DE2742903A1 - Herstellung von direkt iodierten steroidhormonen und verwandten verbindungen - Google Patents
Herstellung von direkt iodierten steroidhormonen und verwandten verbindungenInfo
- Publication number
- DE2742903A1 DE2742903A1 DE19772742903 DE2742903A DE2742903A1 DE 2742903 A1 DE2742903 A1 DE 2742903A1 DE 19772742903 DE19772742903 DE 19772742903 DE 2742903 A DE2742903 A DE 2742903A DE 2742903 A1 DE2742903 A1 DE 2742903A1
- Authority
- DE
- Germany
- Prior art keywords
- radioactive
- steroid
- iodine
- estradiol
- agent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
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- 230000002285 radioactive effect Effects 0.000 claims description 30
- 239000003270 steroid hormone Substances 0.000 claims description 30
- 229960005309 estradiol Drugs 0.000 claims description 21
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0493—Steroids, e.g. cholesterol, testosterone
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/74—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving hormones or other non-cytokine intercellular protein regulatory factors such as growth factors, including receptors to hormones and growth factors
- G01N33/743—Steroid hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2123/00—Preparations for testing in vivo
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Physics & Mathematics (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Medicinal Chemistry (AREA)
- Urology & Nephrology (AREA)
- Cell Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Microbiology (AREA)
- Biotechnology (AREA)
- Analytical Chemistry (AREA)
- Biochemistry (AREA)
- Endocrinology (AREA)
- General Physics & Mathematics (AREA)
- Pathology (AREA)
- Food Science & Technology (AREA)
- Optics & Photonics (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/727,284 US4321208A (en) | 1976-09-27 | 1976-09-27 | Preparation of directly iodinated steroid hormones and related compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE2742903A1 true DE2742903A1 (de) | 1978-03-30 |
Family
ID=24922054
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE19772742903 Withdrawn DE2742903A1 (de) | 1976-09-27 | 1977-09-23 | Herstellung von direkt iodierten steroidhormonen und verwandten verbindungen |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US4321208A (enExample) |
| JP (1) | JPS53127453A (enExample) |
| CA (1) | CA1102305A (enExample) |
| DE (1) | DE2742903A1 (enExample) |
| FR (1) | FR2365587A1 (enExample) |
| GB (1) | GB1591357A (enExample) |
| IN (1) | IN146286B (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4450149A (en) * | 1981-06-15 | 1984-05-22 | Research Corporation | Radiohalogenation method |
| DE3337179A1 (de) * | 1983-10-10 | 1985-05-23 | Schering AG, 1000 Berlin und 4709 Bergkamen | Estran- und androstan-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende praeparate |
| US4780420A (en) * | 1985-09-30 | 1988-10-25 | Yale University | Progesterone receptor ligands |
| IT1296576B1 (it) * | 1997-11-27 | 1999-07-14 | Promau Srl | Apparecchiatura automatica per la curvatura di lamiere, con controllo selettivo digitale |
| US7238338B1 (en) * | 2001-06-22 | 2007-07-03 | Triumf | System and method for the large scale labeling of compounds with radiohalogens |
| DE10141937A1 (de) * | 2001-08-28 | 2003-03-27 | Alfred Schmidt | Markierung der Aromatase |
| US8173983B1 (en) | 2010-01-07 | 2012-05-08 | Velayudhan Sahadevan | All field simultaneous radiation therapy |
| BRPI1101556A2 (pt) * | 2011-04-19 | 2015-07-14 | Univ Fed De Pernambuco Ufpe | Composto antitumoral testosterona - ( iodo radioativo) |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3953431A (en) * | 1971-05-24 | 1976-04-27 | Becton, Dickinson & Company | Derivatives of digoxigenin |
| GB1441253A (en) * | 1972-06-22 | 1976-06-30 | Wellcome Found | Reagents for the assay of cardiac glycosides |
| GB1441101A (en) * | 1972-06-22 | 1976-06-30 | Wellcome Found | Reagents for the assay of cardenolide glycosides and aglycones |
| DE2260933C3 (de) * | 1972-12-08 | 1981-08-20 | Schering Ag Berlin Und Bergkamen, 1000 Berlin | Verfahren zur Herstellung von durch radioaktives Halogen markierten organischen Verbindungen |
| US4013688A (en) * | 1972-12-20 | 1977-03-22 | The Upjohn Company | Radioimmunoassay agents |
-
1976
- 1976-09-27 US US05/727,284 patent/US4321208A/en not_active Expired - Lifetime
-
1977
- 1977-09-13 CA CA286,659A patent/CA1102305A/en not_active Expired
- 1977-09-19 GB GB39175/77A patent/GB1591357A/en not_active Expired
- 1977-09-23 DE DE19772742903 patent/DE2742903A1/de not_active Withdrawn
- 1977-09-26 FR FR7728950A patent/FR2365587A1/fr active Granted
- 1977-09-27 JP JP11525377A patent/JPS53127453A/ja active Pending
- 1977-09-27 IN IN1453/CAL/77A patent/IN146286B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB1591357A (en) | 1981-06-17 |
| US4321208A (en) | 1982-03-23 |
| JPS53127453A (en) | 1978-11-07 |
| FR2365587A1 (fr) | 1978-04-21 |
| IN146286B (enExample) | 1979-04-14 |
| FR2365587B3 (enExample) | 1980-07-11 |
| CA1102305A (en) | 1981-06-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| OD | Request for examination | ||
| 8139 | Disposal/non-payment of the annual fee |