DD232045A5 - Verfahren zur herstellung von vorwirkstoffen entzuendungshemmender oxicame - Google Patents
Verfahren zur herstellung von vorwirkstoffen entzuendungshemmender oxicame Download PDFInfo
- Publication number
- DD232045A5 DD232045A5 DD85273451A DD27345185A DD232045A5 DD 232045 A5 DD232045 A5 DD 232045A5 DD 85273451 A DD85273451 A DD 85273451A DD 27345185 A DD27345185 A DD 27345185A DD 232045 A5 DD232045 A5 DD 232045A5
- Authority
- DD
- German Democratic Republic
- Prior art keywords
- methyl
- dioxide
- carboxamide
- formula
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US58268484A | 1984-02-23 | 1984-02-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DD232045A5 true DD232045A5 (de) | 1986-01-15 |
Family
ID=24330094
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DD85273451A DD232045A5 (de) | 1984-02-23 | 1985-02-21 | Verfahren zur herstellung von vorwirkstoffen entzuendungshemmender oxicame |
Country Status (22)
| Country | Link |
|---|---|
| JP (1) | JPS60184077A (da) |
| KR (1) | KR850006198A (da) |
| AU (1) | AU552478B2 (da) |
| BE (1) | BE901783A (da) |
| DD (1) | DD232045A5 (da) |
| DE (1) | DE3505576A1 (da) |
| DK (1) | DK81185A (da) |
| ES (1) | ES8606312A1 (da) |
| FI (1) | FI850742L (da) |
| FR (1) | FR2565980A1 (da) |
| GB (1) | GB2154585A (da) |
| GR (1) | GR850442B (da) |
| HU (1) | HUT37616A (da) |
| IL (1) | IL74407A0 (da) |
| IT (1) | IT1185514B (da) |
| LU (1) | LU85780A1 (da) |
| NL (1) | NL8500485A (da) |
| NO (1) | NO850725L (da) |
| PL (1) | PL252023A1 (da) |
| PT (1) | PT79988B (da) |
| SE (1) | SE8500889L (da) |
| ZA (1) | ZA851317B (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4623486A (en) * | 1985-05-29 | 1986-11-18 | Pfizer Inc. | [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity |
| US4610982A (en) * | 1985-06-03 | 1986-09-09 | Pfizer Inc. | Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor |
| US20090238763A1 (en) | 2006-07-09 | 2009-09-24 | Chongxi Yu | High penetration compositions and uses thereof |
| US20090221703A1 (en) | 2006-07-09 | 2009-09-03 | Chongxi Yu | High penetration composition and uses thereof |
| JP5378221B2 (ja) * | 2006-10-11 | 2013-12-25 | テックフィールズ バイオケム カンパニー リミテッド | 非常に高い皮膚浸透率を有するオキシカム及び関連化合物の正荷電水溶性プロドラッグ |
| KR101853971B1 (ko) | 2007-06-04 | 2018-05-02 | 테크필즈 인크 | 매우 높은 피부 및 막 침투율을 가지는 비스테로이드성 소염제(ｎｓａｉａ) 약물전구체 및 이들의 새로운 의약적 용도 |
| RU2765463C2 (ru) | 2008-12-04 | 2022-01-31 | Чунси ЮЙ | Композиции интенсивного проникновения и их применение |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3591574A (en) * | 1968-05-29 | 1971-07-06 | American Home Prod | Tri-n-phenylglycyl derivatives of insulin |
| US3787324A (en) * | 1971-03-01 | 1974-01-22 | Warner Lambert Co | 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production |
| US3704298A (en) * | 1971-06-22 | 1972-11-28 | Warner Lambert Co | 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides |
| AU518216B2 (en) * | 1977-09-06 | 1981-09-17 | Hafslund Nycomed Pharma Aktiengesellschaft | Thienothiazine derivatives |
