DE60219068T2 - Substituierte 2-amino-cykloalkankarboxamide und ihre verwendung als cysteinprotease-inhibitoren - Google Patents

Substituierte 2-amino-cykloalkankarboxamide und ihre verwendung als cysteinprotease-inhibitoren Download PDF

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DE60219068T2
DE60219068T2 DE60219068T DE60219068T DE60219068T2 DE 60219068 T2 DE60219068 T2 DE 60219068T2 DE 60219068 T DE60219068 T DE 60219068T DE 60219068 T DE60219068 T DE 60219068T DE 60219068 T2 DE60219068 T2 DE 60219068T2
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amino
cyclohexyl
methyl
indole
carbonyl
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DE60219068D1 (de
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Tobias San Francisco GABRIEL
Nancy Elisabeth Sunnyvale KRAUSS
Taraneh Los Altos MIRZADEGAN
Wylie Solang Mountain View PALMER
David Bernard San Mateo SMITH
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F Hoffmann La Roche AG
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DE60219068T 2001-12-04 2002-11-25 Substituierte 2-amino-cykloalkankarboxamide und ihre verwendung als cysteinprotease-inhibitoren Expired - Fee Related DE60219068T2 (de)

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Application Number Priority Date Filing Date Title
US33675001P 2001-12-04 2001-12-04
US336750P 2001-12-04
PCT/EP2002/013221 WO2003048123A1 (en) 2001-12-04 2002-11-25 Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors

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DE60219068D1 DE60219068D1 (de) 2007-05-03
DE60219068T2 true DE60219068T2 (de) 2007-12-13

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US (1) US6747053B2 (https=)
EP (1) EP1453801B1 (https=)
JP (1) JP2005517640A (https=)
KR (1) KR20050044660A (https=)
CN (1) CN1315806C (https=)
AR (1) AR037683A1 (https=)
AT (1) ATE357432T1 (https=)
AU (1) AU2002352126A1 (https=)
BR (1) BR0214642A (https=)
CA (1) CA2467435A1 (https=)
DE (1) DE60219068T2 (https=)
ES (1) ES2282497T3 (https=)
GT (1) GT200200253A (https=)
HU (1) HUP0402344A2 (https=)
IL (1) IL161992A0 (https=)
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PA (1) PA8559701A1 (https=)
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JP4865129B2 (ja) * 1999-01-13 2012-02-01 ザ・リサーチ・ファウンデーション・オブ・ステイト・ユニバーシティ・オブ・ニューヨーク タンパク質キナーゼ阻害剤を設計するための新規の方法
US7005445B2 (en) * 2001-10-22 2006-02-28 The Research Foundation Of State University Of New York Protein kinase and phosphatase inhibitors and methods for designing them
GB0128996D0 (en) 2001-12-04 2002-01-23 Novartis Ag Organic compounds
AU2003235741B8 (en) * 2002-01-07 2009-01-15 Eisai R&D Management Co., Ltd. Deazapurines and uses thereof
SE0203712D0 (sv) 2002-12-13 2002-12-13 Astrazeneca Ab Novel compounds
GB0403038D0 (en) * 2004-02-11 2004-03-17 Novartis Ag Organic compounds
WO2006007664A1 (en) * 2004-07-22 2006-01-26 Genomics Research Partners Pty Ltd Agents and methods for diagnosing osteoarthritis
JP2008546840A (ja) * 2005-06-28 2008-12-25 メルク エンド カムパニー インコーポレーテッド 非ヌクレオシド逆転写酵素阻害剤
EP1749822B1 (en) * 2005-08-05 2008-10-15 Hybrigenics S.A. Novel cysteine protease inhibitors and their therapeutic applications
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