DK0688772T3 - Quinolincarboxylsyrederivater med 7-(4-aminomethyl-3-oxim)-pyrrolidinsubstituenter og fremgangsmåde til deres fremstilling - Google Patents

Quinolincarboxylsyrederivater med 7-(4-aminomethyl-3-oxim)-pyrrolidinsubstituenter og fremgangsmåde til deres fremstilling

Info

Publication number
DK0688772T3
DK0688772T3 DK95250143T DK95250143T DK0688772T3 DK 0688772 T3 DK0688772 T3 DK 0688772T3 DK 95250143 T DK95250143 T DK 95250143T DK 95250143 T DK95250143 T DK 95250143T DK 0688772 T3 DK0688772 T3 DK 0688772T3
Authority
DK
Denmark
Prior art keywords
aminomethyl
oxime
preparation
carboxylic acid
acid derivatives
Prior art date
Application number
DK95250143T
Other languages
Danish (da)
English (en)
Inventor
Jin Hwan Kwak
Yi Na Jeong
Jeong In Oh
Se Ho Kim
Hoon Choi
Do Hyun Nam
Chang Yong Hong
Young Kwan Kim
Jay Hyok Chang
Mu Yong Kim
Original Assignee
Lg Chemical Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from KR1019940013604A external-priority patent/KR0131999B1/ko
Priority claimed from KR1019940039915A external-priority patent/KR100222082B1/ko
Priority claimed from KR1019940039930A external-priority patent/KR100222083B1/ko
Application filed by Lg Chemical Ltd filed Critical Lg Chemical Ltd
Application granted granted Critical
Publication of DK0688772T3 publication Critical patent/DK0688772T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK95250143T 1994-06-16 1995-06-14 Quinolincarboxylsyrederivater med 7-(4-aminomethyl-3-oxim)-pyrrolidinsubstituenter og fremgangsmåde til deres fremstilling DK0688772T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR1019940013604A KR0131999B1 (ko) 1994-06-16 1994-06-16 7-(4-아미노메틸-3-옥심)피롤리딘 치환제를 갖는 신규 퀴놀린 카르복실산 유도체 및 그의 제조방법
KR1019940039915A KR100222082B1 (ko) 1994-12-30 1994-12-30 7-(3-아미노메틸-4-알킬옥심)피롤리딘 치환체를 갖는 신규 퀴놀린 카복실산 유도체 및 그의 제조방법
KR1019940039930A KR100222083B1 (ko) 1994-12-30 1994-12-30 7-(3-아미노메틸-4-벤질옥심) 피롤리딘 치환체를 갖는 신규 퀴놀린 카복실산 유도체

Publications (1)

Publication Number Publication Date
DK0688772T3 true DK0688772T3 (da) 1999-11-01

Family

ID=27349079

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95250143T DK0688772T3 (da) 1994-06-16 1995-06-14 Quinolincarboxylsyrederivater med 7-(4-aminomethyl-3-oxim)-pyrrolidinsubstituenter og fremgangsmåde til deres fremstilling

Country Status (8)

Country Link
US (5) US5633262A (ja)
EP (1) EP0688772B1 (ja)
JP (1) JP2742248B2 (ja)
CN (1) CN1058010C (ja)
CA (1) CA2151890C (ja)
DE (1) DE69509442T2 (ja)
DK (1) DK0688772T3 (ja)
UA (1) UA54365C2 (ja)

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CN102329315A (zh) * 2011-07-22 2012-01-25 中国医学科学院医药生物技术研究所 含有氟甲氧亚氨基取代的萘啶酮羧酸类化合物及其制备方法
CN103467448B (zh) * 2013-09-18 2015-04-15 浙江司太立制药股份有限公司 7-(3-氨基-4-烷氧亚胺基-1-哌啶基)-1-[(1r,2s)-2-氟环丙基]喹诺酮羧酸类化合物及其制备方法
CN103483315B (zh) * 2013-09-18 2015-07-01 浙江司太立制药股份有限公司 7-(3-氨甲基-4-烷氧亚胺基-1-吡咯烷基)-1-[(1r,2s)-2-氟环丙基]喹诺酮羧酸类化合物及其制备方法
KR102213991B1 (ko) * 2014-05-20 2021-02-09 동화약품주식회사 개선된 자보플록사신의 제조방법
JP6574474B2 (ja) * 2014-07-21 2019-09-11 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． キラルジペプチジルペプチダーゼ−ｉｖ阻害剤の製造方法
CN105585518B (zh) * 2014-10-23 2018-04-24 华仁药业股份有限公司 一种吉米沙星中间体的制备方法
CN104892600B (zh) * 2015-06-04 2017-02-01 浙江司太立制药股份有限公司 7‑（3‑氨甲基‑4‑取代苄氧亚胺基‑1‑吡咯烷基）萘啶酮羧酸类化合物

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Also Published As

Publication number Publication date
JPH0841050A (ja) 1996-02-13
UA54365C2 (uk) 2003-03-17
US5633262A (en) 1997-05-27
US5698570A (en) 1997-12-16
CA2151890C (en) 1999-01-12
CN1114959A (zh) 1996-01-17
EP0688772B1 (en) 1999-05-06
CN1058010C (zh) 2000-11-01
JP2742248B2 (ja) 1998-04-22
EP0688772A1 (en) 1995-12-27
CA2151890A1 (en) 1995-12-17
DE69509442D1 (de) 1999-06-10
US5869670A (en) 1999-02-09
US5962468A (en) 1999-10-05
DE69509442T2 (de) 1999-09-02
US5840916A (en) 1998-11-24

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