, 2-a| PYRIDINE DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DK0695303T3 (da) * 1993-04-22 2002-03-11 Byk Gulden Lomberg Chem Fab Hidtil ukendte pyridiniumsalte og deres anvendelse til bekæmpelse af Helicobacter-bakterier
UA48122C2 (uk) * 1993-10-11 2002-08-15 Бік Гульден Ломберг Хеміше Фабрік Гмбх АЛКОКСІАЛКІЛКАРБАМАТИ ІМІДАЗО[1,2-а]ПІРИДИНІВ, СПОСІБ ЇХ ОДЕРЖАННЯ ТА ЛІКАРСЬКИЙ ЗАСІБ НА ЇХ ОСНОВІ
WO1996003405A1 (de) * 1994-07-28 1996-02-08 Byk Gulden Lomberg Chemische Fabrik Gmbh Imidazopyridin-azolidinone
WO1996005199A1 (de) * 1994-08-12 1996-02-22 Byk Gulden Lomberg Chemische Fabrik Gmbh Imidazopyridinsalz
EP0822194A4 (en) * 1995-04-21 1998-04-29 Shinnippon Pharmaceutical Inc ANNELLLIED IMIDAZO [1,2-a] PYRIDINE
DE19602855A1 (de) * 1996-01-26 1997-07-31 Byk Gulden Lomberg Chem Fab Neue 3-Methylimidazopyridine
WO1997027193A1 (de) * 1996-01-26 1997-07-31 Byk Gulden Lomberg Chemische Fabrik Gmbh Halogenimidazopyridine
JP2000513710A (ja) * 1996-01-26 2000-10-17 ビイク グルデン ロンベルク ヒエーミツシエ フアブリーク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング ３―メチルイミダゾピリジン
SE9700661D0 (sv) * 1997-02-25 1997-02-25 Astra Ab New compounds
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
SE9802794D0 (sv) 1998-08-21 1998-08-21 Astra Ab New compounds
SE9802793D0 (sv) * 1998-08-21 1998-08-21 Astra Ab New compounds
US6852739B1 (en) 1999-02-26 2005-02-08 Nitromed Inc. Methods using proton pump inhibitors and nitric oxide donors
DE10001037C1 (de) 2000-01-13 2001-12-13 Byk Gulden Lomberg Chem Fab Verfahren und Zwischenprodukte zur Herstellung von Imidazopyridinen
CA2311483A1 (en) 2000-06-12 2001-12-12 Gregory N Beatch IMIDAZO [1,2-A] PYRIDINIC ETHERS AND USES THEREOF
SE0003186D0 (sv) * 2000-09-07 2000-09-07 Astrazeneca Ab New process
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
JP2004520422A (ja) * 2001-03-08 2004-07-08 アストラゼネカ・アクチエボラーグ 新しい用途
SE0102808D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab New compounds
DE10145457A1 (de) 2001-09-14 2003-04-03 Basf Ag Substituierte Imidazo[1,2-a]-5,6,7,8-tetrahydropyridin-8-one, Verfahren zu ihrer Herstellung, sowie deren Verwendung zur Herstellung von Imidazo[1,2,-a]pyridinen
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
US7211590B2 (en) 2002-08-01 2007-05-01 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
SE0301904D0 (sv) 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound II with therapeutic effect
WO2005026164A1 (en) * 2003-09-18 2005-03-24 Altana Pharma Ag Pharmacologically active imidazo[4,5-c]pyridines
EP1974730A1 (en) 2003-11-03 2008-10-01 AstraZeneca AB Imidazo[1,2-a]pyridine derivatives for use in the treatment of sleep disturbance due to silent gastro-esophageal reflux
FI20086158A0 (fi) 2008-12-03 2008-12-03 Mikael Dahlstroem Imidatsopyridiinijohdannaiset
UY34305A (es) 2011-09-01 2013-04-30 Novartis Ag Derivados de heterociclos bicíclicos para el tratamiento de la hipertensión arterial pulmonar
US9073921B2 (en) 2013-03-01 2015-07-07 Novartis Ag Salt forms of bicyclic heterocyclic derivatives
KR101777971B1 (ko) 2016-07-05 2017-09-12 제일약품주식회사 이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4096264A (en) * 1975-12-09 1978-06-20 Merck & Co., Inc. Certain substituted imidazo [1,2-a] pyridines
US4105767A (en) * 1977-03-28 1978-08-08 Merck & Co., Inc. Imidazo [1,2-a] pyridines substituted with a thienyl, thiazolyl, or thiadiazolyl group

