CS235309B2 - Method of 20-aminotylosine derivatives production - Google Patents

Method of 20-aminotylosine derivatives production Download PDF

Info

Publication number
CS235309B2
CS235309B2 CS831163A CS116383A CS235309B2 CS 235309 B2 CS235309 B2 CS 235309B2 CS 831163 A CS831163 A CS 831163A CS 116383 A CS116383 A CS 116383A CS 235309 B2 CS235309 B2 CS 235309B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
orbo
atoms
okupiou
compounds
Prior art date
Application number
CS831163A
Other languages
Czech (cs)
English (en)
Inventor
Satoshi Omura
Akira Nakagawa
Original Assignee
Satoshi Omura
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Satoshi Omura filed Critical Satoshi Omura
Priority to CS838673A priority Critical patent/CS235343B2/cs
Publication of CS235309B2 publication Critical patent/CS235309B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS831163A 1982-02-25 1983-02-21 Method of 20-aminotylosine derivatives production CS235309B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS838673A CS235343B2 (cs) 1982-02-25 1983-11-22 Způsob výroby derivátů 20-aminotylosinu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP57029480A JPS58146595A (ja) 1982-02-25 1982-02-25 マクロライド系抗生物質

Publications (1)

Publication Number Publication Date
CS235309B2 true CS235309B2 (en) 1985-05-15

Family

ID=12277244

Family Applications (1)

Application Number Title Priority Date Filing Date
CS831163A CS235309B2 (en) 1982-02-25 1983-02-21 Method of 20-aminotylosine derivatives production

Country Status (24)

Country Link
US (1) US4440759A (fr)
EP (1) EP0087921B1 (fr)
JP (1) JPS58146595A (fr)
KR (1) KR850000962B1 (fr)
AT (1) ATE16008T1 (fr)
AU (1) AU555979B2 (fr)
CA (1) CA1202022A (fr)
CS (1) CS235309B2 (fr)
DD (1) DD210283A5 (fr)
DE (1) DE3360951D1 (fr)
DK (1) DK153795C (fr)
ES (2) ES8403926A1 (fr)
FI (1) FI72322C (fr)
GB (1) GB2115813B (fr)
GR (1) GR78112B (fr)
HU (1) HU194269B (fr)
IL (1) IL67973A0 (fr)
NZ (1) NZ203365A (fr)
PH (1) PH18435A (fr)
PL (1) PL138759B1 (fr)
PT (1) PT76272B (fr)
RO (1) RO85833B (fr)
SU (1) SU1360588A3 (fr)
ZA (1) ZA831206B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820695A (en) * 1982-09-13 1989-04-11 Eli Lilly And Company C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics
IL69666A (en) * 1982-09-13 1987-10-20 Lilly Co Eli 20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
ZA841277B (en) * 1983-02-28 1985-09-25 Lilly Co Eli C-20-and c-23-modified macrolide derivatives
IL71032A0 (en) * 1983-02-28 1984-05-31 Lilly Co Eli C-20 and c-23-modified macrolide derivatives
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
US4801721A (en) * 1984-08-16 1989-01-31 Ryan James W Stereospecific synthesis of carboxyalkyl peptides
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW309505B (fr) * 1993-03-31 1997-07-01 Toto Ltd
WO1996009312A1 (fr) * 1994-09-22 1996-03-28 Pfizer Inc. Macrolides antibiotiques
EP0778283A3 (fr) * 1995-12-05 1998-01-28 Pfizer Inc. Macrolides antibiotiques
CN110590885A (zh) * 2019-09-30 2019-12-20 郑州大学 20-取代-5-o-碳霉胺糖基-泰乐内酯衍生物
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178341A (en) * 1960-06-27 1965-04-13 Lilly Co Eli Antibiotics tylosin and desmycosin and derivatives thereof
GB1587685A (en) * 1977-03-09 1981-04-08 Microbial Chem Res Found Macrolactone derivatives and their production
JPS53132584A (en) * 1977-04-26 1978-11-18 Toyo Jozo Co Ltd 18-cyano-18-substituted amino-18-deoxy-macrolide anibiotic substance derivative
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
US4279896A (en) * 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents

