BR9915822A - Derivados de pirazolopirimidinona para o tratamento de impotência - Google Patents

Derivados de pirazolopirimidinona para o tratamento de impotência

Info

Publication number
BR9915822A
BR9915822A BR9915822-1A BR9915822A BR9915822A BR 9915822 A BR9915822 A BR 9915822A BR 9915822 A BR9915822 A BR 9915822A BR 9915822 A BR9915822 A BR 9915822A
Authority
BR
Brazil
Prior art keywords
impotence
treatment
derivatives
pyrazolopyrimidinone derivatives
pyrazolopyrimidinone
Prior art date
Application number
BR9915822-1A
Other languages
English (en)
Other versions
BRPI9915822B8 (pt
BR9915822B1 (pt
Inventor
Moohi Yoo
Wonbae Kim
Min Sun Chang
Joong In Lim
Dong Sung Kim
Yk Yon Kim
Tae Kyun Lim
Byoung Ok Ahn
Kyung Koo Kang
Miwon Son
Hyounmie Doh
Soonhoe Kim
Hyunjoo Shim
Taeyoung Oh
Heungjae Kim
Dong Goo Kim
Original Assignee
Dong A Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27349839&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9915822(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dong A Pharm Co Ltd filed Critical Dong A Pharm Co Ltd
Publication of BR9915822A publication Critical patent/BR9915822A/pt
Publication of BR9915822B1 publication Critical patent/BR9915822B1/pt
Publication of BRPI9915822B8 publication Critical patent/BRPI9915822B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Patente Invenção: <B>''DERIVADOS DE PIRAZOLOPIRIMIDINONA PARA O TRATAMENTO DE IMPOTêNCIA''<D>. A presente invenção refere-se a derivados de pirazolopirimidinona de fórmula 1, seu método de preparação e composições farmacêuticas contendo os ditos derivados. Os compostos têm eficácia no tratamento de impotência, uma das disfunções sexuais do macho com os efeitos colaterais reduzidos.
BRPI9915822A 1998-11-11 1999-11-10 derivados de pirazolopirimidinona e sua composição farmacêutica para o tratamento de impotência BRPI9915822B8 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
KR19980048100 1998-11-11
KR19990014972 1999-04-27
KR19990049384A KR100353014B1 (ko) 1998-11-11 1999-11-09 발기부전 치료에 효과를 갖는 피라졸로피리미디논 화합물
PCT/KR1999/000675 WO2000027848A1 (en) 1998-11-11 1999-11-10 Pyrazolopyrimidinone derivatives for the treatment of impotence

Publications (3)

Publication Number Publication Date
BR9915822A true BR9915822A (pt) 2001-08-14
BR9915822B1 BR9915822B1 (pt) 2013-08-27
BRPI9915822B8 BRPI9915822B8 (pt) 2021-05-25

Family

ID=27349839

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9915822A BRPI9915822B8 (pt) 1998-11-11 1999-11-10 derivados de pirazolopirimidinona e sua composição farmacêutica para o tratamento de impotência

Country Status (17)

Country Link
US (1) US6583147B1 (pt)
EP (1) EP1129093B1 (pt)
JP (1) JP3577630B2 (pt)
KR (1) KR100353014B1 (pt)
CN (1) CN1136219C (pt)
AT (1) ATE245650T1 (pt)
AU (1) AU760422B2 (pt)
BR (1) BRPI9915822B8 (pt)
CA (1) CA2350538C (pt)
DE (1) DE69909818T2 (pt)
DK (1) DK1129093T3 (pt)
ES (1) ES2204169T3 (pt)
HK (1) HK1039328B (pt)
NZ (1) NZ511015A (pt)
PT (1) PT1129093E (pt)
TR (1) TR200101335T2 (pt)
WO (1) WO2000027848A1 (pt)

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EP1874309A1 (en) 2005-04-19 2008-01-09 Nycomed GmbH Roflumilast for the treatment of pulmonary hypertension
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WO2007114534A1 (en) * 2006-04-04 2007-10-11 Dong-A Pharmaceutical.Co., Ltd. Agent for the prevention and treatment of prostatic hyperplasia comprising pyrazolopyrimidinone compound
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US20090197899A1 (en) * 2006-10-20 2009-08-06 Concert Pharmaceuticals Inc. 3-(Dihydro-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-propoxybenzenesulfonamide Derivatives and Methods of Use
WO2008100886A1 (en) * 2007-02-12 2008-08-21 Auspex Pharmaceuticals, Inc. Preparation and use of deuterated udenafil analogues as highly selective pde5 modulators for the treatment of erectile dysfunction
TWI364290B (en) 2007-05-25 2012-05-21 Ipsen Pharma Sas Melanocortin receptor ligands modifled with hydantoin
CA2690004C (en) 2007-06-04 2018-01-23 Ben-Gurion University Of The Negev Research And Development Authority Tri-aryl compounds and compositions comprising the same
KR101002490B1 (ko) * 2007-06-09 2010-12-17 동아제약주식회사 유데나필을 유효성분으로 함유하는 만성 심부전증 치료용약학적 조성물
JP2010540621A (ja) * 2007-10-02 2010-12-24 ドン ア ファーマシューティカル カンパニー リミテッド 良性前立腺肥大症および下部尿路症状の治療または予防用組成物、およびその治療または予防方法
KR100920125B1 (ko) * 2007-10-02 2009-10-01 동아제약주식회사 양성 전립선 비대증 치료를 위한 피라졸로피리미디논화합물 및 알파 아드레날린성 수용체 길항제를 함유하는약제학적 배합물
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KR20160094956A (ko) 2013-11-05 2016-08-10 벤-구리온 유니버시티 오브 더 네게브 리서치 앤드 디벨럽먼트 어쏘러티 당뇨병 및 당뇨병으로부터 발생하는 합병증 질환의 치료를 위한 화합물
KR20230116098A (ko) 2014-08-12 2023-08-03 주식회사 메지온 유데나필 조성물을 이용하여 폰탄 환자에서 심근 성능을개선시키는 방법
KR101645652B1 (ko) 2014-11-03 2016-08-08 (주)퓨젠바이오농업회사법인 세리포리아 락세라타에 의해 생산되는 세포외다당체를 유효성분으로 함유하는 성기능개선용 조성물
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Also Published As

Publication number Publication date
CN1325398A (zh) 2001-12-05
DE69909818T2 (de) 2004-05-27
NZ511015A (en) 2003-09-26
AU760422B2 (en) 2003-05-15
WO2000027848A1 (en) 2000-05-18
JP3577630B2 (ja) 2004-10-13
EP1129093B1 (en) 2003-07-23
HK1039328B (zh) 2004-06-25
EP1129093A1 (en) 2001-09-05
HK1039328A1 (en) 2002-04-19
CN1136219C (zh) 2004-01-28
ATE245650T1 (de) 2003-08-15
CA2350538A1 (en) 2000-05-18
US6583147B1 (en) 2003-06-24
KR100353014B1 (ko) 2002-09-18
KR20000035324A (ko) 2000-06-26
DK1129093T3 (da) 2003-10-20
JP2002529467A (ja) 2002-09-10
BRPI9915822B8 (pt) 2021-05-25
BR9915822B1 (pt) 2013-08-27
PT1129093E (pt) 2003-12-31
TR200101335T2 (tr) 2001-09-21
AU1081700A (en) 2000-05-29
CA2350538C (en) 2005-06-28
DE69909818D1 (de) 2003-08-28
ES2204169T3 (es) 2004-04-16

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