DE60305053T2 - Pyrimidinderivate als selektive cox-2-inhibitoren - Google Patents

Pyrimidinderivate als selektive cox-2-inhibitoren Download PDF

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Publication number
DE60305053T2
DE60305053T2 DE60305053T DE60305053T DE60305053T2 DE 60305053 T2 DE60305053 T2 DE 60305053T2 DE 60305053 T DE60305053 T DE 60305053T DE 60305053 T DE60305053 T DE 60305053T DE 60305053 T2 DE60305053 T2 DE 60305053T2
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DE60305053D1 (de
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Gordon Stevenage WEINGARTEN
Gianpaolo GlaxoSmithKline Harlow BRAVI
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Glaxo Group Ltd
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Glaxo Group Ltd
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Priority claimed from GB0219304A external-priority patent/GB0219304D0/en
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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DE60305053T 2002-08-19 2003-08-15 Pyrimidinderivate als selektive cox-2-inhibitoren Expired - Fee Related DE60305053T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0219305A GB0219305D0 (en) 2002-08-19 2002-08-19 Pyrimidine derivatives
GB0219305 2002-08-19
GB0219304A GB0219304D0 (en) 2002-08-19 2002-08-19 Pyrimidine derivatives
GB0219304 2002-08-19
PCT/EP2003/009153 WO2004018452A1 (en) 2002-08-19 2003-08-15 Pyrimidine derivatives as selective cox-2 inhibitors

Publications (2)

Publication Number Publication Date
DE60305053D1 DE60305053D1 (de) 2006-06-08
DE60305053T2 true DE60305053T2 (de) 2006-08-31

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DE60305053T Expired - Fee Related DE60305053T2 (de) 2002-08-19 2003-08-15 Pyrimidinderivate als selektive cox-2-inhibitoren

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US (1) US7235560B2 (https=)
EP (1) EP1546128B1 (https=)
JP (1) JP2006500372A (https=)
AT (1) ATE325115T1 (https=)
AU (1) AU2003258630A1 (https=)
DE (1) DE60305053T2 (https=)
ES (1) ES2263058T3 (https=)
WO (1) WO2004018452A1 (https=)

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Publication number Priority date Publication date Assignee Title
ATE325115T1 (de) 2002-08-19 2006-06-15 Glaxo Group Ltd Pyrimidinderivate als selektive cox-2-inhibitoren
GB0221443D0 (en) 2002-09-16 2002-10-23 Glaxo Group Ltd Pyridine derivates
PL2316430T3 (pl) 2004-10-08 2012-11-30 Forward Pharma As Kompozycje farmaceutyczne o kontrolowanym uwalnianiu, zawierające ester kwasu fumarowego
US7759350B2 (en) * 2005-09-15 2010-07-20 Orchid Research Laboratories Ltd. Pyrimidine carboxamides
EP1940382A2 (en) * 2005-10-07 2008-07-09 Aditech Pharma AB Combination therapy with fumaric acid esters for the treatment of autoimmune and/or inflammatory disorders
CN102369001A (zh) 2009-01-09 2012-03-07 前进制药公司 包含溶蚀骨架中的一种或多种富马酸酯的药物制剂
JP2013522240A (ja) * 2010-03-17 2013-06-13 グラクソ グループ リミテッド スフィンゴシン１−リン酸１（ｓ１ｐ１）受容体作用薬として用いるためのピリミジン誘導体
CA3026149A1 (en) * 2016-06-02 2017-12-07 Cadent Therapeutics, Inc. Potassium channel modulators
SI3571193T1 (sl) 2017-01-23 2022-04-29 Cadent Therapeutics, Inc. Modulatorji kalijevega kanalčka
CA3116339A1 (en) 2018-10-22 2020-04-30 Cadent Therapeutics, Inc. Crystalline forms of potassium channel modulators
WO2021050700A1 (en) * 2019-09-13 2021-03-18 The Broad Institute, Inc. Cyclooxygenase-2 inhibitors and uses thereof

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ATE325115T1 (de) 2006-06-15
EP1546128B1 (en) 2006-05-03
ES2263058T3 (es) 2006-12-01
AU2003258630A1 (en) 2004-03-11
US7235560B2 (en) 2007-06-26
DE60305053D1 (de) 2006-06-08
EP1546128A1 (en) 2005-06-29
US20060040967A1 (en) 2006-02-23

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