DK0416410T3 - Piperaziniocephalosporiner - Google Patents
PiperaziniocephalosporinerInfo
- Publication number
- DK0416410T3 DK0416410T3 DK90116330.3T DK90116330T DK0416410T3 DK 0416410 T3 DK0416410 T3 DK 0416410T3 DK 90116330 T DK90116330 T DK 90116330T DK 0416410 T3 DK0416410 T3 DK 0416410T3
- Authority
- DK
- Denmark
- Prior art keywords
- alkyl
- same
- antibacterial
- hydroxyarylpiperaziniocephalosporins
- cephalosporins
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP23263189 | 1989-09-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0416410T3 true DK0416410T3 (da) | 1995-05-15 |
Family
ID=16942341
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK90116330.3T DK0416410T3 (da) | 1989-09-07 | 1990-08-26 | Piperaziniocephalosporiner |
Country Status (7)
Country | Link |
---|---|
US (1) | US5143910A (fr) |
EP (1) | EP0416410B1 (fr) |
JP (1) | JP2969283B2 (fr) |
KR (1) | KR0158452B1 (fr) |
AT (1) | ATE114658T1 (fr) |
DE (1) | DE69014490T2 (fr) |
DK (1) | DK0416410T3 (fr) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0492277A3 (en) * | 1990-12-20 | 1992-10-14 | F. Hoffmann-La Roche Ag | Cephalosporin derivatives |
EP0550775A1 (fr) * | 1992-01-07 | 1993-07-14 | F. Hoffmann-La Roche Ag | Dérivés de céphalosporine |
JP3081773B2 (ja) * | 1995-03-31 | 2000-08-28 | 株式会社資生堂 | N−アシルピペラジン誘導体及び抗菌剤、抗潰瘍剤 |
JP4189043B2 (ja) * | 1996-09-30 | 2008-12-03 | 株式会社資生堂 | N−アシルピペラジン誘導体及び抗菌剤、抗潰瘍剤 |
US6479495B1 (en) | 1997-09-29 | 2002-11-12 | Aventis Pharmaceuticals Inc. | Aminoalkylphenol derivatives and related compounds |
CA2302412C (fr) * | 1997-09-29 | 2005-12-20 | Aventis Pharmaceuticals Inc. | Derives d'amino-alkylphenols et composes associes |
AU2004264342A1 (en) * | 2003-08-05 | 2005-02-24 | Georgetown University | Sigma-1 receptor ligand with acetylcholinesterase inhibition properties |
US20060247248A1 (en) * | 2003-08-05 | 2006-11-02 | Vassilios Papadopoulos | Sigma-1 receptor ligand with acetylcholinesterase |
EP2065057A3 (fr) * | 2006-03-15 | 2009-08-12 | Mallinckrodt Inc. | Conjugués chélatants dotés d'un groupe aromatique et dérivés associés |
US8883772B2 (en) | 2007-10-09 | 2014-11-11 | Sopharmia, Inc. | Broad spectrum beta-lactamase inhibitors |
PT2960244T (pt) | 2008-10-31 | 2016-11-02 | Shionogi & Co | Cefalosporina contendo grupo catecol |
US8883773B2 (en) | 2010-04-05 | 2014-11-11 | Shionogi & Co., Ltd. | Cephem compound having pseudo-catechol group |
EP2557082A4 (fr) | 2010-04-05 | 2013-08-28 | Shionogi & Co | Composé de céphème comprenant un groupe catéchol |
JP5852562B2 (ja) * | 2010-04-28 | 2016-02-03 | 塩野義製薬株式会社 | 新規なセフェム誘導体 |
US9334289B2 (en) | 2011-04-28 | 2016-05-10 | Shionogi & Co., Ltd. | Cephem compound having catechol or pseudo-catechol structure |
EP2705044A1 (fr) | 2011-05-02 | 2014-03-12 | Zoetis Llc | Nouvelles céphalosporines utiles en tant qu'agents antibactériens |
US9242999B2 (en) | 2011-06-27 | 2016-01-26 | Shionogi & Co., Ltd. | Cephem compound having pyridinium group |
JPWO2013051597A1 (ja) | 2011-10-04 | 2015-03-30 | 塩野義製薬株式会社 | カテコール基を有するセフェム誘導体 |
UY35103A (es) | 2012-10-29 | 2014-05-30 | Glaxo Group Ltd | Compuestos de cefem 2-sustituidos |
WO2014069649A1 (fr) | 2012-10-29 | 2014-05-08 | Shionogi & Co., Ltd. | Procédés de production d'intermédiaires de composés de type 2-alkylcephem |
BR112022004107A2 (pt) | 2019-09-06 | 2022-05-31 | Nabriva Therapeutics GmbH | Conjugados de cefalosporina de sideróforo e seus usos |
