CY1108736T1 - Φαινυλ-και πυριδυλπιπεριδινο-παραγωγα ως ρυθμιστες μεταβολισμου γλυκοζης - Google Patents
Φαινυλ-και πυριδυλπιπεριδινο-παραγωγα ως ρυθμιστες μεταβολισμου γλυκοζηςInfo
- Publication number
- CY1108736T1 CY1108736T1 CY20091100109T CY091100109T CY1108736T1 CY 1108736 T1 CY1108736 T1 CY 1108736T1 CY 20091100109 T CY20091100109 T CY 20091100109T CY 091100109 T CY091100109 T CY 091100109T CY 1108736 T1 CY1108736 T1 CY 1108736T1
- Authority
- CY
- Cyprus
- Prior art keywords
- pyrydylpylperidin
- painyl
- producers
- regulators
- glucose
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Η παρούσα εφεύρεση αφορά ορισμένα υποκατεστημένα αρύλ και ετεροαρύλ παράγωγα όπως δείχνονται στο τύπο (la) που είναι ρυθμιστές μεταβολισμού. Συνεπώς, ενώσεις της παρούσας εφεύρεσης είναι χρήσιμες στη προφύλαξη ή τη θεραπεία μεταβολικών διαταραχών και επιπλοκών αυτών, όπως διαβήτη και παχυσαρκίας.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US44978803P | 2003-02-24 | 2003-02-24 | |
EP04713803A EP1606282B1 (en) | 2003-02-24 | 2004-02-23 | Phenyl- and pyridylpipereidinye-derivatives as modulators of glucose metabolism |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1108736T1 true CY1108736T1 (el) | 2014-04-09 |
Family
ID=32927568
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20091100109T CY1108736T1 (el) | 2003-02-24 | 2009-01-29 | Φαινυλ-και πυριδυλπιπεριδινο-παραγωγα ως ρυθμιστες μεταβολισμου γλυκοζης |
Country Status (20)
Country | Link |
---|---|
US (1) | US20070066590A1 (el) |
EP (1) | EP1606282B1 (el) |
JP (1) | JP2006518763A (el) |
KR (1) | KR20050106033A (el) |
CN (1) | CN1751038A (el) |
AT (1) | ATE414076T1 (el) |
AU (1) | AU2004215344B2 (el) |
BR (1) | BRPI0407620A (el) |
CA (1) | CA2515963A1 (el) |
CY (1) | CY1108736T1 (el) |
DE (1) | DE602004017703D1 (el) |
DK (1) | DK1606282T3 (el) |
EA (1) | EA200501348A1 (el) |
ES (1) | ES2316964T3 (el) |
HK (1) | HK1077305A1 (el) |
MX (1) | MXPA05007614A (el) |
PL (1) | PL378295A1 (el) |
PT (1) | PT1606282E (el) |
SI (1) | SI1606282T1 (el) |
WO (1) | WO2004076413A2 (el) |
Families Citing this family (106)
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-
2004
- 2004-02-23 EP EP04713803A patent/EP1606282B1/en not_active Expired - Lifetime
- 2004-02-23 DE DE602004017703T patent/DE602004017703D1/de not_active Expired - Lifetime
- 2004-02-23 BR BRPI0407620-6A patent/BRPI0407620A/pt not_active IP Right Cessation
- 2004-02-23 CA CA002515963A patent/CA2515963A1/en not_active Withdrawn
- 2004-02-23 PL PL378295A patent/PL378295A1/pl not_active Application Discontinuation
- 2004-02-23 AT AT04713803T patent/ATE414076T1/de active
- 2004-02-23 DK DK04713803T patent/DK1606282T3/da active
- 2004-02-23 ES ES04713803T patent/ES2316964T3/es not_active Expired - Lifetime
- 2004-02-23 AU AU2004215344A patent/AU2004215344B2/en not_active Ceased
- 2004-02-23 JP JP2006503856A patent/JP2006518763A/ja active Pending
- 2004-02-23 KR KR1020057015582A patent/KR20050106033A/ko not_active Application Discontinuation
- 2004-02-23 CN CNA2004800044127A patent/CN1751038A/zh active Pending
- 2004-02-23 MX MXPA05007614A patent/MXPA05007614A/es active IP Right Grant
- 2004-02-23 PT PT04713803T patent/PT1606282E/pt unknown
- 2004-02-23 SI SI200431030T patent/SI1606282T1/sl unknown
- 2004-02-23 WO PCT/US2004/005555 patent/WO2004076413A2/en active Application Filing
- 2004-02-23 US US10/546,665 patent/US20070066590A1/en not_active Abandoned
- 2004-02-23 EA EA200501348A patent/EA200501348A1/ru unknown
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2005
- 2005-12-28 HK HK05112041A patent/HK1077305A1/xx not_active IP Right Cessation
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2009
- 2009-01-29 CY CY20091100109T patent/CY1108736T1/el unknown
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DK1606282T3 (da) | 2009-03-16 |
WO2004076413A3 (en) | 2004-12-02 |
EA200501348A1 (ru) | 2006-02-24 |
CA2515963A1 (en) | 2004-09-10 |
WO2004076413A2 (en) | 2004-09-10 |
EP1606282A2 (en) | 2005-12-21 |
ATE414076T1 (de) | 2008-11-15 |
CN1751038A (zh) | 2006-03-22 |
HK1077305A1 (en) | 2006-02-10 |
BRPI0407620A (pt) | 2006-02-21 |
PT1606282E (pt) | 2009-02-10 |
SI1606282T1 (sl) | 2009-04-30 |
US20070066590A1 (en) | 2007-03-22 |
EP1606282B1 (en) | 2008-11-12 |
DE602004017703D1 (de) | 2008-12-24 |
AU2004215344A1 (en) | 2004-09-10 |
KR20050106033A (ko) | 2005-11-08 |
PL378295A1 (pl) | 2006-03-20 |
AU2004215344B2 (en) | 2010-06-24 |
ES2316964T3 (es) | 2009-04-16 |
MXPA05007614A (es) | 2006-05-25 |
JP2006518763A (ja) | 2006-08-17 |
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