DK1129093T3 - Pyrazolopyrimidinonderivater til behandling af impotens - Google Patents

Pyrazolopyrimidinonderivater til behandling af impotens

Info

Publication number
DK1129093T3
DK1129093T3 DK99954478T DK99954478T DK1129093T3 DK 1129093 T3 DK1129093 T3 DK 1129093T3 DK 99954478 T DK99954478 T DK 99954478T DK 99954478 T DK99954478 T DK 99954478T DK 1129093 T3 DK1129093 T3 DK 1129093T3
Authority
DK
Denmark
Prior art keywords
impotence
treatment
derivatives
pyrazolopyrimidinone derivatives
pyrazolopyrimidinone
Prior art date
Application number
DK99954478T
Other languages
English (en)
Inventor
Moohi Yoo
Dong Sung Kim
Ik Yon Kim
M Yoo
Wonbae Kim
Min Sun Chang
Joong In Lim
D S Kim
I Y Kim
Tae Kyun Lim
Byoung Ok Ahn
Kyung Koo Kang
Miwon Son
Hyounmie Doh
Soonhoe Kim
Hyunjoo Shim
Taeyoung Oh
Heungjae Kim
Dong Goo Kim
Original Assignee
Dong A Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27349839&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1129093(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dong A Pharm Co Ltd filed Critical Dong A Pharm Co Ltd
Application granted granted Critical
Publication of DK1129093T3 publication Critical patent/DK1129093T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK99954478T 1998-11-11 1999-11-10 Pyrazolopyrimidinonderivater til behandling af impotens DK1129093T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
KR19980048100 1998-11-11
KR19990014972 1999-04-27
KR19990049384A KR100353014B1 (ko) 1998-11-11 1999-11-09 발기부전 치료에 효과를 갖는 피라졸로피리미디논 화합물
PCT/KR1999/000675 WO2000027848A1 (en) 1998-11-11 1999-11-10 Pyrazolopyrimidinone derivatives for the treatment of impotence

Publications (1)

Publication Number Publication Date
DK1129093T3 true DK1129093T3 (da) 2003-10-20

Family

ID=27349839

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99954478T DK1129093T3 (da) 1998-11-11 1999-11-10 Pyrazolopyrimidinonderivater til behandling af impotens

Country Status (17)

Country Link
US (1) US6583147B1 (da)
EP (1) EP1129093B1 (da)
JP (1) JP3577630B2 (da)
KR (1) KR100353014B1 (da)
CN (1) CN1136219C (da)
AT (1) ATE245650T1 (da)
AU (1) AU760422B2 (da)
BR (1) BRPI9915822B8 (da)
CA (1) CA2350538C (da)
DE (1) DE69909818T2 (da)
DK (1) DK1129093T3 (da)
ES (1) ES2204169T3 (da)
HK (1) HK1039328B (da)
NZ (1) NZ511015A (da)
PT (1) PT1129093E (da)
TR (1) TR200101335T2 (da)
WO (1) WO2000027848A1 (da)

