FI830864A0 - Foerfarande foer framstaellning av substituerade 1h-pyrazolo/1,5-a/pyramidiner - Google Patents

Foerfarande foer framstaellning av substituerade 1h-pyrazolo/1,5-a/pyramidiner

Info

Publication number
FI830864A0
FI830864A0 FI830864A FI830864A FI830864A0 FI 830864 A0 FI830864 A0 FI 830864A0 FI 830864 A FI830864 A FI 830864A FI 830864 A FI830864 A FI 830864A FI 830864 A0 FI830864 A0 FI 830864A0
Authority
FI
Finland
Prior art keywords
pyramidiner
pyrazolo
substances
frequency refrigeration
refrigeration
Prior art date
Application number
FI830864A
Other languages
English (en)
Other versions
FI74469B (fi
FI74469C (fi
FI830864L (fi
Inventor
Gianfederico Doria
Carlo Passarotti
Ada Buttinoni
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838303089A external-priority patent/GB8303089D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of FI830864A0 publication Critical patent/FI830864A0/fi
Publication of FI830864L publication Critical patent/FI830864L/fi
Publication of FI74469B publication Critical patent/FI74469B/fi
Application granted granted Critical
Publication of FI74469C publication Critical patent/FI74469C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
FI830864A 1982-03-16 1983-03-15 Foerfarande foer framstaellning av substituerade 1h-pyrazolo/1,5-a/pyrimidiner. FI74469C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8207637 1982-03-16
GB8207637 1982-03-16
GB838303089A GB8303089D0 (en) 1983-02-04 1983-02-04 Substituted 1h-pyrazolo 1,5-a pyrimidines
GB8303089 1983-02-04

Publications (4)

Publication Number Publication Date
FI830864A0 true FI830864A0 (fi) 1983-03-15
FI830864L FI830864L (fi) 1983-09-17
FI74469B FI74469B (fi) 1987-10-30
FI74469C FI74469C (fi) 1988-02-08

Family

ID=26282260

Family Applications (1)

Application Number Title Priority Date Filing Date
FI830864A FI74469C (fi) 1982-03-16 1983-03-15 Foerfarande foer framstaellning av substituerade 1h-pyrazolo/1,5-a/pyrimidiner.

Country Status (13)

Country Link
US (1) US4482555A (fi)
AU (1) AU557300B2 (fi)
CA (1) CA1192546A (fi)
CH (1) CH654306A5 (fi)
DE (1) DE3309432A1 (fi)
DK (1) DK120783A (fi)
FI (1) FI74469C (fi)
FR (1) FR2523582B1 (fi)
IL (1) IL68133A (fi)
IT (1) IT1194555B (fi)
NL (1) NL8300934A (fi)
SE (1) SE450573B (fi)
SU (1) SU1366060A3 (fi)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6245759B1 (en) * 1999-03-11 2001-06-12 Merck & Co., Inc. Tyrosine kinase inhibitors
MY125533A (en) 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
EP1782859A3 (en) * 2003-04-11 2009-09-30 High Point Pharmaceuticals, LLC Pharmaceutical use of substituted pyrazolo [1,5- a]pyrimidines
EP1615697A2 (en) * 2003-04-11 2006-01-18 Novo Nordisk A/S New pyrazolo[1,5-a] pyrimidine derivatives and pharmaceutical use thereof
US7772232B2 (en) 2004-04-15 2010-08-10 Bristol-Myers Squibb Company Quinazolinyl compounds as inhibitors of potassium channel function
EP1802623A1 (en) * 2004-10-12 2007-07-04 Novo Nordisk A/S 11beta-hydroxysteroid dehydrogenase type 1 active spiro compounds
JP2009514818A (ja) * 2005-11-01 2009-04-09 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー 置換アミドの製薬学的用途
EP1945207A2 (en) * 2005-11-01 2008-07-23 Transtech Pharma, Inc. Pharmaceutical use of substituted amides
US20100168083A1 (en) * 2006-03-21 2010-07-01 Soren Ebdrup Adamantane derivatives for the treatment of the metabolic syndrome
BRPI0710669A2 (pt) 2006-04-07 2011-08-16 High Point Pharmaceuticals Llc compostos ativos de dehidrogenase de 11b-hidroxiesteróide tipo 1
US20090306048A1 (en) * 2006-06-16 2009-12-10 John Paul Kilburn Pharmaceutical use of substituted piperidine carboxamides
US8048908B2 (en) * 2006-07-13 2011-11-01 High Point Pharmaceuticals, Llc 11β-hydroxysteroid dehydrogenase type 1 active compounds
EP1878721A1 (en) * 2006-07-13 2008-01-16 Novo Nordisk A/S 4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors
WO2008101907A2 (en) * 2007-02-23 2008-08-28 High Point Pharmaceuticals, Llc N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EP2125704A1 (en) * 2007-02-23 2009-12-02 High Point Pharmaceuticals, LLC N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
AU2008219326B2 (en) * 2007-02-23 2012-12-13 Vtv Therapeutics Llc N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
WO2008101885A1 (en) * 2007-02-23 2008-08-28 High Point Pharmaceuticals, Llc N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
CA2679866A1 (en) * 2007-03-09 2008-09-18 High Point Pharmaceuticals, Llc Indole- and benzimidazole amides as hydroxysteroid dehydrogenase inhibitors
JP2010522766A (ja) * 2007-03-28 2010-07-08 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー 11ベータ−hsd1活性化合物
US20100137377A1 (en) * 2007-04-11 2010-06-03 Soren Ebdrup Et Al Novel compounds
CA2685036A1 (en) * 2007-04-24 2008-11-06 High Point Pharmaceuticals, Llc Pharmaceutical use of substituted amides

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
BE786611A (fr) * 1971-08-16 1973-01-22 Int Chem & Nuclear Corp Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio
BE792533A (fr) * 1971-12-09 1973-06-08 Int Chem & Nuclear Corp Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US3925385A (en) * 1972-04-20 1975-12-09 Icn Pharmaceuticals 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines
US4093617A (en) * 1974-11-12 1978-06-06 Icn Pharmaceuticals, Inc. 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines
US4048184A (en) * 1976-11-15 1977-09-13 E. R. Squibb & Sons, Inc. 6-Phenyl-2H-pyrazolo[3,4-b]pyridines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents

Also Published As

Publication number Publication date
SU1366060A3 (ru) 1988-01-07
IL68133A (en) 1985-12-31
SE8301412L (sv) 1983-09-17
DK120783A (da) 1983-09-17
FI74469B (fi) 1987-10-30
IT8320024A0 (it) 1983-03-11
IL68133A0 (en) 1983-06-15
DE3309432A1 (de) 1983-09-22
FR2523582B1 (fr) 1985-12-06
AU1230483A (en) 1983-09-22
DK120783D0 (da) 1983-03-15
SE450573B (sv) 1987-07-06
CA1192546A (en) 1985-08-27
CH654306A5 (de) 1986-02-14
SE8301412D0 (sv) 1983-03-15
FI74469C (fi) 1988-02-08
IT1194555B (it) 1988-09-22
NL8300934A (nl) 1983-10-17
FI830864L (fi) 1983-09-17
FR2523582A1 (fr) 1983-09-23
US4482555A (en) 1984-11-13
AU557300B2 (en) 1986-12-18

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A