CZ302847B6 - Orální dávkovací formy obsahující oxcarbazepin - Google Patents
Orální dávkovací formy obsahující oxcarbazepin Download PDFInfo
- Publication number
- CZ302847B6 CZ302847B6 CZ20021529A CZ20021529A CZ302847B6 CZ 302847 B6 CZ302847 B6 CZ 302847B6 CZ 20021529 A CZ20021529 A CZ 20021529A CZ 20021529 A CZ20021529 A CZ 20021529A CZ 302847 B6 CZ302847 B6 CZ 302847B6
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- CZ
- Czechia
- Prior art keywords
- oxcarbazepine
- oral dosage
- use according
- medicament
- dosage form
- Prior art date
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- 229950005425 sodium myristyl sulfate Drugs 0.000 description 1
- 229910052938 sodium sulfate Inorganic materials 0.000 description 1
- 235000011152 sodium sulphate Nutrition 0.000 description 1
- 238000007711 solidification Methods 0.000 description 1
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- 239000000600 sorbitol Substances 0.000 description 1
- 239000007921 spray Substances 0.000 description 1
- 239000008107 starch Substances 0.000 description 1
- 238000010972 statistical evaluation Methods 0.000 description 1
- 208000005809 status epilepticus Diseases 0.000 description 1
- 230000000638 stimulation Effects 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 235000000346 sugar Nutrition 0.000 description 1
- 150000005846 sugar alcohols Chemical class 0.000 description 1
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- 239000004094 surface-active agent Substances 0.000 description 1
- 239000007916 tablet composition Substances 0.000 description 1
- 238000010998 test method Methods 0.000 description 1
- MYOWBHNETUSQPA-UHFFFAOYSA-N tetradecane-1-sulfonic acid Chemical compound CCCCCCCCCCCCCCS(O)(=O)=O MYOWBHNETUSQPA-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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| IL (3) | IL149147A0 (enExample) |
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| US20020022056A1 (en) | 1997-02-14 | 2002-02-21 | Burkhard Schlutermann | Oxacarbazepine film-coated tablets |
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| GB0221956D0 (en) * | 2002-09-20 | 2002-10-30 | Novartis Ag | Organic compounds |
| BRPI0414112A (pt) * | 2003-09-03 | 2006-10-31 | Novartis Ag | uso de oxcarbazepina para o tratamento de dor neuropática diabética e a melhora do sono |
| AR048672A1 (es) * | 2004-03-22 | 2006-05-17 | Novartis Ag | Tabletas de desintegracion que comprenden licarbazepina |
| BRPI0509861A (pt) * | 2004-04-13 | 2007-10-16 | Boehringer Ingelheim Int | uso de simeticona em pacientes constipados |
| WO2006046105A1 (en) * | 2004-10-25 | 2006-05-04 | Ranbaxy Laboratories Limited | Oxcarbazepine dosage forms |
| US20060252745A1 (en) | 2005-05-06 | 2006-11-09 | Almeida Jose L D | Methods of preparing pharmaceutical compositions comprising eslicarbazepine acetate and methods of use |
| US20090143360A1 (en) * | 2005-07-08 | 2009-06-04 | Muhammed Safadi | Oxcarbazepine Formulation |
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| US20070178164A1 (en) * | 2006-01-31 | 2007-08-02 | Sigal Blau | Pharmaceutical formulations of oxcarbazepine and methods for its preparation |
| CN101489560B (zh) * | 2006-04-26 | 2015-11-25 | 苏佩努斯制药公司 | 具有s形释放曲线的奥卡西平控释制剂 |
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| CH649080A5 (de) * | 1981-04-16 | 1985-04-30 | Ciba Geigy Ag | 5h-dibenz(b,f)azepin-5-carboxamide als mittel zur prophylaxe und behandlung von zerebraler leistungsinsuffizienz. |
