DD253823A5 - Verfahren zur herstellung neuartiger thienopyridone - Google Patents
Verfahren zur herstellung neuartiger thienopyridone Download PDFInfo
- Publication number
- DD253823A5 DD253823A5 DD86291289A DD29128986A DD253823A5 DD 253823 A5 DD253823 A5 DD 253823A5 DD 86291289 A DD86291289 A DD 86291289A DD 29128986 A DD29128986 A DD 29128986A DD 253823 A5 DD253823 A5 DD 253823A5
- Authority
- DD
- German Democratic Republic
- Prior art keywords
- formula
- compound
- methyl
- mixture
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/36—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB858515207A GB8515207D0 (en) | 1985-06-15 | 1985-06-15 | Therapeutic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DD253823A5 true DD253823A5 (de) | 1988-02-03 |
Family
ID=10580803
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DD86291289A DD253823A5 (de) | 1985-06-15 | 1986-06-13 | Verfahren zur herstellung neuartiger thienopyridone |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US4710506A (da) |
| EP (1) | EP0209977A3 (da) |
| JP (1) | JPS6236382A (da) |
| KR (1) | KR870000339A (da) |
| AU (1) | AU581595B2 (da) |
| CS (1) | CS258483B2 (da) |
| DD (1) | DD253823A5 (da) |
| DK (1) | DK272486A (da) |
| ES (1) | ES8707243A1 (da) |
| FI (1) | FI862520A (da) |
| GB (1) | GB8515207D0 (da) |
| GR (1) | GR861527B (da) |
| HU (1) | HU195661B (da) |
| JO (1) | JO1482B1 (da) |
| NO (1) | NO862373L (da) |
| PH (1) | PH22293A (da) |
| PL (1) | PL266392A1 (da) |
| PT (1) | PT82759B (da) |
| YU (2) | YU99386A (da) |
| ZA (1) | ZA864396B (da) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8627698D0 (en) * | 1986-11-20 | 1986-12-17 | Boots Co Plc | Therapeutic agents |
| US4767766A (en) * | 1987-01-30 | 1988-08-30 | Merck & Co., Inc. | Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors |
| US4904672A (en) * | 1987-01-30 | 1990-02-27 | Merck & Co., Inc. | Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors |
| NZ230711A (en) * | 1988-09-23 | 1990-10-26 | Ortho Pharma Corp | Substituted thienopyrans as antihypertensive agents |
| AU5509099A (en) * | 1998-08-03 | 2000-02-28 | Basf Corporation | Pyridinones for the treatment of sexual dysfunction |
| US6458804B1 (en) * | 2001-01-26 | 2002-10-01 | R.T. Alamo Venturesi, Llc | Methods for the treatment of central nervous system disorders in certain patient groups |
| US6451813B1 (en) | 2001-01-26 | 2002-09-17 | R. T. Alamo Ventures I, Llc | Treatment of gastroparesis in certain patient groups |
| US6562838B2 (en) | 2001-01-26 | 2003-05-13 | R. T. Alamo Ventures I, L.L.C. | Treatment of cardiovascular disease with quinolinone enantiomers |
| US8329924B2 (en) * | 2001-06-11 | 2012-12-11 | Vertex Pharmaceuticals (Canada) Incorporated | Compounds and methods for the treatment or prevention of Flavivirus infections |
| CN101624391A (zh) * | 2001-06-11 | 2010-01-13 | 病毒化学医药公司 | 用作黄病毒感染抗病毒剂的噻吩衍生物 |
| US6995171B2 (en) * | 2001-06-21 | 2006-02-07 | Agouron Pharmaceuticals, Inc. | Bicyclic pyrimidine and pyrimidine derivatives useful as anticancer agents |
| CN100413861C (zh) * | 2002-12-10 | 2008-08-27 | 维勒凯姆制药股份有限公司 | 用于治疗或预防黄病毒感染的化合物 |
| US7994192B2 (en) * | 2006-09-26 | 2011-08-09 | Crestone, Inc. | Substituted thienopyridone compounds with antibacterial activity |
| US8697720B2 (en) | 2006-09-26 | 2014-04-15 | Crestone, Inc. | Substituted phenylether-thienopyridone compounds with antibacterial activity |
| US7973050B2 (en) * | 2006-09-26 | 2011-07-05 | Crestone, Inc. | Enantiomeric compounds with antibacterial activity |
