DK1173205T3 - Oral formulering til ileum-indgivelse, omfattende en forbindelse til inhibering af ileum-galdesyretransporten - Google Patents

Oral formulering til ileum-indgivelse, omfattende en forbindelse til inhibering af ileum-galdesyretransporten

Info

Publication number
DK1173205T3
DK1173205T3 DK00928046T DK00928046T DK1173205T3 DK 1173205 T3 DK1173205 T3 DK 1173205T3 DK 00928046 T DK00928046 T DK 00928046T DK 00928046 T DK00928046 T DK 00928046T DK 1173205 T3 DK1173205 T3 DK 1173205T3
Authority
DK
Denmark
Prior art keywords
ileum
bile acid
inhibitor compound
compound
inhibiting
Prior art date
Application number
DK00928046T
Other languages
Danish (da)
English (en)
Inventor
Ann-Margret Lindqvist
Bertil Abrahamsson
Anna-Lena Ungell
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of DK1173205T3 publication Critical patent/DK1173205T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
DK00928046T 1999-04-19 2000-04-19 Oral formulering til ileum-indgivelse, omfattende en forbindelse til inhibering af ileum-galdesyretransporten DK1173205T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9901387A SE9901387D0 (sv) 1999-04-19 1999-04-19 New pharmaceutical foromaulations
PCT/SE2000/000755 WO2000062810A1 (en) 1999-04-19 2000-04-19 An oral formulation for ileum administering comprising an inhibitor compound of the ileal bile acid transport
EP00928046A EP1173205B1 (en) 1999-04-19 2000-04-19 An oral formulation for ileum administering comprising an inhibitor compound of the ileal bile acid transport

Publications (1)

Publication Number Publication Date
DK1173205T3 true DK1173205T3 (da) 2005-08-08

Family

ID=20415263

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00928046T DK1173205T3 (da) 1999-04-19 2000-04-19 Oral formulering til ileum-indgivelse, omfattende en forbindelse til inhibering af ileum-galdesyretransporten

Country Status (27)

Country Link
EP (1) EP1173205B1 (et)
JP (1) JP2002542208A (et)
KR (1) KR20010108516A (et)
CN (1) CN1348384A (et)
AT (1) ATE296641T1 (et)
AU (1) AU767425B2 (et)
BR (1) BR0009835A (et)
CA (1) CA2379105A1 (et)
CZ (1) CZ20013743A3 (et)
DE (1) DE60020551T2 (et)
DK (1) DK1173205T3 (et)
EE (1) EE04607B1 (et)
ES (1) ES2241603T3 (et)
HK (1) HK1042850A1 (et)
HU (1) HUP0200793A3 (et)
IL (1) IL145871A0 (et)
IS (1) IS2161B (et)
NO (1) NO20015063D0 (et)
NZ (1) NZ514264A (et)
PL (1) PL351186A1 (et)
PT (1) PT1173205E (et)
SE (1) SE9901387D0 (et)
SI (1) SI1173205T1 (et)
SK (1) SK15282001A3 (et)
TR (1) TR200103033T2 (et)
WO (1) WO2000062810A1 (et)
ZA (1) ZA200108539B (et)

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GB0121337D0 (en) 2001-09-04 2001-10-24 Astrazeneca Ab Chemical compounds
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GB0209467D0 (en) 2002-04-25 2002-06-05 Astrazeneca Ab Chemical compounds
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GB0216321D0 (en) * 2002-07-13 2002-08-21 Astrazeneca Ab Therapeutic treatment
GB0304194D0 (en) 2003-02-25 2003-03-26 Astrazeneca Ab Chemical compounds
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RU2015126651A (ru) 2012-12-10 2017-01-16 Фред Хатчинсон Кэнсер Рисёрч Сентер Способы скрининга
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US11559580B1 (en) 2013-09-17 2023-01-24 Blaze Bioscience, Inc. Tissue-homing peptide conjugates and methods of use thereof
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CN105362244A (zh) * 2015-11-26 2016-03-02 青岛海之源智能技术有限公司 考来烯胺缓释片及制备方法
RU2750937C2 (ru) 2016-02-09 2021-07-06 Альбирео Аб Пероральный состав холестирамина и его применение
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
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ES2874669T3 (es) 2016-02-09 2021-11-05 Albireo Ab Formulación oral de colestiramina y uso de la misma
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JP2023504643A (ja) 2019-12-04 2023-02-06 アルビレオ・アクチボラグ ベンゾチア(ジ)アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
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JP2023537285A (ja) 2020-08-03 2023-08-31 アルビレオ・アクチボラグ ベンゾチア(ジ)アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
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Also Published As

Publication number Publication date
ZA200108539B (en) 2003-01-17
NO20015063L (no) 2001-10-18
EE04607B1 (et) 2006-04-17
EP1173205A1 (en) 2002-01-23
CN1348384A (zh) 2002-05-08
ATE296641T1 (de) 2005-06-15
EE200100545A (et) 2003-02-17
HK1042850A1 (en) 2002-08-30
WO2000062810A1 (en) 2000-10-26
CZ20013743A3 (cs) 2002-01-16
IL145871A0 (en) 2002-07-25
EP1173205B1 (en) 2005-06-01
BR0009835A (pt) 2002-01-08
DE60020551D1 (de) 2005-07-07
CA2379105A1 (en) 2000-10-26
NZ514264A (en) 2003-10-31
AU767425B2 (en) 2003-11-13
JP2002542208A (ja) 2002-12-10
SI1173205T1 (en) 2005-10-31
IS2161B (is) 2006-11-15
PT1173205E (pt) 2005-10-31
KR20010108516A (ko) 2001-12-07
DE60020551T2 (de) 2006-03-23
HUP0200793A3 (en) 2004-07-28
HUP0200793A2 (hu) 2002-07-29
ES2241603T3 (es) 2005-11-01
AU4633500A (en) 2000-11-02
TR200103033T2 (tr) 2002-03-21
NO20015063D0 (no) 2001-10-18
PL351186A1 (en) 2003-03-24
SE9901387D0 (sv) 1999-04-19
IS6109A (is) 2001-10-16
SK15282001A3 (sk) 2002-04-04

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