| FR2699077B1 (fr) * | 1992-12-16 | 1995-01-13 | Rhone Poulenc Rorer Sa | Application d'anticonvulsivants dans le traitement de lésions neurologiques liées à des traumatismes. |
| FR2702148B1 (fr) * | 1993-03-05 | 1995-04-07 | Rhone Poulenc Rorer Sa | Application d'anticonvulsivants dans le traitement du neuro-sida. |
| ZA953078B (en) * | 1994-04-28 | 1996-01-05 | Alza Corp | Effective therapy for epilepsies |
| US20020022056A1 (en) * | 1997-02-14 | 2002-02-21 | Burkhard Schlutermann | Oxacarbazepine film-coated tablets |
-
1999
- 1999-11-02 GB GBGB9925962.4A patent/GB9925962D0/en not_active Ceased
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2000
- 2000-10-31 TR TR2002/00951T patent/TR200200951T2/xx unknown
- 2000-10-31 CN CN00814884A patent/CN1407894A/zh active Pending
- 2000-10-31 SK SK584-2002A patent/SK287479B6/sk not_active IP Right Cessation
- 2000-10-31 MX MXPA02004389A patent/MXPA02004389A/es unknown
- 2000-10-31 EP EP00983101A patent/EP1242091B1/en not_active Expired - Lifetime
- 2000-10-31 DE DE60039629T patent/DE60039629D1/de not_active Expired - Lifetime
- 2000-10-31 RU RU2002113752/15A patent/RU2330666C2/ru not_active IP Right Cessation
- 2000-10-31 HU HU0203556A patent/HU227685B1/hu not_active IP Right Cessation
- 2000-10-31 PL PL366314A patent/PL200273B1/pl unknown
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- 2000-10-31 WO PCT/EP2000/010764 patent/WO2001032183A2/en not_active Ceased
- 2000-10-31 JP JP2001534388A patent/JP2003514780A/ja not_active Withdrawn
- 2000-10-31 AT AT00983101T patent/ATE401892T1/de active
- 2000-10-31 BR BR0015188-2A patent/BR0015188A/pt not_active IP Right Cessation
- 2000-10-31 IL IL14914700A patent/IL149147A0/xx unknown
- 2000-10-31 KR KR10-2002-7005613A patent/KR100493836B1/ko not_active Expired - Fee Related
- 2000-10-31 CZ CZ20021529A patent/CZ302847B6/cs not_active IP Right Cessation
- 2000-10-31 ES ES00983101T patent/ES2311001T3/es not_active Expired - Lifetime
- 2000-10-31 AU AU19978/01A patent/AU777705B2/en not_active Ceased
- 2000-10-31 NZ NZ518378A patent/NZ518378A/en not_active IP Right Cessation
- 2000-10-31 HK HK03101121.7A patent/HK1050839B/en not_active IP Right Cessation
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2002
- 2002-04-15 IL IL149147A patent/IL149147A/en not_active IP Right Cessation
- 2002-04-29 ZA ZA200203394A patent/ZA200203394B/en unknown
- 2002-04-30 NO NO20022058A patent/NO330947B1/no not_active IP Right Cessation
-
2005
- 2005-10-11 US US11/247,932 patent/US20060079502A1/en not_active Abandoned
-
2006
- 2006-10-18 US US11/582,801 patent/US20070037792A1/en not_active Abandoned
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2007
- 2007-04-18 JP JP2007109439A patent/JP2007224041A/ja active Pending
-
2009
- 2009-03-23 US US12/408,770 patent/US20090252793A1/en not_active Abandoned
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2010
- 2010-05-03 IL IL205504A patent/IL205504A0/en unknown
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2012
- 2012-08-03 JP JP2012172912A patent/JP2012211202A/ja active Pending
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0646374A1 (de) * | 1993-09-08 | 1995-04-05 | Ciba-Geigy Ag | Doppelt beschichtete Oxcarbazepin-Tabletten |
| WO1998035681A1 (en) * | 1997-02-14 | 1998-08-20 | Novartis Ag | Oxacarbazepine film-coated tablets |
Non-Patent Citations (1)
| Title |
|---|
| Trileptal Basic Drug Information, str. 3, Ciba-Geigy, LTD, 24.04.1993 * |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Patent lapsed due to non-payment of fee |
Effective date: 20131031 |