| US8658670B2 (en) * | 2006-09-26 | 2014-02-25 | Crestone, Inc. | Methods and compounds for treatment of clostridium based infection |
| ES2392897T3 (es) * | 2006-09-26 | 2012-12-14 | Crestone, Inc. | Compuestos tienopiridona sustituidos con actividad antibacteriana |
| EP2559692A1 (en) | 2006-11-15 | 2013-02-20 | Virochem Pharma Inc. | Thiophene analogues for the treatment or prevention of Flavivirus infections |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3997545A (en) * | 1973-07-23 | 1976-12-14 | Takeda Chemical Industries, Ltd. | Thienopyridine-carboxylic acid derivatives |
| NZ193167A (en) * | 1979-03-27 | 1984-08-24 | Boots Co Plc | Quinoline derivatives and pharmaceutical compositions |
| JPS5742690A (en) * | 1980-08-28 | 1982-03-10 | Kanebo Ltd | Thieno 3,2-b pyridinecarboxylic acid derivative |
| GB2085441B (en) * | 1980-09-26 | 1984-10-17 | Boots The Co Ltd | Therapeutic agents |
| IE51542B1 (en) * | 1980-09-26 | 1987-01-07 | Boots Co Ltd | Therapeutic agents |
| DE3412947A1 (de) * | 1984-04-06 | 1985-10-17 | Bayer Ag, 5090 Leverkusen | Tetrahydothienopyridine, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
-
1985
- 1985-06-15 GB GB858515207A patent/GB8515207D0/en active Pending
-
1986
- 1986-06-05 AU AU58383/86A patent/AU581595B2/en not_active Expired - Fee Related
- 1986-06-09 PH PH33869A patent/PH22293A/en unknown
- 1986-06-09 EP EP86304382A patent/EP0209977A3/en not_active Withdrawn
- 1986-06-10 DK DK272486A patent/DK272486A/da not_active Application Discontinuation
- 1986-06-10 YU YU00993/86A patent/YU99386A/xx unknown
- 1986-06-12 PT PT82759A patent/PT82759B/pt unknown
- 1986-06-12 FI FI862520A patent/FI862520A/fi not_active Application Discontinuation
- 1986-06-12 ZA ZA864396A patent/ZA864396B/xx unknown
- 1986-06-12 GR GR861527A patent/GR861527B/el unknown
- 1986-06-12 CS CS864362A patent/CS258483B2/cs unknown
- 1986-06-13 US US06/874,337 patent/US4710506A/en not_active Expired - Lifetime
- 1986-06-13 DD DD86291289A patent/DD253823A5/de unknown
- 1986-06-13 ES ES556026A patent/ES8707243A1/es not_active Expired
- 1986-06-13 HU HU862521A patent/HU195661B/hu not_active IP Right Cessation
- 1986-06-13 NO NO862373A patent/NO862373L/no unknown
- 1986-06-14 KR KR1019860004737A patent/KR870000339A/ko not_active Application Discontinuation
- 1986-06-14 JO JO19861482A patent/JO1482B1/en active
- 1986-06-16 PL PL1986266392A patent/PL266392A1/xx unknown
- 1986-06-16 JP JP61139953A patent/JPS6236382A/ja active Pending
-
1987
- 1987-06-29 YU YU01211/87A patent/YU121187A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CS436286A2 (en) | 1987-12-17 |
| DK272486D0 (da) | 1986-06-10 |
| JPS6236382A (ja) | 1987-02-17 |
| EP0209977A2 (en) | 1987-01-28 |
| HUT42775A (en) | 1987-08-28 |
| ES8707243A1 (es) | 1987-07-16 |
| GB8515207D0 (en) | 1985-07-17 |
| CS258483B2 (en) | 1988-08-16 |
| ZA864396B (en) | 1987-08-26 |
| NO862373L (no) | 1986-12-16 |
| FI862520A0 (fi) | 1986-06-12 |
| NO862373D0 (no) | 1986-06-13 |
| EP0209977A3 (en) | 1988-06-08 |
| HU195661B (en) | 1988-06-28 |
| AU581595B2 (en) | 1989-02-23 |
| FI862520A (fi) | 1986-12-16 |
| US4710506A (en) | 1987-12-01 |
| PL266392A1 (en) | 1988-02-18 |
| GR861527B (en) | 1986-10-14 |
| KR870000339A (ko) | 1987-02-17 |
| YU99386A (en) | 1988-04-30 |
| AU5838386A (en) | 1986-12-18 |
| JO1482B1 (en) | 1988-03-10 |
| YU121187A (en) | 1988-04-30 |
| PT82759A (en) | 1986-07-01 |
| PH22293A (en) | 1988-07-22 |
| DK272486A (da) | 1986-12-16 |
| ES556026A0 (es) | 1987-07-16 |
| PT82759B (en) | 1988-05-12 |
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