CS253746B2 - Process for preparing new derivatives of pyrrolo /1,2-e//azepinone - Google Patents

Process for preparing new derivatives of pyrrolo /1,2-e//azepinone Download PDF

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Publication number
CS253746B2
CS253746B2 CS861697A CS169786A CS253746B2 CS 253746 B2 CS253746 B2 CS 253746B2 CS 861697 A CS861697 A CS 861697A CS 169786 A CS169786 A CS 169786A CS 253746 B2 CS253746 B2 CS 253746B2
Authority
CS
Czechoslovakia
Prior art keywords
solution
alkyl
piperazinyl
benzyl
optionally substituted
Prior art date
Application number
CS861697A
Other languages
Czech (cs)
English (en)
Inventor
Michel Barreau
Marie-Therese Comte
Daniel Farge
Jean-Luc Malleron
Gerard Ponsinet
Gerard Roussel
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Priority to CS865164A priority Critical patent/CS253750B2/cs
Publication of CS253746B2 publication Critical patent/CS253746B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS861697A 1985-03-15 1986-03-12 Process for preparing new derivatives of pyrrolo /1,2-e//azepinone CS253746B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS865164A CS253750B2 (cs) 1985-03-15 1986-07-08 Způsob výroby nových derivátů pyrrolo[1,2-a]azepinonu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8503840A FR2578842B1 (fr) 1985-03-15 1985-03-15 Nouveaux derives de la pyrrolo(1,2-a) azepinone, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
CS253746B2 true CS253746B2 (en) 1987-12-17

Family

ID=9317228

Family Applications (2)

Application Number Title Priority Date Filing Date
CS861697A CS253746B2 (en) 1985-03-15 1986-03-12 Process for preparing new derivatives of pyrrolo /1,2-e//azepinone
CS865164A CS253750B2 (cs) 1985-03-15 1986-07-08 Způsob výroby nových derivátů pyrrolo[1,2-a]azepinonu

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS865164A CS253750B2 (cs) 1985-03-15 1986-07-08 Způsob výroby nových derivátů pyrrolo[1,2-a]azepinonu

Country Status (23)

Country Link
US (2) US4769366A (de)
EP (1) EP0196955B1 (de)
JP (1) JPS61215392A (de)
KR (1) KR860007262A (de)
AT (1) ATE44032T1 (de)
AU (1) AU576064B2 (de)
CA (1) CA1261323A (de)
CS (2) CS253746B2 (de)
DD (1) DD251351A5 (de)
DE (1) DE3663948D1 (de)
DK (1) DK118886A (de)
ES (2) ES8801275A1 (de)
FI (2) FI861071A (de)
FR (1) FR2578842B1 (de)
GR (1) GR860672B (de)
HU (1) HU195510B (de)
IL (1) IL78135A (de)
MA (1) MA20638A1 (de)
NZ (1) NZ215471A (de)
PT (1) PT82182B (de)
SU (2) SU1447285A3 (de)
TN (1) TNSN86037A1 (de)
ZA (1) ZA861881B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL121432A (en) 1995-12-01 2000-09-28 Suntory Ltd Pyrrolo [3,2-C]azepine-4-one derivatives and pyrrolo [3,4-C]azepine-4-one derivatives their preparation and pharmaceutical compositions containing them

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1189553B (de) * 1962-08-09 1965-03-25 Degussa Verfahren zur Herstellung von racemischen und optisch aktiven Piperazinderivaten
DE2557341A1 (de) * 1975-12-19 1977-06-30 Hoechst Ag Basisch substituierte indolderivate und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
DK118886A (da) 1986-09-16
FI892181A0 (fi) 1989-05-05
US4826974A (en) 1989-05-02
CA1261323A (fr) 1989-09-26
ZA861881B (en) 1986-12-30
ES8800947A1 (es) 1987-12-01
IL78135A0 (en) 1986-07-31
PT82182B (fr) 1988-01-07
CS253750B2 (cs) 1987-12-17
HUT42773A (en) 1987-08-28
JPS61215392A (ja) 1986-09-25
TNSN86037A1 (fr) 1990-01-01
FI892181A (fi) 1989-05-05
AU576064B2 (en) 1988-08-11
MA20638A1 (fr) 1986-10-01
EP0196955B1 (de) 1989-06-14
GR860672B (en) 1986-05-27
SU1447285A3 (ru) 1988-12-23
US4769366A (en) 1988-09-06
NZ215471A (en) 1988-08-30
ES8801275A1 (es) 1987-12-16
ES553028A0 (es) 1987-12-16
DD251351A5 (de) 1987-11-11
FR2578842A1 (fr) 1986-09-19
IL78135A (en) 1989-02-28
KR860007262A (ko) 1986-10-10
AU5470186A (en) 1986-09-18
FI861071A0 (fi) 1986-03-14
DE3663948D1 (en) 1989-07-20
PT82182A (fr) 1986-04-01
ES556722A0 (es) 1987-12-01
DK118886D0 (da) 1986-03-14
FR2578842B1 (fr) 1987-04-10
ATE44032T1 (de) 1989-06-15
FI861071A (fi) 1986-09-16
SU1537139A3 (ru) 1990-01-15
HU195510B (en) 1988-05-30
EP0196955A1 (de) 1986-10-08

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