SE8301412L - Substituerade 1h-pyrazolo(1,5)pyrimidiner och forfarande for deras framstellning - Google Patents
Substituerade 1h-pyrazolo(1,5)pyrimidiner och forfarande for deras framstellningInfo
- Publication number
- SE8301412L SE8301412L SE8301412A SE8301412A SE8301412L SE 8301412 L SE8301412 L SE 8301412L SE 8301412 A SE8301412 A SE 8301412A SE 8301412 A SE8301412 A SE 8301412A SE 8301412 L SE8301412 L SE 8301412L
- Authority
- SE
- Sweden
- Prior art keywords
- alkyl
- pyridyl
- substituted
- hydrogen
- image
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8207637 | 1982-03-16 | ||
GB838303089A GB8303089D0 (en) | 1983-02-04 | 1983-02-04 | Substituted 1h-pyrazolo 1,5-a pyrimidines |
Publications (3)
Publication Number | Publication Date |
---|---|
SE8301412D0 SE8301412D0 (sv) | 1983-03-15 |
SE8301412L true SE8301412L (sv) | 1983-09-17 |
SE450573B SE450573B (sv) | 1987-07-06 |
Family
ID=26282260
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE8301412A SE450573B (sv) | 1982-03-16 | 1983-03-15 | 1h-pyrazolo/1,5-a/pyrimidiner, framstellning derav och farmaceutisk komposition |
Country Status (13)
Country | Link |
---|---|
US (1) | US4482555A (sv) |
AU (1) | AU557300B2 (sv) |
CA (1) | CA1192546A (sv) |
CH (1) | CH654306A5 (sv) |
DE (1) | DE3309432A1 (sv) |
DK (1) | DK120783A (sv) |
FI (1) | FI74469C (sv) |
FR (1) | FR2523582B1 (sv) |
IL (1) | IL68133A (sv) |
IT (1) | IT1194555B (sv) |
NL (1) | NL8300934A (sv) |
SE (1) | SE450573B (sv) |
SU (1) | SU1366060A3 (sv) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6245759B1 (en) | 1999-03-11 | 2001-06-12 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
MY125533A (en) | 1999-12-06 | 2006-08-30 | Bristol Myers Squibb Co | Heterocyclic dihydropyrimidine compounds |
EP1782859A3 (en) * | 2003-04-11 | 2009-09-30 | High Point Pharmaceuticals, LLC | Pharmaceutical use of substituted pyrazolo [1,5- a]pyrimidines |
WO2004089471A2 (en) * | 2003-04-11 | 2004-10-21 | Novo Nordisk A/S | NEW PYRAZOLO[1,5-a] PYRIMIDINES DERIVATIVES AND PHARMACEUTICAL USE THEREOF |
US7772232B2 (en) | 2004-04-15 | 2010-08-10 | Bristol-Myers Squibb Company | Quinazolinyl compounds as inhibitors of potassium channel function |
US8138342B2 (en) * | 2004-10-12 | 2012-03-20 | High Point Pharmacueticals, LLC | 11β-hydroxysteroid dehydrogenase type 1 active spiro compounds |
KR20080069189A (ko) * | 2005-11-01 | 2008-07-25 | 트랜스테크 파르마, 인크. | 치환된 아미드의 약학적 사용 |
WO2007051810A2 (en) * | 2005-11-01 | 2007-05-10 | Transtech Pharma | Pharmaceutical use of substituted amides |
WO2007107550A1 (en) * | 2006-03-21 | 2007-09-27 | High Point Pharmaceuticals, Llc | Adamantane derivatives for the treatment of the metabolic syndrome |
US8053447B2 (en) | 2006-04-07 | 2011-11-08 | High Point Pharmaceuticals, Llc | 11β-hydroxysteroid dehydrogenase type 1 active compounds |
WO2007144394A2 (en) * | 2006-06-16 | 2007-12-21 | High Point Pharmaceuticals, Llc. | Pharmaceutical use of substituted piperidine carboxamides |
EP1878721A1 (en) * | 2006-07-13 | 2008-01-16 | Novo Nordisk A/S | 4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors |
CA2657078A1 (en) * | 2006-07-13 | 2008-01-17 | High Point Pharmaceuticals, Llc | 11beta-hydroxysteroid dehydrogenase type 1 active compounds |
ZA200904916B (en) * | 2007-02-23 | 2010-09-29 | High Point Pharmaceuticals Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
US20110003856A1 (en) * | 2007-02-23 | 2011-01-06 | Soren Ebdrup | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