KR20220130725A (ko) | 2020-01-22 | 2022-09-27 | 상하이 센후이 메디슨 컴퍼니 리미티드 | 세팔로스포린 항균 화합물 및 이의 약제학적 적용 |
US20240132518A1 (en) | 2021-01-12 | 2024-04-25 | Shanghai Senhui Medicine Co., Ltd. | Cephalosporin antibacterial compound and preparation method therefor |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5285187A (en) * | 1976-01-08 | 1977-07-15 | Shionogi & Co Ltd | Antibacterials against pseudomonas aeruginosa |
US4525473A (en) * | 1983-03-30 | 1985-06-25 | Bristol-Myers Company | Cephalosporins |
KR920004820B1 (ko) * | 1984-02-23 | 1992-06-18 | 메이지제과 주식회사 | 새로운 세팔로스포린 유도체의 제조방법 |
JPS6117589A (ja) * | 1984-07-03 | 1986-01-25 | Meiji Seika Kaisha Ltd | 新規セフアロスポリン誘導体及びその製造法 |
US4880795A (en) * | 1984-05-22 | 1989-11-14 | Bayer Aktiengesellschaft | Cephalosporins |
IL77458A (en) * | 1985-01-14 | 1990-07-26 | Eisai Co Ltd | Cephem derivatives,their production and antibacterial compositions containing them and certain novel intermediates therefor |
ZA86405B (en) * | 1985-01-31 | 1986-09-24 | Yamanouchi Pharma Co Ltd | Cephalosporin compounds and slats thereof,and their production |
DE3506159A1 (de) * | 1985-02-22 | 1986-08-28 | Bayer Ag, 5090 Leverkusen | Neue cephalosporine, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
JPS6230786A (ja) * | 1985-04-11 | 1987-02-09 | Eisai Co Ltd | 3−(キヌクリジニオ)メチル−3−セフエム誘導体 |
JPS625961A (ja) * | 1985-07-01 | 1987-01-12 | Meiji Seika Kaisha Ltd | 酸性基を有するピリドチオン類化合物および該化合物より誘導される新規なセフアロスポリン誘導体 |
DE3541095A1 (de) * | 1985-11-21 | 1987-05-27 | Bayer Ag | Neue cephalosporine, verfahren zu deren herstellung sowie ihre verwendung als arzneimittel |
JPS62209082A (ja) * | 1986-03-11 | 1987-09-14 | Banyu Pharmaceut Co Ltd | セフアロスポリン誘導体 |
US4814328A (en) * | 1986-03-19 | 1989-03-21 | Banyu Pharmaceutical Co., Ltd. | Cephalosporin derivatives, and antibacterial agents |
CA1296012C (fr) * | 1986-03-19 | 1992-02-18 | Susumu Nakagawa | Derives de 6,7-dihydroxy-isoquinaline |
US4782155A (en) * | 1986-03-19 | 1988-11-01 | Banyu Pharmaceutical Co., Ltd. | Cephalosporin derivatives, processes for their preparation and antibacterial agents |
EP0272827A3 (fr) * | 1986-12-23 | 1990-02-07 | ZENECA Pharma S.A. | 3-Hétérocycliquethiométhyl céphalosporines |
DE3711343A1 (de) * | 1987-04-03 | 1988-10-20 | Bayer Ag | Cephalosporinderivate, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
PH25965A (en) * | 1988-06-06 | 1992-01-13 | Fujisawa Pharmaceutical Co | New cephem compounds which have antimicrobial activities |
-
1990
- 1990-08-23 US US07/571,411 patent/US5143910A/en not_active Expired - Fee Related
- 1990-08-26 EP EP90116330A patent/EP0416410B1/fr not_active Expired - Lifetime
- 1990-08-26 DE DE69014490T patent/DE69014490T2/de not_active Expired - Fee Related
- 1990-08-26 DK DK90116330.3T patent/DK0416410T3/da active
- 1990-08-26 AT AT90116330T patent/ATE114658T1/de not_active IP Right Cessation
- 1990-09-06 JP JP2237983A patent/JP2969283B2/ja not_active Expired - Fee Related
- 1990-09-07 KR KR1019900014162A patent/KR0158452B1/ko not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
KR910006303A (ko) | 1991-04-29 |
EP0416410A1 (fr) | 1991-03-13 |
ATE114658T1 (de) | 1994-12-15 |
KR0158452B1 (ko) | 1998-12-01 |
DE69014490D1 (de) | 1995-01-12 |
DE69014490T2 (de) | 1995-04-20 |
JP2969283B2 (ja) | 1999-11-02 |
JPH03173893A (ja) | 1991-07-29 |
EP0416410B1 (fr) | 1994-11-30 |
US5143910A (en) | 1992-09-01 |
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