DE2155081C3 - - Google Patents

Info

Publication number
DE2155081C3
DE2155081C3 DE2155081A DE2155081A DE2155081C3 DE 2155081 C3 DE2155081 C3 DE 2155081C3 DE 2155081 A DE2155081 A DE 2155081A DE 2155081 A DE2155081 A DE 2155081A DE 2155081 C3 DE2155081 C3 DE 2155081C3
Authority
DE
Germany
Prior art keywords
acid
protons
cps
general formula
acetamido
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE2155081A
Other languages
German (de)
English (en)
Other versions
DE2155081B2 (de
DE2155081A1 (de
Inventor
Auf Nichtnennung Antrag
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
DSM Delft BV
Original Assignee
Koninklijke Nederlandsche Gist en Spiritusfabriek BV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Koninklijke Nederlandsche Gist en Spiritusfabriek BV filed Critical Koninklijke Nederlandsche Gist en Spiritusfabriek BV
Publication of DE2155081A1 publication Critical patent/DE2155081A1/de
Publication of DE2155081B2 publication Critical patent/DE2155081B2/de
Application granted granted Critical
Publication of DE2155081C3 publication Critical patent/DE2155081C3/de
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE2155081A 1970-11-06 1971-11-05 7- (lsoxazol-5-yl-acetamido)cephalosporansäurederivate, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammensetzungen Granted DE2155081B2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB5304070A GB1364453A (en) 1970-11-06 1970-11-06 Penicillanic and cepholosporanic acid derivatives

Publications (3)

Publication Number Publication Date
DE2155081A1 DE2155081A1 (de) 1972-05-10
DE2155081B2 DE2155081B2 (de) 1975-05-15
DE2155081C3 true DE2155081C3 (he) 1975-12-18

Family

ID=10466394

Family Applications (3)

Application Number Title Priority Date Filing Date
DE19712166468 Pending DE2166468A1 (de) 1970-11-06 1971-11-05 Neue isoxazolylderivate und verfahren zu deren herstellung
DE2155081A Granted DE2155081B2 (de) 1970-11-06 1971-11-05 7- (lsoxazol-5-yl-acetamido)cephalosporansäurederivate, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammensetzungen
DE19712166467 Pending DE2166467A1 (de) 1970-11-06 1971-11-05 Neue penicillansaeurederivate, deren herstellungsverfahren und diese enthaltende pharmazeutische zusammensetzungen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE19712166468 Pending DE2166468A1 (de) 1970-11-06 1971-11-05 Neue isoxazolylderivate und verfahren zu deren herstellung

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE19712166467 Pending DE2166467A1 (de) 1970-11-06 1971-11-05 Neue penicillansaeurederivate, deren herstellungsverfahren und diese enthaltende pharmazeutische zusammensetzungen

Country Status (14)

Country Link
US (1) US3891635A (he)
JP (1) JPS5212200B1 (he)
AU (1) AU463230B2 (he)
BE (1) BE775012A (he)
CA (1) CA983920A (he)
CH (3) CH573436A5 (he)
DE (3) DE2166468A1 (he)
ES (2) ES396720A1 (he)
FR (1) FR2112504B1 (he)
GB (1) GB1364453A (he)
HU (1) HU162822B (he)
NL (1) NL150117B (he)
SU (1) SU520050A3 (he)
ZA (1) ZA717433B (he)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1459392A (en) * 1972-12-22 1976-12-22 Gist Brocades Nv Heterocyclic compounds
FR2219775A1 (en) * 1973-03-02 1974-09-27 Gist Brocades Nv Isoxazolylacetamido penicillanic and cephalosporanic acids - partic. active against Gram-positive bacteria
JPS5760345B2 (he) * 1974-12-19 1982-12-18 Takeda Chemical Industries Ltd
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
CA1088049A (en) * 1975-06-03 1980-10-21 Takashi Masugi 3-substituted-7-substituted alkanamido-3-cephem-4- carboxylic acid compounds and processes for preparation thereof
MD227C2 (ro) * 1976-01-23 1995-11-30 Roussel Uclaf, Societe Anonyme Procedeu de obţinere a derivaţilor acidului 7-(2-(2-aminotiazolil-4)-2-oxiiminoacetamido)-3-acetoximetil-3-cefem- 4-carbonic sub formă de sin-izomeri
JPS6052713B2 (ja) * 1978-04-11 1985-11-20 三共株式会社 ７−メトキシセフアロスポリン化合物、その製法及びその化合物を主成分とする抗菌剤
CA1128526A (en) * 1979-10-05 1982-07-27 Cdc Life Sciences Inc. 3,4-diarylisoxazol-5-acetic acids
US4526977A (en) * 1981-10-07 1985-07-02 American Home Products Corporation 2-(3-Amino-5-isoxazolyl)-2-oxyimino-acetic acids
JPS60141367U (ja) * 1984-02-29 1985-09-19 タキロン株式会社 天窓のロツク装置
US4562187A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (Isoxazol-3-yl)arylmethanones, compositions and pharmaceutical use
US7427680B2 (en) * 2001-01-12 2008-09-23 The Regents Of The University Of California Fluorogenic substrates for BETA-lactamase gene expression
AU2002251755C1 (en) * 2001-01-12 2008-07-10 The Regents Of The University Of California Beta-lactamase substrates having phenolic ethers

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3218318A (en) * 1962-08-31 1965-11-16 Lilly Co Eli 7-heterocyclic-substituted-acylamido cephalosporins
US3459746A (en) * 1965-10-04 1969-08-05 Lilly Co Eli 7 - heteromonocyclic-substituted acylamido derivatives of desacetyl cephalosporanic acid

Also Published As

Publication number Publication date
DE2166468A1 (de) 1974-02-14
CA983920A (en) 1976-02-17
GB1364453A (en) 1974-08-21
ES423795A1 (es) 1976-12-16
FR2112504B1 (he) 1975-10-31
BE775012A (fr) 1972-05-05
AU463230B2 (en) 1975-07-17
AU3543171A (en) 1973-05-10
US3891635A (en) 1975-06-24
CH573436A5 (he) 1976-03-15
NL7115231A (he) 1972-05-09
ES396720A1 (es) 1975-04-16
SU520050A3 (ru) 1976-06-30
HU162822B (he) 1973-04-28
FR2112504A1 (he) 1972-06-16
DE2155081B2 (de) 1975-05-15
ZA717433B (en) 1972-07-26
CH572935A5 (he) 1976-02-27
DE2155081A1 (de) 1972-05-10
DE2166467A1 (de) 1974-02-14
JPS5212200B1 (he) 1977-04-05
NL150117B (nl) 1976-07-15
CH572936A5 (he) 1976-02-27

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Legal Events

Date Code Title Description
C3 Grant after two publication steps (3rd publication)
E77 Valid patent as to the heymanns-index 1977
EHJ Ceased/non-payment of the annual fee