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US7649002B2 (en) 2004-02-04 2010-01-19 Pfizer Inc (3,5-dimethylpiperidin-1yl)(4-phenylpyrrolidin-3-yl)methanone derivatives as MCR4 agonists
JP2008530247A (ja) * 2005-02-18 2008-08-07 サーフェイス ロジックス，インコーポレイティド 薬物動態学的に改善された化合物
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DK2366393T3 (da) 2005-04-19 2013-10-21 Takeda Gmbh Roflumilast til behandlingen af pulmonal hypertension
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NZ571673A (en) * 2006-04-04 2011-08-26 Dong A Pharm Co Ltd A pyrazolopyrimidinone derivative for the prevention and treatment of prostatic hyperplasia
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AR062501A1 (es) 2006-08-29 2008-11-12 Actelion Pharmaceuticals Ltd Composiciones terapeuticas
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US20090197899A1 (en) * 2006-10-20 2009-08-06 Concert Pharmaceuticals Inc. 3-(Dihydro-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-propoxybenzenesulfonamide Derivatives and Methods of Use
US20090270425A1 (en) * 2006-10-20 2009-10-29 Concert Pharmaceuticals Inc. 3-(dihydro-1h-pyrazolo[4,3-d]pyrimidin-5-yl)-4-propoxybenzenesulfonamide derivatives and methods of use
EP2089392A4 (en) * 2006-10-20 2010-05-05 Concert Pharmaceuticals Inc 3- (DIHYDRO-1H-PYRAZOLO Ý4,3-D¨PYRIMIDIN-5-YL) -4-PROPOXYBENZENESULFONAMIDE DERIVATIVES AND METHODS OF USE
US20080194529A1 (en) * 2007-02-12 2008-08-14 Auspex Pharmaceuticals, Inc. HIGHLY SELECTIVE and LONG-ACTING PDE5 MODULATORS
ES2618315T3 (es) 2007-05-25 2017-06-21 Ipsen Pharma S.A.S. Ligandos del receptor de melanocortina modificados con hidantoína
US8604245B2 (en) 2007-06-04 2013-12-10 Ben-Gurion University Of The Negev Research And Development Authority Tri-aryl compounds and compositions comprising the same
KR101002490B1 (ko) * 2007-06-09 2010-12-17 동아제약주식회사 유데나필을 유효성분으로 함유하는 만성 심부전증 치료용약학적 조성물
KR100920125B1 (ko) * 2007-10-02 2009-10-01 동아제약주식회사 양성 전립선 비대증 치료를 위한 피라졸로피리미디논화합물 및 알파 아드레날린성 수용체 길항제를 함유하는약제학적 배합물
JP2010540621A (ja) * 2007-10-02 2010-12-24 ドン ア ファーマシューティカル カンパニー リミテッド 良性前立腺肥大症および下部尿路症状の治療または予防用組成物、およびその治療または予防方法
WO2009099620A1 (en) * 2008-02-04 2009-08-13 Concert Pharmaceuticals Inc. 3-(dihydro-1h-pyrazolo[4,3-d]pyrimidin-5-yl)-4-propoxybenzenesulfonamide derivatives and methods of use
KR20090087795A (ko) * 2008-02-13 2009-08-18 한양대학교 산학협력단 혈관 재협착 예방 및 치료를 위한 약학 조성물 및 이를포함하는 스텐트
KR101071877B1 (ko) * 2009-02-18 2011-10-10 동아제약주식회사 유데나필 산부가염, 그의 제조방법 및 이를 포함하는 약학적 조성물
GB0903493D0 (en) 2009-02-27 2009-04-08 Vantia Ltd New compounds
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CN102952138B (zh) * 2011-08-17 2016-07-06 上海特化医药科技有限公司 一种吡唑并嘧啶酮化合物的盐、多晶型物及其药物组合物、制备方法和应用
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KR101953735B1 (ko) 2012-12-14 2019-03-04 한미약품 주식회사 포스포다이에스터라제-5 억제제를 포함하는 츄정
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EP3180008B1 (en) * 2014-08-12 2023-11-29 Mezzion Pharma Co., Ltd. Methods of improving myocardial performance in fontan patients using udenafil compositions
KR101645652B1 (ko) 2014-11-03 2016-08-08 (주)퓨젠바이오농업회사법인 세리포리아 락세라타에 의해 생산되는 세포외다당체를 유효성분으로 함유하는 성기능개선용 조성물
WO2017168174A1 (en) 2016-04-02 2017-10-05 N4 Pharma Uk Limited New pharmaceutical forms of sildenafil
CN107759603B (zh) * 2016-08-18 2020-09-01 四川科伦药物研究院有限公司 一种杂环化合物的制备方法
CN113493459B (zh) * 2020-04-07 2022-12-13 广州白云山医药集团股份有限公司白云山制药总厂 Pde5抑制剂化合物及其制备方法和应用
WO2022123310A1 (en) 2020-12-11 2022-06-16 Ildong Pharmaceutical Co., Ltd. Novel compounds as androgen receptor and phosphodiesterase dual inhibitor

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Also Published As

Publication number Publication date
BRPI9915822B8 (pt) 2021-05-25
CA2350538A1 (en) 2000-05-18
DE69909818T2 (de) 2004-05-27
EP1129093A1 (en) 2001-09-05
WO2000027848A1 (en) 2000-05-18
HK1039328A1 (en) 2002-04-19
BR9915822A (pt) 2001-08-14
CN1136219C (zh) 2004-01-28
EP1129093B1 (en) 2003-07-23
JP3577630B2 (ja) 2004-10-13
AU1081700A (en) 2000-05-29
CA2350538C (en) 2005-06-28
ES2204169T3 (es) 2004-04-16
HK1039328B (zh) 2004-06-25
CN1325398A (zh) 2001-12-05
US6583147B1 (en) 2003-06-24
NZ511015A (en) 2003-09-26
BR9915822B1 (pt) 2013-08-27
DE69909818D1 (de) 2003-08-28
KR20000035324A (ko) 2000-06-26
AU760422B2 (en) 2003-05-15
ATE245650T1 (de) 2003-08-15
JP2002529467A (ja) 2002-09-10
KR100353014B1 (ko) 2002-09-18
TR200101335T2 (tr) 2001-09-21
PT1129093E (pt) 2003-12-31

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