CY1109304T1 - Αμινοξεα με συναφεια για την αλφα-2-δελτα-πρωτεϊνη - Google Patents

Αμινοξεα με συναφεια για την αλφα-2-δελτα-πρωτεϊνη

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Publication number
CY1109304T1
CY1109304T1 CY20091100858T CY091100858T CY1109304T1 CY 1109304 T1 CY1109304 T1 CY 1109304T1 CY 20091100858 T CY20091100858 T CY 20091100858T CY 091100858 T CY091100858 T CY 091100858T CY 1109304 T1 CY1109304 T1 CY 1109304T1
Authority
CY
Cyprus
Prior art keywords
delta
alpha
amino acids
affinity
protein
Prior art date
Application number
CY20091100858T
Other languages
English (en)
Inventor
Nancy Sue Barta
Jacob Bradley Schwarz
Andrew John Thorpe
David Juergen Wustrow
Original Assignee
Warner-Lambert Company Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=28675482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1109304(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner-Lambert Company Llc filed Critical Warner-Lambert Company Llc
Publication of CY1109304T1 publication Critical patent/CY1109304T1/el

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    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
    • C07C229/08—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to hydrogen atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
    • A61K31/198—Alpha-aminoacids, e.g. alanine, edetic acids [EDTA]
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/28—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and containing rings
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    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
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    • C07C2601/00—Systems containing only non-condensed rings
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    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

Η εφεύρεση αυτή αφορά ορισμένα β-αμινοξέα που συνδέονται προς την αλφα-2-δελτα (α2δ) υπομονάδα ενός διαύλου ασβεστίου. Αυτές οι ενώσεις και τα φαρμακευτικώς αποδεκτά άλατα αυτών είναι χρήσιμα στη θεραπεία μια ποικιλίας ψυχιατρικών, πόνου και άλλων διαταραχών.
CY20091100858T 2002-03-28 2009-08-12 Αμινοξεα με συναφεια για την αλφα-2-δελτα-πρωτεϊνη CY1109304T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36841302P 2002-03-28 2002-03-28
EP03706831A EP1492761B1 (en) 2002-03-28 2003-03-17 Amino acids with affinity for the alpha-2-delta-protein

Publications (1)

Publication Number Publication Date
CY1109304T1 true CY1109304T1 (el) 2014-07-02

Family

ID=28675482

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20091100858T CY1109304T1 (el) 2002-03-28 2009-08-12 Αμινοξεα με συναφεια για την αλφα-2-δελτα-πρωτεϊνη

Country Status (43)

Country Link
US (3) US7064147B2 (el)
EP (2) EP1492761B1 (el)
JP (2) JP3831379B2 (el)
KR (2) KR100694719B1 (el)
CN (2) CN100462351C (el)
AP (1) AP1791A (el)
AR (2) AR039154A1 (el)
AU (1) AU2003208538B2 (el)
BR (1) BR0308814A (el)
CA (1) CA2480872C (el)
CR (1) CR7501A (el)
CU (1) CU23331B7 (el)
CY (1) CY1109304T1 (el)
DE (1) DE60328469D1 (el)
DK (1) DK1492761T3 (el)
EA (2) EA008709B1 (el)
EC (1) ECSP045319A (el)
ES (1) ES2327910T3 (el)
GE (2) GEP20084298B (el)
GT (2) GT200300072A (el)
HK (1) HK1076627A1 (el)
HR (2) HRP20040891A2 (el)
IL (2) IL164110A0 (el)
IS (2) IS7451A (el)
MA (1) MA27188A1 (el)
MX (1) MXPA04009373A (el)
MY (1) MY131424A (el)
NI (1) NI200300043A (el)
NO (2) NO20044614L (el)
NZ (2) NZ535364A (el)
OA (1) OA12795A (el)
PA (1) PA8570001A1 (el)
PE (1) PE20040349A1 (el)
PL (1) PL209750B1 (el)
PT (1) PT1492761E (el)
RS (2) RS20050667A (el)
SI (1) SI1492761T1 (el)
TN (1) TNSN04186A1 (el)
TW (1) TWI225864B (el)
UA (2) UA80116C2 (el)
UY (1) UY27738A1 (el)
WO (1) WO2003082807A2 (el)
ZA (1) ZA200407536B (el)

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KR20070107147A (ko) * 2005-03-24 2007-11-06 파마시아 앤드 업존 캄파니 엘엘씨 알파-2-델타 단백질에 친화성을 갖는 광학적으로 순수한베타-아미노산의 제조
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