| JPS5714589A (en) * | 1980-06-27 | 1982-01-25 | Mitsui Toatsu Chem Inc | Benzothiazine derivative, its preparation and drug composition |
| US4309427A (en) * | 1981-01-15 | 1982-01-05 | Pfizer Inc. | Benzothiazine dioxide derivatives |
| IT8219486A0 (it) * | 1982-02-05 | 1982-02-05 | Chiesi Farma Spa | Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche. |
| IT1206525B (it) * | 1982-12-10 | 1989-04-27 | Zionale S R L A Roma | Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione |
-
1985
- 1985-01-23 JP JP60010722A patent/JPS60184077A/ja active Pending
- 1985-02-18 DE DE19853505576 patent/DE3505576A1/de not_active Ceased
- 1985-02-19 PL PL25202385A patent/PL252023A1/xx unknown
- 1985-02-20 GB GB08504355A patent/GB2154585A/en not_active Withdrawn
- 1985-02-20 PT PT79988A patent/PT79988B/pt unknown
- 1985-02-20 GR GR850442A patent/GR850442B/el unknown
- 1985-02-20 LU LU85780A patent/LU85780A1/fr unknown
- 1985-02-21 IT IT8519585A patent/IT1185514B/it active
- 1985-02-21 NL NL8500485A patent/NL8500485A/nl not_active Application Discontinuation
- 1985-02-21 ZA ZA851317A patent/ZA851317B/xx unknown
- 1985-02-21 ES ES540590A patent/ES8606312A1/es not_active Expired
- 1985-02-21 BE BE0/214544A patent/BE901783A/fr not_active IP Right Cessation
- 1985-02-21 DD DD85273451A patent/DD232045A5/de unknown
- 1985-02-21 IL IL74407A patent/IL74407A0/xx unknown
- 1985-02-22 DK DK81185A patent/DK81185A/da not_active Application Discontinuation
- 1985-02-22 SE SE8500889A patent/SE8500889L/xx not_active Application Discontinuation
- 1985-02-22 FR FR8502586A patent/FR2565980A1/fr active Pending
- 1985-02-22 KR KR1019850001106A patent/KR850006198A/ko not_active Application Discontinuation
- 1985-02-22 NO NO850725A patent/NO850725L/no unknown
- 1985-02-22 HU HU85678A patent/HUT37616A/hu unknown
- 1985-02-22 FI FI850742A patent/FI850742L/fi not_active Application Discontinuation
- 1985-02-22 AU AU39066/85A patent/AU552478B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| NL8500485A (nl) | 1985-09-16 |
| GR850442B (da) | 1985-06-19 |
| PT79988A (en) | 1985-03-01 |
| FI850742A0 (fi) | 1985-02-22 |
| AU3906685A (en) | 1985-09-05 |
| GB2154585A (en) | 1985-09-11 |
| DK81185D0 (da) | 1985-02-22 |
| JPS60184077A (ja) | 1985-09-19 |
| IL74407A0 (en) | 1985-05-31 |
| HUT37616A (en) | 1986-01-23 |
| KR850006198A (ko) | 1985-10-02 |
| BE901783A (fr) | 1985-08-21 |
| PL252023A1 (en) | 1985-11-05 |
| PT79988B (en) | 1987-02-02 |
| GB8504355D0 (en) | 1985-03-20 |
| NO850725L (no) | 1985-08-26 |
| DK81185A (da) | 1985-09-10 |
| SE8500889L (sv) | 1985-08-24 |
| FI850742L (fi) | 1985-08-24 |
| LU85780A1 (fr) | 1985-12-11 |
| IT8519585A0 (it) | 1985-02-21 |
| AU552478B2 (en) | 1986-06-05 |
| IT1185514B (it) | 1987-11-12 |
| ES8606312A1 (es) | 1986-04-16 |
| ES540590A0 (es) | 1986-04-16 |
| FR2565980A1 (fr) | 1985-12-20 |
| ZA851317B (en) | 1986-10-29 |
| DE3505576A1 (de) | 1985-09-05 |
| SE8500889D0 (sv) | 1985-02-22 |
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