WO2008101885A1 (en) * | 2007-02-23 | 2008-08-28 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
US8334305B2 (en) * | 2007-02-23 | 2012-12-18 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-β-hydroxysteroid dehydrogenase |
JP2010520864A (ja) * | 2007-03-09 | 2010-06-17 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | ヒドロキシステロイドデヒドロゲナーゼインヒビターとしてのインドール−及びベンズイミダゾールアミド類 |
JP2010522766A (ja) * | 2007-03-28 | 2010-07-08 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 11ベータ−hsd1活性化合物 |
CA2683852A1 (en) * | 2007-04-11 | 2008-10-23 | High Point Pharmaceuticals, Llc | Novel compounds |
CA2685036A1 (en) * | 2007-04-24 | 2008-11-06 | High Point Pharmaceuticals, Llc | Pharmaceutical use of substituted amides |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3907799A (en) * | 1971-08-16 | 1975-09-23 | Icn Pharmaceuticals | Xanthine oxidase inhibitors |
BE786611A (fr) * | 1971-08-16 | 1973-01-22 | Int Chem & Nuclear Corp | Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio |
BE792533A (fr) * | 1971-12-09 | 1973-06-08 | Int Chem & Nuclear Corp | Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation |
US3925385A (en) * | 1972-04-20 | 1975-12-09 | Icn Pharmaceuticals | 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines |
US4093617A (en) * | 1974-11-12 | 1978-06-06 | Icn Pharmaceuticals, Inc. | 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines |
US4048184A (en) * | 1976-11-15 | 1977-09-13 | E. R. Squibb & Sons, Inc. | 6-Phenyl-2H-pyrazolo[3,4-b]pyridines |
US4281000A (en) * | 1979-07-09 | 1981-07-28 | American Cyanamid Company | Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents |
-
1983
- 1983-03-09 AU AU12304/83A patent/AU557300B2/en not_active Ceased
- 1983-03-10 US US06/474,205 patent/US4482555A/en not_active Expired - Fee Related
- 1983-03-11 CH CH1325/83A patent/CH654306A5/de not_active IP Right Cessation
- 1983-03-11 IT IT20024/83A patent/IT1194555B/it active
- 1983-03-15 CA CA000423644A patent/CA1192546A/en not_active Expired
- 1983-03-15 SE SE8301412A patent/SE450573B/sv not_active IP Right Cessation
- 1983-03-15 FI FI830864A patent/FI74469C/sv not_active IP Right Cessation
- 1983-03-15 SU SU833565748A patent/SU1366060A3/ru active
- 1983-03-15 NL NL8300934A patent/NL8300934A/xx active Search and Examination
- 1983-03-15 IL IL68133A patent/IL68133A/xx unknown
- 1983-03-15 DK DK120783A patent/DK120783A/da not_active Application Discontinuation
- 1983-03-15 FR FR8304253A patent/FR2523582B1/fr not_active Expired
- 1983-03-16 DE DE19833309432 patent/DE3309432A1/de not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
CH654306A5 (de) | 1986-02-14 |
NL8300934A (nl) | 1983-10-17 |
DE3309432A1 (de) | 1983-09-22 |
US4482555A (en) | 1984-11-13 |
IT1194555B (it) | 1988-09-22 |
SU1366060A3 (ru) | 1988-01-07 |
FI830864A0 (fi) | 1983-03-15 |
IL68133A0 (en) | 1983-06-15 |
AU1230483A (en) | 1983-09-22 |
SE450573B (sv) | 1987-07-06 |
DK120783A (da) | 1983-09-17 |
AU557300B2 (en) | 1986-12-18 |
IT8320024A0 (it) | 1983-03-11 |
FI74469B (fi) | 1987-10-30 |
FR2523582B1 (fr) | 1985-12-06 |
FR2523582A1 (fr) | 1983-09-23 |
SE8301412D0 (sv) | 1983-03-15 |
FI74469C (sv) | 1988-02-08 |
DK120783D0 (da) | 1983-03-15 |
IL68133A (en) | 1985-12-31 |
CA1192546A (en) | 1985-08-27 |
FI830864L (fi) | 1983-09-17 |
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Legal Events
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NUG | Patent has lapsed |
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