Also Published As

Publication number Publication date
AU540840B2 (en) 1984-12-06
CA1167845A (en) 1984-05-22
IL61939A (en) 1986-01-31
FI810147L (fi) 1981-07-24
PT72370B (en) 1982-07-23
MA19048A1 (fr) 1981-10-01
SG70887G (en) 1988-03-04
PT72370A (en) 1981-02-01
JPS56113782A (en) 1981-09-07
NO810198L (no) 1981-07-24
MY8700760A (en) 1987-12-31
HK94187A (en) 1987-12-18
DE3166531D1 (en) 1984-11-15
IL61939A0 (en) 1981-02-27
KR850000240B1 (ko) 1985-03-12
KR830005212A (ko) 1983-08-03
NO157781B (no) 1988-02-08
IE50682B1 (en) 1986-06-11
AU6633781A (en) 1981-07-30
NO157781C (no) 1988-05-25
GR72960B (da) 1984-01-19
IE810108L (en) 1981-07-23
EP0033094A1 (en) 1981-08-05
NZ196071A (en) 1984-05-31
OA06727A (fr) 1982-06-30
HU185857B (en) 1985-04-28
ZA81219B (en) 1982-01-27
EP0033094B1 (en) 1984-10-10

Similar Documents

Publication Publication Date Title
DK25081A (da) Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner
DK138281A (da) Fremgangsmaade til fremstilling af 3-(1-piperidinylalkyl)-4h-pyrido (1,2-a) pyrimidin-4-on-derivater
DK153561C (da) Fremgangsmaade til fremstilling af 1,4-diketopyrrolo-(3,4-c)-pyrroler
DK214685D0 (da) Fremgangsmaade til fremstilling af pyrido-imidazo-rifamyciner
DK157551C (da) Analogifremgangsmaade til fremstilling af 1,3-dihydro-6-methyl-7-hydroxy-furo-(3,4-c)-pyridiner
DK173983D0 (da) Fremgangsmade til fremstilling af imidazo (1,2-alfa)pyridiner
DK194183D0 (da) Fremgangsmade til fremstilling af 2-phenyl-imidazo(4,5-c)pyridiner
DK120783D0 (da) Fremgangsmade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner
DK159878C (da) Fremgangsmaade til fremstilling af 2-amino-3-carbethoxyamino-6-(p-fluor-benzylamino)-pyridin-maleat
DK540984A (da) Fremgangsmaade til fremstilling af 1,2,4-triazolo-(1,5-a)pyrimidin-2-sulfonylchlorider
DK457583D0 (da) Fremgangsmade til fremstilling af dihydropyrazolo(3,4-b)pyridin-derivater
DK457480A (da) Fremgangsmaade til fremstilling af 3,6,7,8-substitueret-s-triazol (4,3-b) pyridaziner
DK390583D0 (da) Fremgangsmade til fremstilling af imidazo(1,2-a)pyrimidiner
DK133482A (da) Fremgangsmaade til fremstilling af imidazo(1,2-a)pyrimidiner
DK200280A (da) Fremgangsmaade til fremstilling af substituerede pyrido (1,2-a) pyrimidiner
DK314682A (da) Fremgangsmaade til fremstilling af substituerede thiazolo-(3,2-a)pyrimidiner
DK17784D0 (da) Fremgangsmade til fremstilling af substituerede pyridiner
DK277682A (da) Fremgangsmaade til fremstilling af substituerede imidazo (1,5-a)pyridiner eller salte deraf
DK114381A (da) Fremgangsmaade til fremstilling af pyrazolopyridinderivater
AR229600A1 (es) Procedimiento para preparar derivados de 1,2,3-triazolo(4,5-b)(1,5)benzodiazepina
DK161706C (da) Fremgangsmaade til fremstilling af pyrido-imidazo-rifamyciner
DE3267918D1 (de) Pyrazolo(3,4-b)pyridine derivatives
DK226881A (da) Fremgangsmaade til fremstilling af 3-picolin
DK269478A (da) Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridinforbindelser
DK253382A (da) Fremgangsmaade til fremstilling af 1,4,9,10-tetrahydro-pyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-oner

Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment