DE602004008105D1 - 42-o-alkoxyalkylrapamycinderivate und diese enthaltende zusammensetzungen - Google Patents

42-o-alkoxyalkylrapamycinderivate und diese enthaltende zusammensetzungen

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Publication number
DE602004008105D1
DE602004008105D1 DE602004008105T DE602004008105T DE602004008105D1 DE 602004008105 D1 DE602004008105 D1 DE 602004008105D1 DE 602004008105 T DE602004008105 T DE 602004008105T DE 602004008105 T DE602004008105 T DE 602004008105T DE 602004008105 D1 DE602004008105 D1 DE 602004008105D1
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Prior art keywords
derivatives
alkoxyalkylrapamycin
compositions containing
alkoxyalkyl
rapamycin
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DE602004008105T
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DE602004008105T2 (de
Inventor
Ronald E Betts
Douglas R Savage
John E Shulze
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Biosensors International Group Ltd
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Sun Biomedical Ltd
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Materials For Medical Uses (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
DE602004008105T 2003-11-12 2004-11-12 42-o-alkoxyalkylrapamycinderivate und diese enthaltende zusammensetzungen Active DE602004008105T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US706055 1985-02-26
US10/706,055 US7220755B2 (en) 2003-11-12 2003-11-12 42-O-alkoxyalkyl rapamycin derivatives and compositions comprising same
PCT/US2004/037701 WO2005047295A1 (en) 2003-11-12 2004-11-12 42-o-alkoxyalkyl rapamycin derivatives and compositions comprising same

Publications (2)

Publication Number Publication Date
DE602004008105D1 true DE602004008105D1 (de) 2007-09-20
DE602004008105T2 DE602004008105T2 (de) 2008-04-30

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Country Status (7)

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US (2) US7220755B2 (de)
EP (2) EP1689754B1 (de)
AT (1) ATE369372T1 (de)
DE (1) DE602004008105T2 (de)
ES (1) ES2516692T3 (de)
HK (1) HK1097828A1 (de)
WO (1) WO2005047295A1 (de)

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ES2516692T3 (es) 2014-10-31
EP1852437B1 (de) 2014-09-17
EP1689754B1 (de) 2007-08-08
US20050131008A1 (en) 2005-06-16
DE602004008105T2 (de) 2008-04-30
US20050101624A1 (en) 2005-05-12
EP1852437A2 (de) 2007-11-07
ATE369372T1 (de) 2007-08-15
WO2005047295A1 (en) 2005-05-26
US7220755B2 (en) 2007-05-22
EP1852437A3 (de) 2008-03-12
EP1689754A1 (de) 2006-08-16
HK1097828A1 (en) 2007-07-06

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