Also Published As

Publication number Publication date
AU555979B2 (en) 1986-10-16
ES520037A0 (es) 1984-04-01
US4440759A (en) 1984-04-03
DK153795B (da) 1988-09-05
RO85833B (ro) 1984-11-30
KR850000962B1 (ko) 1985-07-02
FI72322B (fi) 1987-01-30
DK153795C (da) 1989-01-23
FI830585L (fi) 1983-08-26
GB2115813A (en) 1983-09-14
DE3360951D1 (en) 1985-11-14
CA1202022A (fr) 1986-03-18
DK87783D0 (da) 1983-02-24
FI72322C (fi) 1987-05-11
AU1180183A (en) 1983-09-01
ZA831206B (en) 1983-11-30
PH18435A (en) 1985-07-08
GR78112B (fr) 1984-09-26
PL138759B1 (en) 1986-10-31
HU194269B (en) 1988-01-28
GB8305005D0 (en) 1983-03-30
ES8505207A1 (es) 1985-05-16
RO85833A (fr) 1984-11-25
ES526529A0 (es) 1985-05-16
EP0087921A1 (fr) 1983-09-07
DK87783A (da) 1983-08-26
SU1360588A3 (ru) 1987-12-15
ES8403926A1 (es) 1984-04-01
KR840003646A (ko) 1984-09-15
PT76272B (en) 1986-02-04
PT76272A (en) 1983-03-01
DD210283A5 (de) 1984-06-06
ATE16008T1 (de) 1985-10-15
GB2115813B (en) 1985-09-11
JPH0142277B2 (fr) 1989-09-11
JPS58146595A (ja) 1983-09-01
NZ203365A (en) 1985-07-12
FI830585A0 (fi) 1983-02-22
PL240735A1 (en) 1983-09-26
EP0087921B1 (fr) 1985-10-09
IL67973A0 (en) 1983-06-15

Similar Documents

Publication Publication Date Title
KR100486053B1 (ko) 신규에리트로마이신유도체,그의제조방법및약제로서의그의용도
US5444051A (en) Erythromycin compounds
US4474768A (en) N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
CS235309B2 (en) Method of 20-aminotylosine derivatives production
EP0001841B1 (fr) Dérivés de la tylosine
US5786339A (en) Erythromycins
EP0103465B1 (fr) 20-Amino-macrolides
EP1025114B1 (fr) Derives d'erythromycine cetolides, modifies en n-3' et substitues en o-6, possedant une activite antibacterienne
JP2001525331A (ja) ６−ｏ−アルキルエリスロマイシンｂオキシム
EP0124216B1 (fr) Dérivés de macrolides modifiés en C-20 et C-23
US5716939A (en) Amide derivatives of 16-membered ring antibiotic macrolides
CA1229336A (fr) Derives de macrolide modifies en c-20
EP1206476B1 (fr) 9a-azalides a activite antibacterienne
EP0316128B1 (fr) Dérivés à activité antibactérienne 9-déoxo-9a-allyl et propargyl-9a-aza-9a-homoérythromycine A
US4468511A (en) C-20- And C-23-Modified macrolide derivatives
US4629786A (en) C-20- and C-23 modified macrolide derivatives
US4820694A (en) Modifications of 3-O-demethylmycinose in macrocin and lactenocin
EP0099746B1 (fr) Dérivés d'antibiotiques macrolides modifiés en position C-23
EP1233971A2 (fr) Derives de ketolide substitues par 6-o-alkyl-2-nor-2-
JPS5931794A (ja) Ｎ―メチル１１―アザ―１０―デオキソ―１０―ジヒドロエリスロマイシンａ製造用中間体
CS235343B2 (cs) Způsob výroby derivátů 20-aminotylosinu
JPH0196190A (ja) ６−０−アルキル−エリスロマイシンａ　サイクリック１１，１２−カーボネート
MXPA00003644A (en) NOVEL 3,6-HEMIKETALS FROM THE CLASS OF 9a-AZALIDES